Affinity DataKi: 6.43E+3nMAssay Description:Antagonist activity at LPA1 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataIC50: <10nMAssay Description:Inhibition of LPA2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of LPA2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of LPA2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of LPA2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of LPA2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human LPA5 receptor by FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Antagonist activity at human LPA5 receptor assessed as inhibition of LPS-induced cAMP accumulation incubated for 20 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 95nMAssay Description:Antagonist activity at human LPA1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human LPA1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human LPA1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human LPA1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human LPA1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human LPA1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human LPA1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Antagonist activity at human LPA1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Antagonist activity at human LPA1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: <500nMAssay Description:Antagonist activity at LPA2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: <500nMAssay Description:Antagonist activity at LPA2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: <500nMAssay Description:Antagonist activity at LPA2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+3nMAssay Description:Antagonist activity at human LPA2 receptor assessed as inhibition of LPS-induced calcium releaseMore data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+3nMAssay Description:Antagonist activity at human LPA2 receptor assessed as inhibition of LPS-induced calcium releaseMore data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+3nMAssay Description:Antagonist activity at human LPA2 receptor assessed as inhibition of LPS-induced calcium releaseMore data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+3nMAssay Description:Antagonist activity at human LPA2 receptor assessed as inhibition of LPS-induced calcium releaseMore data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+3nMAssay Description:Antagonist activity at human LPA2 receptor assessed as inhibition of LPS-induced calcium releaseMore data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+3nMAssay Description:Antagonist activity at human LPA2 receptor assessed as inhibition of LPS-induced calcium releaseMore data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+3nMAssay Description:Antagonist activity at human LPA2 receptor assessed as inhibition of LPS-induced calcium releaseMore data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+3nMAssay Description:Antagonist activity at human LPA2 receptor assessed as inhibition of LPS-induced calcium releaseMore data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+3nMAssay Description:Antagonist activity at human LPA2 receptor assessed as inhibition of LPS-induced calcium releaseMore data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+3nMAssay Description:Antagonist activity at human LPA2 receptor assessed as inhibition of LPS-induced calcium releaseMore data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+3nMAssay Description:Antagonist activity at human LPA2 receptor assessed as inhibition of LPS-induced calcium releaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Antagonist activity at human LPA5 receptor by FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Antagonist activity at human LPA5 receptor by FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+3nMAssay Description:Antagonist activity at human LPA5 receptor expressed in CHO cells assessed as inhibition of LPA stimulated calcium release incubated for 20 mins foll...More data for this Ligand-Target Pair
Affinity DataEC50: <50nMAssay Description:Antagonist activity at human LPA3 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: <50nMAssay Description:Antagonist activity at human LPA3 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: <50nMAssay Description:Antagonist activity at human LPA1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: <50nMAssay Description:Antagonist activity at human LPA1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: <50nMAssay Description:Antagonist activity at human LPA1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: <50nMAssay Description:Antagonist activity at human LPA3 receptorMore data for this Ligand-Target Pair
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