TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 2.22E+3nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 2.20E+3nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 637nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 955nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 603nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 3.60E+3nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 2.58E+3nMAssay Description:Transactivation of Gal4-fused human PPARgamma expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 4.40E+3nMAssay Description:Transactivation of Gal4-fused human PPARgamma expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 542nMAssay Description:Transactivation of Gal4-fused human PPARgamma expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 1.07E+3nMAssay Description:Transactivation of Gal4-fused human PPARgamma expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 980nMAssay Description:Transactivation of Gal4-fused human PPARgamma expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 987nMAssay Description:Transactivation of Gal4-fused human PPARgamma expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 680nMAssay Description:Transactivation of Gal4-fused human PPARgamma expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 263nMAssay Description:Transactivation of Gal4-fused human PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 9.5nMAssay Description:Transactivation of Gal4-fused human PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 16nMAssay Description:Transactivation of Gal4-fused human PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 93nMAssay Description:Transactivation of Gal4-fused human PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 110nMAssay Description:Transactivation of Gal4-fused human PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 19nMAssay Description:Transactivation of Gal4-fused human PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Transactivation of Gal4-fused human PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Affinity DataEC50: 1.06E+3nMAssay Description:Transactivation of Gal4-fused mouse PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Affinity DataEC50: 76nMAssay Description:Transactivation of Gal4-fused mouse PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Affinity DataEC50: 71nMAssay Description:Transactivation of Gal4-fused mouse PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Affinity DataEC50: 151nMAssay Description:Transactivation of Gal4-fused mouse PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Affinity DataEC50: 830nMAssay Description:Transactivation of Gal4-fused mouse PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Affinity DataEC50: 49nMAssay Description:Transactivation of Gal4-fused mouse PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Affinity DataEC50: 330nMAssay Description:Transactivation of Gal4-fused mouse PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 1.10E+3nMAssay Description:Agonist activity at human PPAR-alpha assessed as receptor transactivation by measuring maximum induction of alkaline phosphatase activityMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 1nMAssay Description:Agonist activity at human PPAR-delta assessed as receptor transactivation by measuring maximum induction of alkaline phosphatase activityMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 850nMAssay Description:Agonist activity at human PPAR-gamma assessed as receptor transactivation by measuring maximum induction of alkaline phosphatase activityMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 16nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 33nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 5.40nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 5nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 16nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 19nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 7.90nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 17nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 2.70nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 17nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 1.5nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 3.60nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 9.5nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 21nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 9.90nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 6.90nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 10nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 6.20nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 6.20nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Shionogi
Curated by ChEMBL
Shionogi
Curated by ChEMBL
Affinity DataEC50: 3.10nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair