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Found 859 with Last Name = 'lever' and Initial = 's'
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50372600(CHEMBL414138)
Affinity DataKi:  0.370nMAssay Description:Displacement of [3H](+)-PTZ from sigma1 receptor in Hartley guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50372603(CHEMBL271395)
Affinity DataKi:  0.390nMAssay Description:Displacement of [3H](+)-PTZ from sigma1 receptor in Hartley guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50372607(CHEMBL270474)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H](+)-PTZ from sigma1 receptor in Hartley guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50372598(CHEMBL273041)
Affinity DataKi:  0.660nMAssay Description:Displacement of [3H](+)-PTZ from sigma1 receptor in Hartley guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50372605(CHEMBL272650)
Affinity DataKi:  0.760nMAssay Description:Displacement of [3H](+)-PTZ from sigma1 receptor in Hartley guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  0.830nMAssay Description:Displacement of [3H]-(+)-pentazocine from Sigma1-receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  0.830nMAssay Description:Displacement of [3H](+)-PTZ from sigma1 receptor in Hartley guinea pig brainMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50372602(CHEMBL408821)
Affinity DataKi:  0.870nMAssay Description:Displacement of [3H](+)-PTZ from sigma1 receptor in Hartley guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50372601(CHEMBL272050)
Affinity DataKi:  0.930nMAssay Description:Displacement of [3H](+)-PTZ from sigma1 receptor in Hartley guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50372599(CHEMBL269870)
Affinity DataKi:  1.17nMAssay Description:Displacement of [3H](+)-PTZ from sigma1 receptor in Hartley guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50068459(1-[2-(4-Methoxy-phenyl)-ethyl]-4-(3-phenyl-propyl)...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50372606(CHEMBL271396)
Affinity DataKi:  1.36nMAssay Description:Displacement of [3H](+)-PTZ from sigma1 receptor in Hartley guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50068454(1-[2-(3-Methoxy-phenyl)-ethyl]-4-(3-phenyl-propyl)...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50035131((+)-(6R,11S)-6,11-dimethyl-3-(3-methyl-but-2-enyl)...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50040266(CHEMBL3359513)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50068452(1-[2-(3,4-Dichloro-phenyl)-ethyl]-4-(3-phenyl-prop...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50040256(CHEMBL3352893)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50372604(CHEMBL272819)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H](+)-PTZ from sigma1 receptor in Hartley guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50068450(1-[2-(2-Methoxy-phenyl)-ethyl]-4-(3-phenyl-propyl)...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50338990(1-(3,4-dimethoxyphenethyl)-4-(3-phenylpropyl)piper...)
Affinity DataKi:  4.34nMAssay Description:Displacement of [3H](+)-PTZ from sigma1 receptor in Hartley guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50338990(1-(3,4-dimethoxyphenethyl)-4-(3-phenylpropyl)piper...)
Affinity DataKi:  4.34nMAssay Description:Displacement of [3H]-(+)-pentazocine from Sigma1-receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50338990(1-(3,4-dimethoxyphenethyl)-4-(3-phenylpropyl)piper...)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50040264(CHEMBL3360017)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50040265(CHEMBL3360016)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50040258(CHEMBL3360026)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50040263(CHEMBL3360019)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(MOUSE)
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM22165(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-(3-pheny...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]RTI-121 from mouse DAT in striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50040261(CHEMBL3360024)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50040251(CHEMBL3360018)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50040259(CHEMBL3360025)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50040257(CHEMBL3360027)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50040255(CHEMBL3360023)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(MOUSE)
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM22165(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-(3-pheny...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]paroxetine from mouse SERT in whole brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50040262(CHEMBL3360021)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50040252(CHEMBL3360020)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50040254(CHEMBL3360022)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50009307(DITOLYLGUANIDINE | Di-o-tolylguanidine)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50206200(5-bromo-N-(4-(7,8-dihydro-[1,3]dioxolo[4,5-g]isoqu...)
Affinity DataKi:  82.2nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(MOUSE)
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50040259(CHEMBL3360025)
Affinity DataKi:  87nMAssay Description:Displacement of [3H]RTI-121 from mouse DAT in striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(MOUSE)
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50040255(CHEMBL3360023)
Affinity DataKi:  121nMAssay Description:Displacement of [3H]RTI-121 from mouse DAT in striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(MOUSE)
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50040252(CHEMBL3360020)
Affinity DataKi:  124nMAssay Description:Displacement of [3H]paroxetine from mouse SERT in whole brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(MOUSE)
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50040255(CHEMBL3360023)
Affinity DataKi:  128nMAssay Description:Displacement of [3H]paroxetine from mouse SERT in whole brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(MOUSE)
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50040251(CHEMBL3360018)
Affinity DataKi:  174nMAssay Description:Displacement of [3H]paroxetine from mouse SERT in whole brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(MOUSE)
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50040263(CHEMBL3360019)
Affinity DataKi:  237nMAssay Description:Displacement of [3H]RTI-121 from mouse DAT in striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(MOUSE)
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50040254(CHEMBL3360022)
Affinity DataKi:  295nMAssay Description:Displacement of [3H]paroxetine from mouse SERT in whole brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50206201(5-bromo-2,3-dimethoxy-N-(4-(2,3,8,9-tetrahydro-[1,...)
Affinity DataKi:  338nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(MOUSE)
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50040256(CHEMBL3352893)
Affinity DataKi:  468nMAssay Description:Displacement of [3H]paroxetine from mouse SERT in whole brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(MOUSE)
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50040251(CHEMBL3360018)
Affinity DataKi:  560nMAssay Description:Displacement of [3H]RTI-121 from mouse DAT in striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50338989(5-Bromo-N-(4-((3,4-dimethoxyphenethyl)(methyl)-ami...)
Affinity DataKi:  583nMAssay Description:Displacement of [3H]-(+)-pentazocine from Sigma1-receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(MOUSE)
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50338990(1-(3,4-dimethoxyphenethyl)-4-(3-phenylpropyl)piper...)
Affinity DataKi:  760nMAssay Description:Displacement of [3H]paroxetine from mouse SERT in whole brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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