Compile Data Set for Download or QSAR
maximum 50k data
Found 156 with Last Name = 'matsumura' and Initial = 'ki'
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50596499(CHEMBL5185420)
Affinity DataEC50:  2.22E+3nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataEC50:  2.20E+3nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50596500(CHEMBL5180073)
Affinity DataEC50:  637nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50596501(CHEMBL5193666)
Affinity DataEC50:  955nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50596502(CHEMBL5180328)
Affinity DataEC50:  603nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50596503(CHEMBL5183133)
Affinity DataEC50:  3.60E+3nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50596499(CHEMBL5185420)
Affinity DataEC50:  2.58E+3nMAssay Description:Transactivation of Gal4-fused human PPARgamma expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataEC50:  4.40E+3nMAssay Description:Transactivation of Gal4-fused human PPARgamma expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50596500(CHEMBL5180073)
Affinity DataEC50:  542nMAssay Description:Transactivation of Gal4-fused human PPARgamma expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50596501(CHEMBL5193666)
Affinity DataEC50:  1.07E+3nMAssay Description:Transactivation of Gal4-fused human PPARgamma expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50596504(CHEMBL5178616)
Affinity DataEC50:  980nMAssay Description:Transactivation of Gal4-fused human PPARgamma expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50596502(CHEMBL5180328)
Affinity DataEC50:  987nMAssay Description:Transactivation of Gal4-fused human PPARgamma expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50596503(CHEMBL5183133)
Affinity DataEC50:  680nMAssay Description:Transactivation of Gal4-fused human PPARgamma expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50596499(CHEMBL5185420)
Affinity DataEC50:  263nMAssay Description:Transactivation of Gal4-fused human PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataEC50:  9.5nMAssay Description:Transactivation of Gal4-fused human PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50596500(CHEMBL5180073)
Affinity DataEC50:  16nMAssay Description:Transactivation of Gal4-fused human PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50596501(CHEMBL5193666)
Affinity DataEC50:  93nMAssay Description:Transactivation of Gal4-fused human PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50596504(CHEMBL5178616)
Affinity DataEC50:  110nMAssay Description:Transactivation of Gal4-fused human PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50596502(CHEMBL5180328)
Affinity DataEC50:  19nMAssay Description:Transactivation of Gal4-fused human PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50596503(CHEMBL5183133)
Affinity DataEC50:  120nMAssay Description:Transactivation of Gal4-fused human PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50596499(CHEMBL5185420)
Affinity DataEC50:  1.06E+3nMAssay Description:Transactivation of Gal4-fused mouse PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Shionogi

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataEC50:  76nMAssay Description:Transactivation of Gal4-fused mouse PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50596500(CHEMBL5180073)
Affinity DataEC50:  71nMAssay Description:Transactivation of Gal4-fused mouse PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50596501(CHEMBL5193666)
Affinity DataEC50:  151nMAssay Description:Transactivation of Gal4-fused mouse PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50596504(CHEMBL5178616)
Affinity DataEC50:  830nMAssay Description:Transactivation of Gal4-fused mouse PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50596502(CHEMBL5180328)
Affinity DataEC50:  49nMAssay Description:Transactivation of Gal4-fused mouse PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50596503(CHEMBL5183133)
Affinity DataEC50:  330nMAssay Description:Transactivation of Gal4-fused mouse PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at human PPAR-alpha assessed as receptor transactivation by measuring maximum induction of alkaline phosphatase activityMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human PPAR-delta assessed as receptor transactivation by measuring maximum induction of alkaline phosphatase activityMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataEC50:  850nMAssay Description:Agonist activity at human PPAR-gamma assessed as receptor transactivation by measuring maximum induction of alkaline phosphatase activityMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50596500(CHEMBL5180073)
Affinity DataEC50:  16nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50615945(CHEMBL5267326)
Affinity DataEC50:  33nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50615946(CHEMBL5271479)
Affinity DataEC50:  5.40nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50615947(CHEMBL5278892)
Affinity DataEC50:  5nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50615948(CHEMBL5281528)
Affinity DataEC50:  16nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50615949(CHEMBL5278648)
Affinity DataEC50:  19nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50615950(CHEMBL5288454)
Affinity DataEC50:  7.90nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50615951(CHEMBL5285352)
Affinity DataEC50:  17nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50615952(CHEMBL5267473)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50615953(CHEMBL5271300)
Affinity DataEC50:  17nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50615954(CHEMBL5290870)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50615955(CHEMBL5283926)
Affinity DataEC50:  3.60nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataEC50:  9.5nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50615956(CHEMBL5272924)
Affinity DataEC50:  21nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50615957(CHEMBL5268646)
Affinity DataEC50:  9.90nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50615958(CHEMBL5279586)
Affinity DataEC50:  6.90nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50615959(CHEMBL5273427)
Affinity DataEC50:  10nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50615960(CHEMBL5289017)
Affinity DataEC50:  6.20nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50615961(CHEMBL5268424)
Affinity DataEC50:  6.20nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50615962(CHEMBL5272996)
Affinity DataEC50:  3.10nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
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