TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 0.467nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 0.476nMAssay Description:Binding affinity was determined by displacement of [3H]- DAMGO at Opioid receptor mu 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 32.8nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 109nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 152nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 218nMAssay Description:Binding affinity was determined by displacement of [3H]- DAMGO at Opioid receptor mu 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 450nMAssay Description:Binding affinity was determined by displacement of [3H]- DAMGO at Opioid receptor mu 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 486nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 759nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 1.07E+3nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was determined by displacement of [3H]- DAMGO at Opioid receptor mu 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was determined by displacement of [3H]- DAMGO at Opioid receptor mu 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was determined by displacement of [3H]- DAMGO at Opioid receptor mu 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was determined by displacement of [3H]- DAMGO at Opioid receptor mu 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0550nMAssay Description:Inhibitory activity was determined against human vitronectin receptor (alpha V beta 3)More data for this Ligand-Target Pair
Affinity DataIC50: 0.0560nMAssay Description:Inhibition of binding to human alphaV-beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0580nMAssay Description:Inhibitory activity was determined against human alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0630nMAssay Description:Inhibitory activity was determined against human alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 0.150nMAssay Description:Inhibitory activity was determined against human vitronectin receptor (alpha V beta 3)More data for this Ligand-Target Pair
Affinity DataIC50: 0.160nMAssay Description:Inhibition of binding to human alphaV-beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 0.220nMAssay Description:Inhibitory activity was determined against human alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibitory activity was determined against human alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 0.320nMAssay Description:Inhibitory activity was determined against human alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 0.380nMAssay Description:Inhibitory activity was determined against human vitronectin receptor (alpha V beta 3)More data for this Ligand-Target Pair
Affinity DataIC50: 0.590nMAssay Description:Inhibitory activity was determined against human vitronectin receptor (alpha V beta 3)More data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibitory activity was determined against human vitronectin receptor (alpha V beta 3)More data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibitory activity was determined against human alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60nMAssay Description:Inhibitory activity was determined against human vitronectin receptor (alpha V beta 3)More data for this Ligand-Target Pair
Affinity DataIC50: 6.80nMAssay Description:Inhibitory activity was determined against human alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibitory activity was determined against human vitronectin receptor (alpha V beta 3)More data for this Ligand-Target Pair
Affinity DataIC50: 88nMAssay Description:Inhibitory activity was determined against human alpha IIb beta3 integrinMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataIC50: 165nMAssay Description:Compound was tested for delta antagonist activity against tachykinin NK-1.Tachykinin receptor 1More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataIC50: 216nMAssay Description:Compound was tested for delta antagonist activity against Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:Inhibitory activity was determined against human vitronectin receptor (alpha V beta 3)More data for this Ligand-Target Pair
Affinity DataIC50: 540nMAssay Description:Inhibitory activity was determined against human alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 660nMAssay Description:Inhibitory activity was determined against human vitronectin receptor (alpha V beta 3)More data for this Ligand-Target Pair
Affinity DataIC50: 720nMAssay Description:Inhibition of binding to human alphaV-beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity was determined against human vitronectin receptor (alpha V beta 3)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity was determined against human alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity was determined against human vitronectin receptor (alpha V beta 3)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity was determined against human alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity was determined against human alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity was determined against human alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity was determined against human alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity was determined against human alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory activity was determined against human vitronectin receptor (alpha V beta 3)More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataIC50: 1.05E+3nMAssay Description:Compound was tested for delta antagonist activity against Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataIC50: 5.30E+3nMAssay Description:Tested for inhibitory activity of compound against Phospholipase A2 (PLA2)More data for this Ligand-Target Pair
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Kwansei Gakuin University
Curated by ChEMBL
Kwansei Gakuin University
Curated by ChEMBL
Affinity DataIC50: 5.30E+3nMAssay Description:Compound was tested for inhibitory activity against type II Phospholipase A2 (PLA2) isolated from japanese mamushi (A. halys blomhoffii) venomMore data for this Ligand-Target Pair
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Kwansei Gakuin University
Curated by ChEMBL
Kwansei Gakuin University
Curated by ChEMBL
Affinity DataIC50: 1.98E+4nMAssay Description:Compound was tested for inhibitory activity against type II Phospholipase A2 (PLA2) isolated from japanese mamushi (A. halys blomhoffii) venomMore data for this Ligand-Target Pair
![](/img/powered_by_small.gif)