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LigandPNGBDBM50413752(CHEMBL2012519 | L-783277)
Affinity DataIC50:  2nMAssay Description:Inhibition of VEGFR2 by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136890(CHEMBL152208 | [2-Chloro-4-(4-fluoro-2-methyl-phen...)
Affinity DataIC50:  4nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136887(CHEMBL356455 | [4-(2-Amino-phenylamino)-2-chloro-p...)
Affinity DataIC50:  5nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50:  5.80nMAssay Description:Inhibition of VEGFR2 by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136897((2-Chloro-4-phenylamino-phenyl)-o-tolyl-methanone ...)
Affinity DataIC50:  7nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136886(CHEMBL152767 | [4-(2-Amino-phenylamino)-2-chloro-p...)
Affinity DataIC50:  10nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136884((2-Chloro-4-o-tolylamino-phenyl)-o-tolyl-methanone...)
Affinity DataIC50:  12nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136898(CHEMBL152820 | [4-(2-Amino-phenylamino)-2-methyl-p...)
Affinity DataIC50:  13nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50413752(CHEMBL2012519 | L-783277)
Affinity DataIC50:  15nMAssay Description:Inhibition of MEK2 by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136900(1-{2-[3-Chloro-4-(2-methyl-benzoyl)-phenylamino]-p...)
Affinity DataIC50:  21nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM15244(5-(2,6-dichlorophenyl)-2-(2,4-difluorophenyl)sulfa...)
Affinity DataIC50:  29nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136903(CHEMBL357732 | [4-(2-Amino-phenylamino)-phenyl]-o-...)
Affinity DataIC50:  29nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50099331(4-(4-(4-fluorophenyl)-1-(piperidin-4-yl)-1H-imidaz...)
Affinity DataIC50:  38nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136885(CHEMBL347496 | [4-(2-Amino-4-bromo-phenylamino)-2-...)
Affinity DataIC50:  39nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136888(CHEMBL153012 | {2-[3-Chloro-4-(2-methyl-benzoyl)-p...)
Affinity DataIC50:  42nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136899(CHEMBL152440 | [4-(2-Amino-phenylamino)-phenyl]-(2...)
Affinity DataIC50:  54nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50413752(CHEMBL2012519 | L-783277)
Affinity DataIC50:  57nMAssay Description:Inhibition of VEGFR2 autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136901(CHEMBL422510 | N-{2-[3-Chloro-4-(2-methyl-benzoyl)...)
Affinity DataIC50:  63nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136895(CHEMBL347770 | {4-[(2-Amino-phenyl)-methyl-amino]-...)
Affinity DataIC50:  101nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136902(CHEMBL155448 | [4-(2-Amino-phenylamino)-2-chloro-p...)
Affinity DataIC50:  139nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136896(CHEMBL356157 | [4-(2-Amino-phenylamino)-3-methyl-p...)
Affinity DataIC50:  143nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136882(CHEMBL152596 | [4-(2-Amino-phenylamino)-phenyl]-ph...)
Affinity DataIC50:  145nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50:  150nMAssay Description:Inhibition of MNK2 by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50335376((S)-16-hydroxy-14-methoxy-3-methyl-3,4,9,10,11,12-...)
Affinity DataIC50:  170nMAssay Description:Inhibition of VEGFR2 by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50:  190nMAssay Description:Inhibition of VEGFR2 by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136891(CHEMBL152349 | Phenyl-(4-phenylamino-phenyl)-metha...)
Affinity DataIC50:  193nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50413752(CHEMBL2012519 | L-783277)
Affinity DataIC50:  303nMAssay Description:Inhibition of cKIT by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136883(CHEMBL347576 | [2-Chloro-4-(2-nitro-phenylamino)-p...)
Affinity DataIC50:  437nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136893(CHEMBL152209 | [4-(2-Amino-phenylamino)-phenyl]-m-...)
Affinity DataIC50:  574nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50413752(CHEMBL2012519 | L-783277)
Affinity DataIC50:  640nMAssay Description:Inhibition of MK5 by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50:  673nMAssay Description:Inhibition of cKIT by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50413752(CHEMBL2012519 | L-783277)
Affinity DataIC50:  763nMAssay Description:Inhibition of ALK by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50:  763nMAssay Description:Inhibition of ALK by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136892(CHEMBL356809 | [4-(2-Amino-phenylamino)-phenyl]-bi...)
Affinity DataIC50:  811nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50413752(CHEMBL2012519 | L-783277)
Affinity DataIC50:  950nMAssay Description:Inhibition of ERK2 by Caliper mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136889(CHEMBL152403 | N-[3-Chloro-4-(1-o-tolyl-vinyl)-phe...)
Affinity DataIC50:  1.55E+3nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50335376((S)-16-hydroxy-14-methoxy-3-methyl-3,4,9,10,11,12-...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of ALK by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50413752(CHEMBL2012519 | L-783277)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of TYK2 by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of TYK2 by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of LCK by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50413752(CHEMBL2012519 | L-783277)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibition of LCK by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibition of ERK2 by Caliper mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50335376((S)-16-hydroxy-14-methoxy-3-methyl-3,4,9,10,11,12-...)
Affinity DataIC50:  6.84E+3nMAssay Description:Inhibition of MEK2 by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of RET by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibition of EPHB4 by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of cKIT by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of LCK by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50335374((3S,9S)-9,16-dihydroxy-14-methoxy-3-methyl-3,4,9,1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of TYK2 by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Human)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50413752(CHEMBL2012519 | L-783277)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of p38alpha by Caliper mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50413752(CHEMBL2012519 | L-783277)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK2A by Caliper mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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