TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Duquesne University Mylan School Of Pharmacy
Curated by ChEMBL
Duquesne University Mylan School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Displacement of [3H]WIN35428 from human dopamine transporter expressed in mouse N2A cells by scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Duquesne University Mylan School Of Pharmacy
Curated by ChEMBL
Duquesne University Mylan School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Displacement of [3H]WIN35428 from human dopamine transporter expressed in mouse N2A cells by scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Duquesne University Mylan School Of Pharmacy
Curated by ChEMBL
Duquesne University Mylan School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 28nMAssay Description:Displacement of [3H]WIN35428 from human dopamine transporter expressed in mouse N2A cells by scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Duquesne University Mylan School Of Pharmacy
Curated by ChEMBL
Duquesne University Mylan School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 78nMAssay Description:Displacement of [3H]WIN35428 from human dopamine transporter expressed in mouse N2A cells by scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Duquesne University Mylan School Of Pharmacy
Curated by ChEMBL
Duquesne University Mylan School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 441nMAssay Description:Displacement of [3H]WIN35428 from human dopamine transporter expressed in mouse N2A cells by scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Duquesne University Mylan School Of Pharmacy
Curated by ChEMBL
Duquesne University Mylan School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 3.07E+3nMAssay Description:Displacement of [3H]WIN-35,428 from human DAT expressed in N2A cells after 15 mins by photoaffinity labelingMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Duquesne University Mylan School Of Pharmacy
Curated by ChEMBL
Duquesne University Mylan School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of [3H]dopamine uptake at human dopamine transporter expressed in mouse N2A cells by scintillation countingMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of human 5alpha-2 reductase expressed in HEK293 cells assessed as suppression of conversion of [3]androstenedione incubated for 30 mins by...More data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 22.1nMAssay Description:Inhibition of human type-2 5-alpha reductase expressed in HEK293 cells using [3H]-androstenedione as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 26.5nMAssay Description:Inhibition of human type-2 5-alpha reductase expressed in HEK293 cells using [3H]-androstenedione as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 30.3nMAssay Description:Inhibition of human type-2 5-alpha reductase expressed in HEK293 cells using [3H]-androstenedione as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Duquesne University Mylan School Of Pharmacy
Curated by ChEMBL
Duquesne University Mylan School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of [3H]dopamine uptake at human dopamine transporter expressed in mouse N2A cells by scintillation countingMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of human 5alpha-2 reductase expressed in HEK293 cells assessed as suppression of conversion of [3]androstenedione incubated for 30 mins by...More data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 54.1nMAssay Description:Inhibition of human type-2 5-alpha reductase expressed in HEK293 cells using [3H]-androstenedione as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 72.8nMAssay Description:Inhibition of human type-2 5-alpha reductase expressed in HEK293 cells using [3H]-androstenedione as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 84nMAssay Description:Inhibition of human 5alpha-2 reductase expressed in HEK293 cells assessed as suppression of conversion of [3]androstenedione incubated for 30 mins by...More data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 157nMAssay Description:Inhibition of human 5alpha-2 reductase expressed in HEK293 cells assessed as suppression of conversion of [3]androstenedione incubated for 30 mins by...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Duquesne University Mylan School Of Pharmacy
Curated by ChEMBL
Duquesne University Mylan School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 175nMAssay Description:Inhibition of [3H]dopamine uptake at human dopamine transporter expressed in mouse N2A cells by scintillation countingMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 213nMAssay Description:Inhibition of human type-2 5-alpha reductase expressed in HEK293 cells using [3H]-androstenedione as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of human 5alpha-2 reductase expressed in HEK293 cells assessed as suppression of conversion of [3]androstenedione incubated for 30 mins by...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Duquesne University Mylan School Of Pharmacy
Curated by ChEMBL
Duquesne University Mylan School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 264nMAssay Description:Inhibition of [3H]dopamine uptake at human dopamine transporter expressed in mouse N2A cells by scintillation countingMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 274nMAssay Description:Inhibition of human 5alpha-2 reductase expressed in HEK293 cells assessed as suppression of conversion of [3]androstenedione incubated for 30 mins by...More data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 453nMAssay Description:Inhibition of human 5alpha-1 reductase expressed in HEK293 cells assessed as suppression of conversion of [3]androstenedione incubated for 30 mins by...More data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 453nMAssay Description:Inhibition of human type-1 5-alpha reductase expressed in HEK293 cells using [3H]-androstenedione as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
University Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 547nMAssay Description:Inhibition of human 5alpha-1 reductase expressed in HEK293 cells assessed as suppression of conversion of [3]androstenedione incubated for 30 mins by...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Duquesne University Mylan School Of Pharmacy
Curated by ChEMBL
Duquesne University Mylan School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 1.57E+3nMAssay Description:Inhibition of [3H]dopamine uptake at human dopamine transporter expressed in mouse N2A cells by scintillation countingMore data for this Ligand-Target Pair
![](/img/powered_by_small.gif)