Affinity DataKi: 0.700nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Binding affinity to mu opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]DAMGO from human recombinant opioid mu receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting meth...More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]-DAMGO from human mu opioid receptor expressed in CHO cells membrane after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by ChEMBL
National Institute On Drug Abuse
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]U69,593 from human recombinant opioid kappa receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by ChEMBL
National Institute On Drug Abuse
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]U69,593 from human recombinant opioid kappa receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Displacement of [3H]DAMGO from human recombinant opioid mu receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting meth...More data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Displacement of [3H]-DAMGO from human mu opioid receptor expressed in CHO cells membrane after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Displacement of [3H]DAMGO from human recombinant opioid mu receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting meth...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by ChEMBL
National Institute On Drug Abuse
Curated by ChEMBL
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]U69,593 from human recombinant kappa opioid receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by ChEMBL
National Institute On Drug Abuse
Curated by ChEMBL
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]-U69593 from human kappa opioid receptor expressed in CHO cells membrane after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by ChEMBL
National Institute On Drug Abuse
Curated by ChEMBL
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]U69,593 from human recombinant opioid kappa receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by ChEMBL
National Institute On Drug Abuse
Curated by ChEMBL
Affinity DataKi: 3.70nMAssay Description:Displacement of [3H]U69,593 from human recombinant opioid kappa receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Displacement of [3H]DAMGO from human recombinant opioid mu receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting meth...More data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Displacement of [3H]DAMGO from human recombinant opioid mu receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting meth...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity to mu opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Displacement of [3H]DAMGO from human recombinant opioid mu receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting meth...More data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Displacement of [3H]-DAMGO from human mu opioid receptor expressed in CHO cells membrane after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mus musculus (Mouse))
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by ChEMBL
National Institute On Drug Abuse
Curated by ChEMBL
Affinity DataKi: 5.10nMAssay Description:Displacement of [3H]U69,593 from human recombinant opioid kappa receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataKi: 5.5nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataKi: 5.5nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by ChEMBL
National Institute On Drug Abuse
Curated by ChEMBL
Affinity DataKi: 5.5nMAssay Description:Displacement of [3H]DADLE from human recombinant opioid delta receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting m...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataKi: 5.5nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Displacement of [3H]DAMGO from human recombinant opioid mu receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting meth...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mus musculus (Mouse))
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataKi: 5.70nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 5.80nMAssay Description:Displacement of [3H]DAMGO from human recombinant opioid mu receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting meth...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataKi: 5.90nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataKi: 6.40nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by ChEMBL
National Institute On Drug Abuse
Curated by ChEMBL
Affinity DataKi: 6.90nMAssay Description:Displacement of [3H]DADLE from human recombinant opioid delta receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting m...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mus musculus (Mouse))
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by ChEMBL
National Institute On Drug Abuse
Curated by ChEMBL
Affinity DataKi: 7.10nMAssay Description:Displacement of [3H]DADLE from human recombinant opioid delta receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting m...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse
Curated by ChEMBL
National Institute On Drug Abuse
Curated by ChEMBL
Affinity DataKi: 7.30nMAssay Description:Displacement of [3H]DADLE from human recombinant opioid delta receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting m...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataKi: 7.40nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair