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Found 129 with Last Name = 'logan' and Initial = 'j'
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031845((4-Biphenyl-4-yl-1-phosphono-butyl)-phosphonic aci...)
Affinity DataIC50:  0.700nMAssay Description:Inhibitory activity against rat liver microsomal squalene synthase was determined using [3H]-FPP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031845((4-Biphenyl-4-yl-1-phosphono-butyl)-phosphonic aci...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50049232(CHEMBL348349 | Tetrasodium salt of 4-(4'-Methyl-bi...)
Affinity DataIC50:  1nMAssay Description:Inhibitory activity against rat liver microsomal squalene synthase was determined using [3H]-FPP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031839(((E)-6,10-Dimethyl-1-phosphono-undeca-5,9-dienyl)-...)
Affinity DataIC50:  1nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50173389(CHEMBL198150 | N-Ethyl-2-(4-methanesulfonyl-phenyl...)
Affinity DataIC50:  1.70nMAssay Description:Displacement of [125I]-MIP-1 alpha from human C-C chemokine receptor type 5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50173388(CHEMBL197641 | N-Ethyl-2-(4-methanesulfonyl-phenyl...)
Affinity DataIC50:  2.30nMAssay Description:Displacement of [125I]-MIP-1 alpha from human C-C chemokine receptor type 5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031843(((E)-8,12-Dimethyl-1-phosphono-trideca-7,11-dienyl...)
Affinity DataIC50:  2.5nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031848(((E)-7,11-Dimethyl-1-phosphono-dodeca-6,10-dienyl)...)
Affinity DataIC50:  2.60nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031844(((E)-1-Hydroxyphosphinoyl-6,10-dimethyl-undeca-5,9...)
Affinity DataIC50:  4nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031851(((E)-10,14-Dimethyl-1-phosphono-pentadeca-9,13-die...)
Affinity DataIC50:  4.20nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031842(CHEMBL86867 | [(5E,9E)-1-(Hydroxy-hydroxymethyl-ph...)
Affinity DataIC50:  4.70nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031847(((5E,9E)-6,10,14-Trimethyl-1-phosphono-pentadeca-5...)
Affinity DataIC50:  5.70nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50049227(CHEMBL158707 | Trisodium salt of [1-(Dimethoxy-pho...)
Affinity DataIC50:  5.70nMAssay Description:Inhibitory activity against rat liver microsomal squalene synthase was determined using [3H]-FPP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50173383(CHEMBL199118 | N-Ethyl-2-(4-methanesulfonyl-phenyl...)
Affinity DataIC50:  5.90nMAssay Description:Displacement of [125I]-MIP-1 alpha from human C-C chemokine receptor type 5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50173398(CHEMBL371691 | N-Ethyl-2-(4-methanesulfonyl-phenyl...)
Affinity DataIC50:  6.30nMAssay Description:Displacement of [125I]-MIP-1 alpha from human C-C chemokine receptor type 5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031832(CHEMBL87922 | [(6E,10E)-1-(Hydroxy-methyl-phosphin...)
Affinity DataIC50:  6.5nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031859(CHEMBL314797 | [(5E,9E)-1-(Hydroxy-methoxymethyl-p...)
Affinity DataIC50:  6.5nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50173393(4-[3-(4-{Ethyl-[2-(4-methanesulfonyl-phenyl)-acety...)
Affinity DataIC50:  7.10nMAssay Description:Displacement of [125I]-MIP-1 alpha from human C-C chemokine receptor type 5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50173391(CHEMBL370826 | N-{1-[3-(4-Acetylamino-phenyl)-3-(3...)
Affinity DataIC50:  7.90nMAssay Description:Displacement of [125I]-MIP-1 alpha from human C-C chemokine receptor type 5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50173378(CHEMBL198277 | N-{1-[3-(4-Chloro-phenyl)-3-phenyl-...)
Affinity DataIC50:  8.5nMAssay Description:Displacement of [125I]-MIP-1 alpha from human C-C chemokine receptor type 5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031862(CHEMBL84629 | [(E)-1-(Hydroxy-methyl-phosphinoyl)-...)
Affinity DataIC50:  8.70nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50173382(CHEMBL373214 | N-Ethyl-N-{1-[3-(3-fluoro-phenyl)-3...)
Affinity DataIC50:  9.10nMAssay Description:Displacement of [125I]-MIP-1 alpha from human C-C chemokine receptor type 5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50173380(CHEMBL372733 | N-Ethyl-2-(4-methanesulfonyl-phenyl...)
Affinity DataIC50:  11nMAssay Description:Displacement of [125I]-MIP-1 alpha from human C-C chemokine receptor type 5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bos taurus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50126193(CHEMBL27660 | {4-[9-(2,2,2-Trifluoro-ethylcarbamoy...)
Affinity DataIC50:  11nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031836(((8E,12E)-9,13,17-Trimethyl-1-phosphono-octadeca-8...)
Affinity DataIC50:  11.8nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50173395(CHEMBL372134 | N-Ethyl-2-(4-methanesulfonyl-phenyl...)
