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Found 38 with Last Name = 'silverman' and Initial = 'rh'
Target2-5A-dependent ribonuclease(Mus musculus)
Gunma University

Curated by ChEMBL
LigandPNGBDBM50370219(CHEMBL610868)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]-labeled 2-5A from 2-5A dependent Ribonuclease L (RNase L) of mouse liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Mus musculus)
Gunma University

Curated by ChEMBL
LigandPNGBDBM50370220(CHEMBL1163094)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]-labeled 2-5A from 2-5A dependent Ribonuclease L (RNase L) of mouse liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Mus musculus)
Gunma University

Curated by ChEMBL
LigandPNGBDBM50373177(CHEMBL404038)
Affinity DataIC50:  3nMAssay Description:Displacement of [125I]-labeled 2-5A from 2-5A dependent Ribonuclease L (RNase L) of mouse liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Mus musculus)
Gunma University

Curated by ChEMBL
LigandPNGBDBM50421415(CHEMBL414948)
Affinity DataIC50:  4nMAssay Description:Displacement of [125I]-labeled 2-5A from 2-5A dependent Ribonuclease L (RNase L) of mouse liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Mus musculus)
Gunma University

Curated by ChEMBL
LigandPNGBDBM50370222(CHEMBL610866)
Affinity DataIC50:  50nMAssay Description:Displacement of [125I]-labeled 2-5A from 2-5A dependent Ribonuclease L (RNase L) of mouse liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Mus musculus)
Gunma University

Curated by ChEMBL
LigandPNGBDBM50370227(CHEMBL610609)
Affinity DataIC50:  70nMAssay Description:Displacement of [125I]-labeled 2-5A from 2-5A dependent Ribonuclease L (RNase L) of mouse liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Mus musculus)
Gunma University

Curated by ChEMBL
LigandPNGBDBM50370221(CHEMBL610855)
Affinity DataIC50:  500nMAssay Description:Displacement of [125I]-labeled 2-5A from 2-5A dependent Ribonuclease L (RNase L) of mouse liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Mus musculus)
Gunma University

Curated by ChEMBL
LigandPNGBDBM50370224(CHEMBL610867)
Affinity DataIC50:  1.00E+3nMAssay Description:Displacement of [125I]-labeled 2-5A from 2-5A dependent Ribonuclease L (RNase L) of mouse liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM50241367(2-(3,4-Dihydroxy-phenyl)-5,7-dihydroxy-3-((2S,4R,5...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human CYP2D6 preincubated for 5 min by LC-MS/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM50241367(2-(3,4-Dihydroxy-phenyl)-5,7-dihydroxy-3-((2S,4R,5...)
Affinity DataIC50:  1.32E+3nMAssay Description:Inhibition of full length H-RNAase L expressed in Escherichia coli BL21 (DE3) assessed as inhibition rate incubated for 15 min in presence of 5 nM 2-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM50241367(2-(3,4-Dihydroxy-phenyl)-5,7-dihydroxy-3-((2S,4R,5...)
Affinity DataIC50:  1.36E+3nMAssay Description:Inhibition of full length H-RNAase L expressed in Escherichia coli BL21 (DE3) assessed as inhibition rate incubated for 15 min in presence of 1 nM 2-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM50241367(2-(3,4-Dihydroxy-phenyl)-5,7-dihydroxy-3-((2S,4R,5...)
Affinity DataIC50:  1.42E+3nMAssay Description:Inhibition of full length H-RNAase L expressed in Escherichia coli BL21 (DE3) assessed as inhibition rate incubated for 15 min in presence of 20 nM 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM50241367(2-(3,4-Dihydroxy-phenyl)-5,7-dihydroxy-3-((2S,4R,5...)
Affinity DataIC50:  1.63E+3nMAssay Description:Inhibition of recombinant full length H-RNAase L (1 to 741 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition rate in presence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Mus musculus)
Gunma University

