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TargetM-phase inducer phosphatase 2(Mouse)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104684((4-Hexadecanoyl-3-hydroxy-5-oxo-2,5-dihydro-furan-...)
Affinity DataIC50:  380nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mouse)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104691(CHEMBL423508 | Diazo-[2-(4-hexadecanoyl-3-hydroxy-...)
Affinity DataIC50:  400nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mouse)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104690((4-Hexadecanoyl-3-hydroxy-5-oxo-2,5-dihydro-furan-...)
Affinity DataIC50:  520nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandPNGBDBM125988(US8772297, Y244)
Affinity DataIC50:  600nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetM-phase inducer phosphatase 2(Mouse)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104674((4-Hexadecanoyl-3-hydroxy-5-oxo-2,5-dihydro-furan-...)
Affinity DataIC50:  600nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandPNGBDBM125985(US8772297, Y241)
Affinity DataIC50:  700nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetM-phase inducer phosphatase 2(Mouse)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104693(4-Hydroxy-5-hydroxymethyl-3-octadec-9-enoyl-5H-fur...)
Affinity DataIC50:  900nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKynurenine/alpha-aminoadipate aminotransferase, mitochondrial(Human)
University of Piemonte Orientale Amedeo Avogadro

Curated by ChEMBL
LigandPNGBDBM50324539((S)-(-)-9-(4-aminopiperazin-1-yl)-8-fluoro-3-methy...)
Affinity DataIC50:  910nMAssay Description:Inhibition of human recombinant MBP-KAT2 expressed in HEK293 cells assessed as conversion of L-kynurenine to kynurenic acid after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetKynurenine/alpha-aminoadipate aminotransferase, mitochondrial(Rat)
University of Piemonte Orientale Amedeo Avogadro

Curated by ChEMBL
LigandPNGBDBM50324539((S)-(-)-9-(4-aminopiperazin-1-yl)-8-fluoro-3-methy...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of rat brain KAT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKynurenine/alpha-aminoadipate aminotransferase, mitochondrial(Human)
University of Piemonte Orientale Amedeo Avogadro

Curated by ChEMBL
LigandPNGBDBM50324539((S)-(-)-9-(4-aminopiperazin-1-yl)-8-fluoro-3-methy...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of KAT2 in human prefrontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetM-phase inducer phosphatase 2(Mouse)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104677(3-Hexadecanoyl-4-hydroxy-5-methylene-5H-furan-2-on...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50567332(CHEMBL4853586)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of hypoxia-induced HIF1 alpha transcriptional activity in human HeLa cells transfected with luciferase reporter containing of HRE assessed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50567336(CHEMBL4876055)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of hypoxia-induced HIF1 alpha transcriptional activity in human HeLa cells transfected with luciferase reporter containing of HRE assessed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mouse)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104676((4-Hexadecanoyl-3-hydroxy-5-oxo-2,5-dihydro-furan-...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mouse)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104681(CHEMBL109357 | Methanesulfonic acid 4-hexadecanoyl...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50567334(CHEMBL4869045)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of hypoxia-induced HIF1 alpha transcriptional activity in human HeLa cells transfected with luciferase reporter containing of HRE assessed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandPNGBDBM125986(US8772297, Y260)
Affinity DataIC50:  1.50E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetKynurenine/alpha-aminoadipate aminotransferase, mitochondrial(Human)
University of Piemonte Orientale Amedeo Avogadro

Curated by ChEMBL
LigandPNGBDBM50416560(CHEMBL1215660)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human recombinant MBP-KAT2 expressed in HEK293 cells assessed as conversion of L-kynurenine to kynurenic acid after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Human)
Japan Science and Technology Agency

