Affinity DataKi: 82nMAssay Description:Competitive inhibition of Trypanosoma cruzi cruzaine expressed in Escherichia coli SG13009 using Z-FR-AMC as substrate by Lineweaver-Burk plot analys...More data for this Ligand-Target Pair
TargetThioredoxin reductase(Plasmodium falciparum (isolate 3D7))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Binding affinity to Plasmodium falciparum TrxR in presence of NADPHMore data for this Ligand-Target Pair
TargetThioredoxin reductase(Plasmodium falciparum (isolate 3D7))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Binding affinity to Plasmodium falciparum TrxR in presence of thioredoxinMore data for this Ligand-Target Pair
TargetThioredoxin reductase(Plasmodium falciparum (isolate 3D7))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataKi: 650nMAssay Description:Binding affinity to Plasmodium falciparum TrxR in presence of thioredoxinMore data for this Ligand-Target Pair
TargetThioredoxin reductase(Plasmodium falciparum (isolate 3D7))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Binding affinity to Plasmodium falciparum TrxR in presence of NADPHMore data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine expressed in Escherichia coli SG13009 using Z-FR-AMC as substrate after 5 minsMore data for this Ligand-Target Pair
TargetThioredoxin reductase(Plasmodium falciparum (isolate 3D7))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of Plasmodium falciparum TrxRMore data for this Ligand-Target Pair
Affinity DataIC50: 540nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine expressed in Escherichia coli SG13009 using Z-FR-AMC as substrate after 5 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine expressed in Escherichia coli SG13009 using Z-FR-AMC as substrate after 5 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 620nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine expressed in Escherichia coli SG13009 using Z-FR-AMC as substrate after 5 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine expressed in Escherichia coli SG13009 using Z-FR-AMC as substrate after 5 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine expressed in Escherichia coli SG13009 using Z-FR-AMC as substrate after 5 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine expressed in Escherichia coli SG13009 using Z-FR-AMC as substrate after 5 minsMore data for this Ligand-Target Pair
TargetThioredoxin reductase(Plasmodium falciparum (isolate 3D7))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Plasmodium falciparum TrxRMore data for this Ligand-Target Pair
TargetThioredoxin reductase 1, cytoplasmic/2, mitochondrial/3(Homo sapiens (Human))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human TrxRMore data for this Ligand-Target Pair
TargetThioredoxin reductase(Plasmodium falciparum (isolate 3D7))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Plasmodium falciparum TrxRMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine expressed in Escherichia coli SG13009 using Z-FR-AMC as substrate after 5 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine expressed in Escherichia coli SG13009 using Z-FR-AMC as substrate after 5 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine expressed in Escherichia coli SG13009 using Z-FR-AMC as substrate after 5 minsMore data for this Ligand-Target Pair
TargetThioredoxin reductase 1, cytoplasmic/2, mitochondrial/3(Homo sapiens (Human))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of human TrxRMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine expressed in Escherichia coli SG13009 using Z-FR-AMC as substrate after 5 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine expressed in Escherichia coli SG13009 using Z-FR-AMC as substrate after 5 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine expressed in Escherichia coli SG13009 using Z-FR-AMC as substrate after 5 minsMore data for this Ligand-Target Pair
TargetThioredoxin reductase(Plasmodium falciparum (isolate 3D7))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of Plasmodium falciparum TrxRMore data for this Ligand-Target Pair
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine expressed in Escherichia coli SG13009 using Z-FR-AMC as substrate after 5 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.90E+3nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine expressed in Escherichia coli SG13009 using Z-FR-AMC as substrate after 5 minsMore data for this Ligand-Target Pair
TargetThioredoxin reductase(Plasmodium falciparum (isolate 3D7))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum TrxRMore data for this Ligand-Target Pair
TargetThioredoxin reductase(Plasmodium falciparum (isolate 3D7))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum TrxRMore data for this Ligand-Target Pair
TargetThioredoxin reductase(Plasmodium falciparum (isolate 3D7))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum TrxRMore data for this Ligand-Target Pair
Affinity DataIC50: 1.09E+4nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine expressed in Escherichia coli SG13009 using Z-FR-AMC as substrate after 5 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.12E+4nMAssay Description:Inhibition of Trypanosoma cruzi cruzain expressed in Escherichia coli M15/DH5alpha using Z-Phe-Arg-AMC as substrate by spectrofluorometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.27E+4nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine expressed in Escherichia coli SG13009 using Z-FR-AMC as substrate after 5 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.32E+4nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine expressed in Escherichia coli SG13009 using Z-FR-AMC as substrate after 5 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine expressed in Escherichia coli SG13009 using Z-FR-AMC as substrate after 5 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.51E+4nMAssay Description:Inhibition of Trypanosoma cruzi cruzain expressed in Escherichia coli M15/DH5alpha using Z-Phe-Arg-AMC as substrate by spectrofluorometryMore data for this Ligand-Target Pair
TargetThioredoxin reductase(Plasmodium falciparum (isolate 3D7))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of Plasmodium falciparum TrxRMore data for this Ligand-Target Pair
Affinity DataIC50: 2.39E+4nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine expressed in Escherichia coli SG13009 using Z-FR-AMC as substrate after 5 minsMore data for this Ligand-Target Pair
TargetThioredoxin reductase(Plasmodium falciparum (isolate 3D7))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Plasmodium falciparum TrxRMore data for this Ligand-Target Pair
Affinity DataIC50: 3.84E+4nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine expressed in Escherichia coli SG13009 using Z-FR-AMC as substrate after 5 minsMore data for this Ligand-Target Pair
TargetThioredoxin reductase(Plasmodium falciparum (isolate 3D7))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of Plasmodium falciparum TrxRMore data for this Ligand-Target Pair
TargetThioredoxin reductase 1, cytoplasmic/2, mitochondrial/3(Homo sapiens (Human))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human TrxRMore data for this Ligand-Target Pair
Affinity DataIC50: 6.51E+4nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine expressed in Escherichia coli SG13009 using Z-FR-AMC as substrate after 5 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.75E+4nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine expressed in Escherichia coli SG13009 using Z-FR-AMC as substrate after 5 minsMore data for this Ligand-Target Pair
TargetThioredoxin reductase 1, cytoplasmic/2, mitochondrial/3(Homo sapiens (Human))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of human TrxRMore data for this Ligand-Target Pair
TargetThioredoxin reductase 1, cytoplasmic/2, mitochondrial/3(Homo sapiens (Human))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataIC50: 9.00E+4nMAssay Description:Inhibition of human TrxRMore data for this Ligand-Target Pair
TargetThioredoxin reductase 1, cytoplasmic/2, mitochondrial/3(Homo sapiens (Human))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human TrxRMore data for this Ligand-Target Pair
TargetThioredoxin reductase 1, cytoplasmic/2, mitochondrial/3(Homo sapiens (Human))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataIC50: 1.40E+5nMAssay Description:Inhibition of human TrxRMore data for this Ligand-Target Pair
TargetThioredoxin reductase 1, cytoplasmic/2, mitochondrial/3(Homo sapiens (Human))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Inhibition of human TrxRMore data for this Ligand-Target Pair
TargetThioredoxin reductase 1, cytoplasmic/2, mitochondrial/3(Homo sapiens (Human))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human TrxRMore data for this Ligand-Target Pair
TargetThioredoxin reductase 1, cytoplasmic/2, mitochondrial/3(Homo sapiens (Human))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human TrxRMore data for this Ligand-Target Pair
![](/img/powered_by_small.gif)