Curated by ChEMBL
LigandPNGBDBM50370229(CHEMBL607600)
Affinity DataIC50:  5.00E+3nMAssay Description:Displacement of [125I]-labeled 2-5A from 2-5A dependent Ribonuclease L (RNase L) of mouse liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Mus musculus)
Gunma University

Curated by ChEMBL
LigandPNGBDBM50370225(CHEMBL608161)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [125I]-labeled 2-5A from 2-5A dependent Ribonuclease L (RNase L) of mouse liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Mus musculus)
Gunma University

Curated by ChEMBL
LigandPNGBDBM50370226(CHEMBL607595)
Affinity DataIC50:  1.00E+5nMAssay Description:Displacement of [125I]-labeled 2-5A from 2-5A dependent Ribonuclease L (RNase L) of mouse liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Mus musculus)
Gunma University

Curated by ChEMBL
LigandPNGBDBM50370230(CHEMBL610610)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [125I]-labeled 2-5A from 2-5A dependent Ribonuclease L (RNase L) of mouse liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Mus musculus)
Gunma University

Curated by ChEMBL
LigandPNGBDBM50370223(CHEMBL607888)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [125I]-labeled 2-5A from 2-5A dependent Ribonuclease L (RNase L) of mouse liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Mus musculus)
Gunma University

Curated by ChEMBL
LigandPNGBDBM50370228(CHEMBL607882)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [125I]-labeled 2-5A from 2-5A dependent Ribonuclease L (RNase L) of mouse liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM50362886(VITEXIN)
Affinity DataIC50:  1.90E+5nMAssay Description:Inhibition of recombinant full length H-RNAase L (1 to 741 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition rate in presence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM15236(3,5,7-trihydroxy-2-(3,4,5-trihydroxyphenyl)-4H-chr...)
Affinity DataIC50:  2.64E+5nMAssay Description:Inhibition of recombinant full length H-RNAase L (1 to 741 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition rate in presence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM23448(BUTYLPARABEN | Butyl paraben | Nipabutyl | butyl 4...)
Affinity DataIC50:  2.40E+6nMAssay Description:Inhibition of recombinant full length H-RNAase L (1 to 741 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition rate in presence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM50373166(CHEMBL259819)
Affinity DataKd:  1.80E+4nMAssay Description:Displacement of 5'-phosphorylated, 2',5'-oligoadenylate from human recombinant RNase L assessed as decrease in resonance by surface plasma resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM50373176(C-5950331 | CHEMBL259633)
Affinity DataKd:  1.20E+4nMAssay Description:Displacement of 5'-phosphorylated, 2',5'-oligoadenylate from human recombinant RNase L assessed as decrease in resonance by surface plasma resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM50373177(CHEMBL404038)
Affinity DataKd:  0.0400nMAssay Description:Binding affinity to human recombinant recombinant RNase LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM50373177(CHEMBL404038)
Affinity DataEC50:  0.5nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM50373177(CHEMBL404038)
Affinity DataKd:  0.220nMAssay Description:Displacement of 5'-phosphorylated, 2',5'-oligoadenylate from human recombinant RNase L assessed as decrease in resonance by surface plasma resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM50373176(C-5950331 | CHEMBL259633)
Affinity DataEC50:  2.20E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM50373175(C-5972155 | CHEMBL411931)
Affinity DataEC50:  4.90E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM50373174(C-6131864 | CHEMBL265469)
Affinity DataEC50:  7.90E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM50373173(CHEMBL410485)
Affinity DataEC50:  4.90E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM50373172(C-6474572 | CHEMBL265438)
Affinity DataEC50:  2.60E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM50373171(CHEMBL260229)
Affinity DataEC50:  5.00E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM50373170(CHEMBL408340)
Affinity DataEC50:  9.00E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM50373169(C-5142087 | CHEMBL259804)
Affinity DataEC50:  2.20E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM50373168(C-5947495 | CHEMBL261864)
Affinity DataEC50:  4.80E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM50373166(CHEMBL259819)
Affinity DataEC50:  2.60E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-5A-dependent ribonuclease(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM50373167(CHEMBL406556)
Affinity DataEC50:  9.90E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed