Affinity DataIC50: <1nMAssay Description:Inhibition of human MB-COMT expressed in HEK293 cells using dopamine as substrate and SAM as cofactor preincubated for 30 mins followed by substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Inhibition of human MB-COMT expressed in HEK293 cells using dopamine as substrate and SAM as cofactor preincubated for 30 mins followed by substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human MB-COMT expressed in HEK293 cells using dopamine as substrate and SAM as cofactor preincubated for 30 mins followed by substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human MB-COMT expressed in HEK293 cells using dopamine as substrate and SAM as cofactor preincubated for 30 mins followed by substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of human MB-COMT expressed in HEK293 cells using dopamine as substrate and SAM as cofactor preincubated for 30 mins followed by substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human CCR3 receptor assessed as inhibition of calcium fluxMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human CCR3 receptor assessed as inhibition of eotaxin-induced eosinophil shape changeMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of human MB-COMT expressed in HEK293 cells using dopamine as substrate and SAM as cofactor preincubated for 30 mins followed by substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Displacement of [125I]C3a from human C3a receptor expressed in HMC1 cells co-expressing aequorinMore data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Inhibition of human MB-COMT expressed in HEK293 cells using dopamine as substrate and SAM as cofactor preincubated for 30 mins followed by substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of human MB-COMT expressed in HEK293 cells using dopamine as substrate and SAM as cofactor preincubated for 30 mins followed by substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of human MB-COMT expressed in HEK293 cells using dopamine as substrate and SAM as cofactor preincubated for 30 mins followed by substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of human MB-COMT expressed in HEK293 cells using dopamine as substrate and SAM as cofactor preincubated for 30 mins followed by substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Displacement of [125I]C3a from human C3a receptor expressed in HMC1 cells co-expressing aequorinMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of human MB-COMT expressed in HEK293 cells using dopamine as substrate and SAM as cofactor preincubated for 30 mins followed by substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of human MB-COMT expressed in HEK293 cells using dopamine as substrate and SAM as cofactor preincubated for 30 mins followed by substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of human MB-COMT expressed in HEK293 cells using dopamine as substrate and SAM as cofactor preincubated for 30 mins followed by substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Inhibition of human MB-COMT expressed in HEK293 cells using dopamine as substrate and SAM as cofactor preincubated for 30 mins followed by substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 79nMAssay Description:Displacement of [125I]C3a from human C3a receptor expressed in HMC1 cells co-expressing aequorinMore data for this Ligand-Target Pair
Affinity DataIC50: 79nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of human MB-COMT expressed in HEK293 cells using dopamine as substrate and SAM as cofactor preincubated for 30 mins followed by substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Displacement of [125I]C3a from human C3a receptor expressed in HMC1 cells co-expressing aequorinMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Displacement of [125I]C3a from human C3a receptor expressed in HMC1 cells co-expressing aequorinMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Displacement of [125I]C3a from human C3a receptor expressed in HMC1 cells co-expressing aequorinMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Displacement of [125I]C3a from human C3a receptor expressed in HMC1 cells co-expressing aequorinMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Displacement of [125I]C3a from human C3a receptor expressed in HMC1 cells co-expressing aequorinMore data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibition of human MB-COMT expressed in HEK293 cells using dopamine as substrate and SAM as cofactor preincubated for 30 mins followed by substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Inhibition of human MB-COMT expressed in HEK293 cells using dopamine as substrate and SAM as cofactor preincubated for 30 mins followed by substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Displacement of [125I]eotaxin from CCR3 receptor in human eosinophilsMore data for this Ligand-Target Pair
Affinity DataIC50: 316nMAssay Description:Displacement of [125I]C3a from human C3a receptor expressed in HMC1 cells co-expressing aequorinMore data for this Ligand-Target Pair
Affinity DataIC50: 316nMAssay Description:Displacement of [125I]C3a from human C3a receptor expressed in HMC1 cells co-expressing aequorinMore data for this Ligand-Target Pair