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Found 262 with Last Name = 'gao' and Initial = 'lj'
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50076089((3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[2-((R)-1-methy...)
Affinity DataKi:  10nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50076089((3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[2-((R)-1-methy...)
Affinity DataKi:  10nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50076089((3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[2-((R)-1-methy...)
Affinity DataKi:  11nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50076089((3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[2-((R)-1-methy...)
Affinity DataKi:  11nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50076089((3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[2-((R)-1-methy...)
Affinity DataKi:  93nMAssay Description:Binding affinity against human muscarine receptor (hM3) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50076089((3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[2-((R)-1-methy...)
Affinity DataKi:  93.3nMAssay Description:Binding affinity against human muscarine receptor (hM3) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219978(CHEMBL301670)
Affinity DataKi:  95nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50076089((3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[2-((R)-1-methy...)
Affinity DataKi:  107nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50076089((3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[2-((R)-1-methy...)
Affinity DataKi:  107nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219977(CHEMBL57485)
Affinity DataKi:  170nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219978(CHEMBL301670)
Affinity DataKi:  174nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219972(CHEMBL294663)
Affinity DataKi:  309nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424331(CHEMBL2314497)
Affinity DataKi:  390nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219978(CHEMBL301670)
Affinity DataKi:  427nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50304501(6-(4-Methylpiperazin-1-yl)pyrimidine-2,4-diamine |...)
Affinity DataKi:  530nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50273541(CHEMBL516312 | N-(5-(4-cyanophenyl)-1H-pyrrolo[2,3...)
Affinity DataKi:  541nMAssay Description:Binding affinity to biotinylated AAK1 (unknown origin) incubated for 1.5 hrs by fluorescent tracer dependent TR-FRET based binding displacement assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219977(CHEMBL57485)
Affinity DataKi:  617nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219974(CHEMBL56275)
Affinity DataKi:  676nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219974(CHEMBL56275)
Affinity DataKi:  676nMAssay Description:Binding affinity against human muscarine receptor (hM3) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219979(CHEMBL58824)
Affinity DataKi:  794nMAssay Description:Binding affinity against human muscarine receptor (hM3) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219979(CHEMBL58824)
Affinity DataKi:  794nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219979(CHEMBL58824)
Affinity DataKi:  851nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219976(CHEMBL55698)
Affinity DataKi:  891nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219972(CHEMBL294663)
Affinity DataKi:  891nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424324(CHEMBL2314761)
Affinity DataKi:  980nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219974(CHEMBL56275)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50304501(6-(4-Methylpiperazin-1-yl)pyrimidine-2,4-diamine |...)
Affinity DataKi:  1.08E+3nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from human histamine H3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219973(CHEMBL291562)
Affinity DataKi:  1.15E+3nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219975(CHEMBL430587)
Affinity DataKi:  1.18E+3nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424327(CHEMBL2314501)
Affinity DataKi:  1.41E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424340(CHEMBL2314772)
Affinity DataKi:  1.41E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219976(CHEMBL55698)
Affinity DataKi:  1.51E+3nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219978(CHEMBL301670)
Affinity DataKi:  1.62E+3nMAssay Description:Binding affinity against human muscarine receptor (hM3) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424325(CHEMBL2314760)
Affinity DataKi:  1.71E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219976(CHEMBL55698)
Affinity DataKi:  1.74E+3nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219977(CHEMBL57485)
Affinity DataKi:  1.74E+3nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219973(CHEMBL291562)
Affinity DataKi:  1.74E+3nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50273541(CHEMBL516312 | N-(5-(4-cyanophenyl)-1H-pyrrolo[2,3...)
Affinity DataKi:  1.75E+3nMAssay Description:Binding affinity to biotinylated GAK (unknown origin) incubated for 1.5 hrs by fluorescent tracer dependent TR-FRET based binding displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219976(CHEMBL55698)
Affinity DataKi:  1.95E+3nMAssay Description:Binding affinity against human muscarine receptor (hM3) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219975(CHEMBL430587)
Affinity DataKi:  1.95E+3nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219977(CHEMBL57485)
Affinity DataKi:  2.09E+3nMAssay Description:Binding affinity against human muscarine receptor (hM3) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219974(CHEMBL56275)
Affinity DataKi:  2.34E+3nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219979(CHEMBL58824)
Affinity DataKi:  2.57E+3nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424338(CHEMBL2314774)
Affinity DataKi:  2.64E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424341(CHEMBL2314771)
Affinity DataKi:  2.67E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424326(CHEMBL2314759)
Affinity DataKi:  2.93E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219975(CHEMBL430587)
Affinity DataKi:  3.24E+3nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219972(CHEMBL294663)
Affinity DataKi:  3.24E+3nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424337(CHEMBL2314775)
Affinity DataKi:  3.28E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50219972(CHEMBL294663)
Affinity DataKi:  3.31E+3nMAssay Description:Binding affinity against human muscarine receptor (hM3) cloned in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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