Affinity DataKi: 10nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 93nMAssay Description:Binding affinity against human muscarine receptor (hM3) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 93.3nMAssay Description:Binding affinity against human muscarine receptor (hM3) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 95nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 107nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 107nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 174nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 309nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
Affinity DataKi: 427nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 530nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
Affinity DataKi: 541nMAssay Description:Binding affinity to biotinylated AAK1 (unknown origin) incubated for 1.5 hrs by fluorescent tracer dependent TR-FRET based binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 617nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 676nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 676nMAssay Description:Binding affinity against human muscarine receptor (hM3) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 794nMAssay Description:Binding affinity against human muscarine receptor (hM3) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 794nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 851nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 891nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 891nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 980nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.08E+3nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from human histamine H3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.15E+3nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.18E+3nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.41E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
Affinity DataKi: 1.41E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
Affinity DataKi: 1.51E+3nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.62E+3nMAssay Description:Binding affinity against human muscarine receptor (hM3) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.71E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
Affinity DataKi: 1.74E+3nMAssay Description:Binding affinity against human muscarine receptor (hM2) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.74E+3nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.74E+3nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.75E+3nMAssay Description:Binding affinity to biotinylated GAK (unknown origin) incubated for 1.5 hrs by fluorescent tracer dependent TR-FRET based binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.95E+3nMAssay Description:Binding affinity against human muscarine receptor (hM3) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.95E+3nMAssay Description:Binding affinity against human muscarine receptor (hM4) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.09E+3nMAssay Description:Binding affinity against human muscarine receptor (hM3) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.34E+3nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.57E+3nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.64E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
Affinity DataKi: 2.67E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
Affinity DataKi: 2.93E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
Affinity DataKi: 3.24E+3nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.24E+3nMAssay Description:Binding affinity against human muscarine receptor (hM1) cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.28E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
Affinity DataKi: 3.31E+3nMAssay Description:Binding affinity against human muscarine receptor (hM3) cloned in CHO cellsMore data for this Ligand-Target Pair