TargetDelta-type opioid receptor(Homo sapiens (Human))
Memorial Sloan-Kettering Cancer Center
Curated by ChEMBL
Memorial Sloan-Kettering Cancer Center
Curated by ChEMBL
Affinity DataKi: 0.950nMAssay Description:Displacement of [125]IBNtxA from DOR-1 (unknown origin) transfected in CHO cells after 90 mins by competitive binding assayMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Memorial Sloan-Kettering Cancer Center
Curated by ChEMBL
Memorial Sloan-Kettering Cancer Center
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Displacement of [125]IBNtxA from DOR-1 (unknown origin) transfected in CHO cells after 90 mins by competitive binding assayMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Memorial Sloan-Kettering Cancer Center
Curated by ChEMBL
Memorial Sloan-Kettering Cancer Center
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Displacement of [125]IBNtxA from DOR-1 (unknown origin) transfected in CHO cells after 90 mins by competitive binding assayMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Memorial Sloan-Kettering Cancer Center
Curated by ChEMBL
Memorial Sloan-Kettering Cancer Center
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Displacement of [125]IBNtxA from KOR-1 (unknown origin) transfected in CHO cells after 90 mins by competitive binding assayMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Memorial Sloan-Kettering Cancer Center
Curated by ChEMBL
Memorial Sloan-Kettering Cancer Center
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Displacement of [125]IBNtxA from DOR-1 (unknown origin) transfected in CHO cells after 90 mins by competitive binding assayMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Memorial Sloan-Kettering Cancer Center
Curated by ChEMBL
Memorial Sloan-Kettering Cancer Center
Curated by ChEMBL
Affinity DataKi: 3.5nMAssay Description:Displacement of [125]IBNtxA from KOR-1 (unknown origin) transfected in CHO cells after 90 mins by competitive binding assayMore data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 6.20nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Memorial Sloan-Kettering Cancer Center
Curated by ChEMBL
Memorial Sloan-Kettering Cancer Center
Curated by ChEMBL
Affinity DataKi: 6.60nMAssay Description:Displacement of [125]IBNtxA from MOR-1 (unknown origin) transfected in CHO cells after 90 mins by competitive binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Memorial Sloan-Kettering Cancer Center
Curated by ChEMBL
Memorial Sloan-Kettering Cancer Center
Curated by ChEMBL
Affinity DataKi: 7.30nMAssay Description:Displacement of [125]IBNtxA from MOR-1 (unknown origin) transfected in CHO cells after 90 mins by competitive binding assayMore data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 8.20nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 8.30nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 8.5nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 9.10nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Memorial Sloan-Kettering Cancer Center
Curated by ChEMBL
Memorial Sloan-Kettering Cancer Center
Curated by ChEMBL
Affinity DataKi: 9.30nMAssay Description:Displacement of [125]IBNtxA from MOR-1 (unknown origin) transfected in CHO cells after 90 mins by competitive binding assayMore data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Memorial Sloan-Kettering Cancer Center
Curated by ChEMBL
Memorial Sloan-Kettering Cancer Center
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [125]IBNtxA from KOR-1 (unknown origin) transfected in CHO cells after 90 mins by competitive binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Memorial Sloan-Kettering Cancer Center
Curated by ChEMBL
Memorial Sloan-Kettering Cancer Center
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [125]IBNtxA from MOR-1 (unknown origin) transfected in CHO cells after 90 mins by competitive binding assayMore data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Memorial Sloan-Kettering Cancer Center
Curated by ChEMBL
Memorial Sloan-Kettering Cancer Center
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Displacement of [125]IBNtxA from KOR-1 (unknown origin) transfected in CHO cells after 90 mins by competitive binding assayMore data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 36nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 39nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 42nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 44nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 51nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 53nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataKi: 59nMAssay Description:Binding affinity to human recombinant mGlur2 assessed as inhibition constant by cAMP Glosensor assayMore data for this Ligand-Target Pair
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 59nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 59nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataKi: 59nMAssay Description:Binding affinity to human recombinant mGlur2 assessed as inhibition constant by cAMP Glosensor assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Binding affinity to human recombinant mGlur2 assessed as inhibition constant by cAMP Glosensor assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Binding affinity to human recombinant mGlur2 assessed as inhibition constant by cAMP Glosensor assayMore data for this Ligand-Target Pair