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Found 111 with Last Name = 'khair' and Initial = 'nz'
LigandPNGBDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataKi:  1nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM370121(6-(difluoromethyl)-8-[(1R,2R)-2-hydroxy-2-methylcy...)
Affinity DataKi:  1nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50611455(CHEMBL5286090)
Affinity DataKi:  1nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50611459(CHEMBL5277565)
Affinity DataKi:  2nMAssay Description:Inhibition of CDK5/p25 (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff equat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50431360(CHEMBL2347597)
Affinity DataKi:  3nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff ...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50431360(CHEMBL2347597)
Affinity DataKi:  3nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataKi:  3nMAssay Description:Inhibition of CDK1/Cyclin B (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50431360(CHEMBL2347597)
Affinity DataKi:  4nMAssay Description:Inhibition of CDK1/Cyclin B (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50431360(CHEMBL2347597)
Affinity DataKi:  4nMAssay Description:Inhibition of CDK1/Cyclin B (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff ...More data for this Ligand-Target Pair
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LigandPNGBDBM50431360(CHEMBL2347597)
Affinity DataKi:  4nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff...More data for this Ligand-Target Pair
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LigandPNGBDBM50431360(CHEMBL2347597)
Affinity DataKi:  4nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50611454(CHEMBL5277074)
Affinity DataKi:  5nMAssay Description:Inhibition of CDK1/Cyclin B (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50611455(CHEMBL5286090)
Affinity DataKi:  5nMAssay Description:Inhibition of CDK1/Cyclin B (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50611451(CHEMBL5286978)
Affinity DataKi:  5nMAssay Description:Inhibition of CDK1/Cyclin B (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50593923(CHEMBL5195030)
Affinity DataKi:  5nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50611456(CHEMBL5281179)
Affinity DataKi:  6nMAssay Description:Inhibition of CDK1/Cyclin B (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff ...More data for this Ligand-Target Pair
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LigandPNGBDBM50611452(CHEMBL5286271)
Affinity DataKi:  6nMAssay Description:Inhibition of CDK1/Cyclin B (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50611456(CHEMBL5281179)
Affinity DataKi:  7nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50611457(CHEMBL5285230)
Affinity DataKi:  8nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50611457(CHEMBL5285230)
Affinity DataKi:  9nMAssay Description:Inhibition of CDK5/p25 (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff equat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50611459(CHEMBL5277565)
Affinity DataKi:  12nMAssay Description:Inhibition of CDK1/Cyclin B (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50611459(CHEMBL5277565)
Affinity DataKi:  16nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50611455(CHEMBL5286090)
Affinity DataKi:  17nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50611458(CHEMBL5286293)
Affinity DataKi:  18nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50611452(CHEMBL5286271)
Affinity DataKi:  19nMAssay Description:Inhibition of CDK5/p25 (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff equat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50611452(CHEMBL5286271)
Affinity DataKi:  21nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50611451(CHEMBL5286978)
Affinity DataKi:  23nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50611457(CHEMBL5285230)
Affinity DataKi:  26nMAssay Description:Inhibition of CDK1/Cyclin B (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50611451(CHEMBL5286978)
Affinity DataKi:  26nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50611455(CHEMBL5286090)
Affinity DataKi:  33nMAssay Description:Inhibition of CDK5/p25 (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff equat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50611458(CHEMBL5286293)
Affinity DataKi:  36nMAssay Description:Inhibition of CDK5/p25 (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff equat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50611456(CHEMBL5281179)
Affinity DataKi:  36nMAssay Description:Inhibition of CDK5/p25 (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff equat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50611453(CHEMBL5270069)
Affinity DataKi:  42nMAssay Description:Inhibition of CDK5/p25 (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff equat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50113281(AT-7519)
Affinity DataKi:  47nMAssay Description:Inhibition of CDK2/cyclin A (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
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LigandPNGBDBM50611460(CHEMBL5277367)
Affinity DataKi:  70nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50611451(CHEMBL5286978)
Affinity DataKi:  77nMAssay Description:Inhibition of CDK5/p25 (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff equat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50611461(CHEMBL5273574)
Affinity DataKi:  87nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50611454(CHEMBL5277074)
Affinity DataKi:  92nMAssay Description:Inhibition of CDK5/p25 (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff equat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50611458(CHEMBL5286293)
Affinity DataKi:  99nMAssay Description:Inhibition of CDK1/Cyclin B (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50611453(CHEMBL5270069)
Affinity DataKi:  146nMAssay Description:Inhibition of CDK1/Cyclin B (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50611461(CHEMBL5273574)
Affinity DataKi:  147nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University Of South Australia

Curated by ChEMBL
LigandPNGBDBM50525155(CHEMBL4561424)
Affinity DataKi:  160nMAssay Description:Inhibition of recombinant full length N-terminal GST tagged human CDK5/p25 expressed in baculovirus infected sf9 cells using histone H1 as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50611462(CHEMBL5287252)
Affinity DataKi:  171nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50611454(CHEMBL5277074)
Affinity DataKi:  176nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50113281(AT-7519)
Affinity DataKi:  190nMAssay Description:Inhibition of CDK1/Cyclin B (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50611456(CHEMBL5281179)
Affinity DataKi:  229nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
University Of South Australia

Curated by ChEMBL
LigandPNGBDBM50525155(CHEMBL4561424)
Affinity DataKi:  270nMAssay Description:Inhibition of recombinant full length N-terminal GST tagged human CDK2/CyclinA expressed in baculovirus infected sf9 cells using histone H1 as substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50611452(CHEMBL5286271)
Affinity DataKi:  271nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50611454(CHEMBL5277074)
Affinity DataKi:  301nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) assessed as inhibition constant incubated for 30 to 60 mins presence of dithiothreitol by Cheng-Prusoff...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50593923(CHEMBL5195030)
Affinity DataKi:  578nMAssay Description:Inhibition of CDK1/Cyclin B (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
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