Affinity DataIC50:  12nMAssay Description:Displacement of [125I]-MIP-1 alpha from human C-C chemokine receptor type 5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031849(CHEMBL86918 | [(5E,9E)-1-(Hydroxy-methyl-phosphino...)
Affinity DataIC50:  12.9nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50049217(CHEMBL158517 | Tripotassium salt of 1-Phosphono-4-...)
Affinity DataIC50:  13nMAssay Description:Inhibitory activity against rat liver microsomal squalene synthase was determined using [3H]-FPP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50157000(CHEMBL180155 | N-Allyl-N-[1-(3,3-diphenyl-propyl)-...)
Affinity DataIC50:  13nMAssay Description:Displacement of [125I]-MIP-1 alpha from human C-C chemokine receptor type 5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031837(CHEMBL87489 | [(E)-1-(Hydroxy-methoxymethyl-phosph...)
Affinity DataIC50:  13.1nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bos taurus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50126188(CHEMBL28348 | [4-(9-Propylcarbamoyl-9H-fluoren-9-y...)
Affinity DataIC50:  14nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031840(CHEMBL84961 | [4-Biphenyl-4-yl-1-(hydroxy-methoxym...)
Affinity DataIC50:  14.8nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50049233(CHEMBL160240 | Tripotassium salt of 4-Biphenyl-4-y...)
Affinity DataIC50:  15nMAssay Description:Inhibitory activity against rat liver microsomal squalene synthase was determined using [3H]-FPP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50049230(CHEMBL160267 | Tripotassium salt of 4-{3-[2-(4-Met...)
Affinity DataIC50:  17nMAssay Description:Inhibitory activity against rat liver microsomal squalene synthase was determined using [3H]-FPP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031854(((E)-9,13-Dimethyl-1-phosphono-tetradeca-8,12-dien...)
Affinity DataIC50:  17.6nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50049215(1-Phosphono-4-[3-(2-benzylphenoxy)phenyl]butylsulf...)
Affinity DataIC50:  18nMAssay Description:Inhibitory activity against rat liver microsomal squalene synthase was determined using [3H]-FPP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50173376(CHEMBL198114 | N-Ethyl-N-{1-[3-(4-methanesulfonyla...)
Affinity DataIC50:  18nMAssay Description:Displacement of [125I]-MIP-1 alpha from human C-C chemokine receptor type 5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50157032(CHEMBL369311 | N-[1-(3,3-Diphenyl-propyl)-piperidi...)
Affinity DataIC50:  18nMAssay Description:Displacement of [125I]-MIP-1 alpha from human C-C chemokine receptor type 5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50173386(CHEMBL370998 | N-{1-[3-(4-Chloro-phenyl)-3-(3-fluo...)
Affinity DataIC50:  19nMAssay Description:Displacement of [125I]-MIP-1 alpha from human C-C chemokine receptor type 5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50049228(CHEMBL158448 | Tripotassium salt of 4-{3-[2-(3-Met...)
Affinity DataIC50:  19nMAssay Description:Inhibitory activity against rat liver microsomal squalene synthase was determined using [3H]-FPP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bos taurus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50126207((4-{9-[2-(4-Methoxy-phenyl)-ethylcarbamoyl]-9H-flu...)
Affinity DataIC50:  21nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bos taurus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50126201(CHEMBL282785 | {4-[9-(2,2,2-Trifluoro-ethylcarbamo...)
Affinity DataIC50:  22nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50173397(CHEMBL370552 | N-{4-[3-(4-{Ethyl-[2-(4-methanesulf...)
Affinity DataIC50:  22nMAssay Description:Displacement of [125I]-MIP-1 alpha from human C-C chemokine receptor type 5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bos taurus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50126201(CHEMBL282785 | {4-[9-(2,2,2-Trifluoro-ethylcarbamo...)
Affinity DataIC50:  22nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50031855(CHEMBL86621 | [4-Biphenyl-4-yl-1-(hydroxy-hydroxym...)
Affinity DataIC50:  23.9nMAssay Description:Inhibition rat liver microsomal squalene synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bos taurus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50126209(CHEMBL283897 | {4-[9-(2,2,2-Trifluoro-ethylcarbamo...)
Affinity DataIC50:  24nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50173376(CHEMBL198114 | N-Ethyl-N-{1-[3-(4-methanesulfonyla...)
Affinity DataIC50:  24nMAssay Description:Inhibition of MIP-1beta stimulated calcium transients in CCR5-expressing CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bos taurus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50126225(CHEMBL26665 | {4-[9-(2,2,2-Trifluoro-ethylcarbamoy...)
Affinity DataIC50:  25nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50173374(CHEMBL198497 | N-{1-[3-(4-Acetylamino-phenyl)-3-ph...)
Affinity DataIC50:  26nMAssay Description:Displacement of [125I]-MIP-1 alpha from human C-C chemokine receptor type 5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bos taurus)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50126212(CHEMBL280283 | {4-[9-(2,2,2-Trifluoro-ethylcarbamo...)
Affinity DataIC50:  27nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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