Curated by ChEMBL
LigandPNGBDBM50012280(CHEMBL3260030)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of Vaccinia H1-related phosphatase (unknown origin) by fluorescence emission assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mouse)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104696(4-Hydroxy-5-hydroxymethyl-2-oxo-2,5-dihydro-furan-...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50567333(CHEMBL4865589)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of hypoxia-induced HIF1 alpha transcriptional activity in human HeLa cells transfected with luciferase reporter containing of HRE assessed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mouse)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104688(4-Hydroxy-5-hydroxymethyl-2-oxo-2,5-dihydro-furan-...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandPNGBDBM125979(US8772297, Y177)
Affinity DataIC50:  2.00E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetM-phase inducer phosphatase 2(Mouse)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104694((R)-4-hydroxy-5-(hydroxymethyl)-3-palmitoylfuran-2...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mouse)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104697((4-Hexadecanoyl-3-hydroxy-5-oxo-2,5-dihydro-furan-...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandPNGBDBM125980(US8772297, Y224)
Affinity DataIC50:  2.40E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandPNGBDBM125989(US8772297, Y250)
Affinity DataIC50:  2.50E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetM-phase inducer phosphatase 2(Mouse)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104692(4-Hydroxy-5-nonyloxycarbonylmethyl-2-oxo-2,5-dihyd...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mouse)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104700(3-Hexadecanoyl-4-hydroxy-5H-furan-2-one | CHEMBL32...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mouse)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104703(4-Hydroxy-5-hydroxymethyl-2-oxo-2,5-dihydro-furan-...)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mouse)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104673(4-Hydroxy-5-hydroxymethyl-2-oxo-2,5-dihydro-furan-...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandPNGBDBM125981(US8772297, Y186)
Affinity DataIC50:  3.60E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetM-phase inducer phosphatase 2(Mouse)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104683(3-Hexadecanoyl-4-hydroxy-5-methyl-5H-furan-2-one |...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Human)
Japan Science and Technology Agency

Curated by ChEMBL
LigandPNGBDBM50104684((4-Hexadecanoyl-3-hydroxy-5-oxo-2,5-dihydro-furan-...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibitory activity against vaccinia VH1-related phosphatase(VHR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Human)
Japan Science and Technology Agency

Curated by ChEMBL
LigandPNGBDBM50104690((4-Hexadecanoyl-3-hydroxy-5-oxo-2,5-dihydro-furan-...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibitory activity against vaccinia VH1-related phosphatase(VHR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Human)
Japan Science and Technology Agency

Curated by ChEMBL
LigandPNGBDBM50012323(CHEMBL3260378)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of Vaccinia H1-related phosphatase (unknown origin) by fluorescence emission assay in presence of 0.001% NP-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandPNGBDBM125991(US8772297, Y296)
Affinity DataIC50:  4.60E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetDual specificity protein phosphatase 3(Human)
Japan Science and Technology Agency

Curated by ChEMBL
LigandPNGBDBM50104674((4-Hexadecanoyl-3-hydroxy-5-oxo-2,5-dihydro-furan-...)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibitory activity against vaccinia VH1-related phosphatase(VHR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mouse)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104694((R)-4-hydroxy-5-(hydroxymethyl)-3-palmitoylfuran-2...)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50567331(CHEMBL4850885)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of hypoxia-induced HIF1 alpha transcriptional activity in human HeLa cells transfected with luciferase reporter containing of HRE assessed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mouse)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104699(4-Hydroxy-5-methoxycarbonylmethyl-2-oxo-2,5-dihydr...)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandPNGBDBM125990(US8772297, Y284)
Affinity DataIC50:  6.70E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetHypoxia-inducible factor 1-alpha(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50567335(CHEMBL4854814)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of hypoxia-induced HIF1 alpha transcriptional activity in human HeLa cells transfected with luciferase reporter containing of HRE assessed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandPNGBDBM125987(US8772297, Y366)
Affinity DataIC50:  7.30E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetDual specificity protein phosphatase 3(Human)
Japan Science and Technology Agency

Curated by ChEMBL
LigandPNGBDBM50012321(CHEMBL3260377)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of Vaccinia H1-related phosphatase (unknown origin) by fluorescence emission assay in presence of 0.001% NP-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mouse)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104686(4-Hydroxy-5-hydroxymethyl-2-oxo-2,5-dihydro-furan-...)
Affinity DataIC50:  7.90E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandPNGBDBM125976(US8772297, Y145)
Affinity DataIC50:  8.00E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetDual specificity protein phosphatase 3(Human)
Japan Science and Technology Agency

Curated by ChEMBL
LigandPNGBDBM50012320(CHEMBL3260376)
Affinity DataIC50:  8.20E+3nMAssay Description:Inhibition of Vaccinia H1-related phosphatase (unknown origin) by fluorescence emission assay in presence of 0.001% NP-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Human)
Japan Science and Technology Agency

Curated by ChEMBL
LigandPNGBDBM50104681(CHEMBL109357 | Methanesulfonic acid 4-hexadecanoyl...)
Affinity DataIC50:  9.20E+3nMAssay Description:Inhibitory activity against vaccinia VH1-related phosphatase(VHR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Human)
Japan Science and Technology Agency

Curated by ChEMBL
LigandPNGBDBM50104677(3-Hexadecanoyl-4-hydroxy-5-methylene-5H-furan-2-on...)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibitory activity against vaccinia VH1-related phosphatase(VHR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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