Affinity DataKi: 4.30nMAssay Description:Displacement of [3H]-CP-55940 from rat CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 8.20nMAssay Description:Displacement of [3H]-CP-55940 from rat CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 8.60nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 9.20nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]-CP-55940 from rat CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]-CP-55940 from rat CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]-CP-55,940 from rat CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]-CP-55940 from rat CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Displacement of [3H]-CP-55,940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of [3H]-CP-55940 from rat CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [3H]-CP-55940 from rat CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Displacement of [3H]-CP-55,940 from rat CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Displacement of [3H]-CP-55940 from rat CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Binding affinity to rat CB2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Displacement of [3H]-CP-55940 from rat CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Displacement of [3H]-CP-55940 from rat CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Displacement of [3H]-CP-55940 from rat CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Displacement of [3H]-CP-55940 from rat CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Displacement of [3H]-CP-55940 from rat CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Displacement of [3H]-CP-55,940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Displacement of [3H]-CP-55940 from rat CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 82nMAssay Description:Displacement of [3H]-CP-55,940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 84nMAssay Description:Displacement of [3H]-CP-55,940 from rat CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 84nMAssay Description:Displacement of [3H]-CP-55940 from rat CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 87nMAssay Description:Displacement of [3H]-CP-55940 from rat CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 87nMAssay Description:Displacement of [3H]-CP-55940 from rat CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 104nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 459nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 459nMAssay Description:Displacement of [3H]-CP-55940 from rat CB2 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Lilly Research Laboratories
Curated by ChEMBL
Lilly Research Laboratories
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human ERGMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:In vitro inhibition of Acyl coenzyme A:cholesterol acyltransferase 1 from rat liver.More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat A10 cell Endothelin A receptor.More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat A10 cell Endothelin A receptor.More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair