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Found 101 with Last Name = 'mandel' and Initial = 's'
TargetPeripheral plasma membrane protein CASK(Homo sapiens (Human))
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50574225(CHEMBL4850857)
Affinity DataKi:  11nMAssay Description:Inhibition of tracer K5 binding to NanoLuc-fused CASK (unknown origin) expressed in HEK293T cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
TargetPeripheral plasma membrane protein CASK(Homo sapiens (Human))
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50574224(CHEMBL4876584)
Affinity DataKi:  15nMAssay Description:Inhibition of tracer K5 binding to NanoLuc-fused CASK (unknown origin) expressed in HEK293T cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPeripheral plasma membrane protein CASK(Homo sapiens (Human))
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50425829(CHEMBL2312304)
Affinity DataKi:  15nMAssay Description:Inhibition of tracer K5 binding to NanoLuc-fused CASK (unknown origin) expressed in HEK293T cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50425829(CHEMBL2312304)
Affinity DataKi:  120nMAssay Description:Inhibition of tracer K5 binding to NanoLuc-fused TYRO3 (unknown origin) expressed in HEK293T cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM15581(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Affinity DataIC50:  27nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
TargetPeripheral plasma membrane protein CASK(Homo sapiens (Human))
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50574225(CHEMBL4850857)
Affinity DataIC50:  80nMAssay Description:Inhibition of tracer K5 binding to NanoLuc-fused CASK (unknown origin) expressed in HEK293T cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
TargetPeripheral plasma membrane protein CASK(Homo sapiens (Human))
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50574224(CHEMBL4876584)
Affinity DataIC50:  106nMAssay Description:Inhibition of tracer K5 binding to NanoLuc-fused CASK (unknown origin) expressed in HEK293T cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPeripheral plasma membrane protein CASK(Homo sapiens (Human))
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50425829(CHEMBL2312304)
Affinity DataIC50:  130nMAssay Description:Inhibition of tracer K5 binding to NanoLuc-fused CASK (unknown origin) expressed in HEK293T cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM113080(US8633208, 23)
Affinity DataIC50:  150nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM113058(US8633208, 1)
Affinity DataIC50:  220nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM113077(US8633208, 20)
Affinity DataIC50:  250nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM113081(US8633208, 24)
Affinity DataIC50:  280nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM113071(US8633208, 14)
Affinity DataIC50:  350nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM113082(US8633208, 25)
Affinity DataIC50:  450nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM15579(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Affinity DataIC50:  480nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM113075(US8633208, 18)
Affinity DataIC50:  670nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50425829(CHEMBL2312304)
Affinity DataIC50:  700nMAssay Description:Inhibition of tracer K5 binding to NanoLuc-fused TYRO3 (unknown origin) expressed in HEK293T cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM50019848(2-(2,3-dihydro-1,4-benzodioxin-2-yl)-4,5-dihydro-1...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM50019848(2-(2,3-dihydro-1,4-benzodioxin-2-yl)-4,5-dihydro-1...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM113074(US8633208, 17)
Affinity DataIC50:  1.13E+3nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM113079(US8633208, 22)
Affinity DataIC50:  1.49E+3nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPeripheral plasma membrane protein CASK(Homo sapiens (Human))
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50574221(CHEMBL4847568)
Affinity DataIC50:  1.93E+3nMAssay Description:Inhibition of tracer K5 binding to NanoLuc-fused CASK (unknown origin) expressed in HEK293T cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM113061(US8633208, 4)
Affinity DataIC50:  2.06E+3nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM113079(US8633208, 22)
Affinity DataIC50:  2.09E+3nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50574225(CHEMBL4850857)
Affinity DataIC50:  3.79E+3nMAssay Description:Inhibition of tracer K5 binding to NanoLuc-fused TYRO3 (unknown origin) expressed in HEK293T cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50574222(CHEMBL4856516)
Affinity DataIC50:  4.48E+3nMAssay Description:Inhibition of tracer K5 binding to NanoLuc-fused MERTK (unknown origin) expressed in HEK293T cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCytochrome P450 3A4(Homo sapiens (Human))
Rottapharm Madaus

Curated by ChEMBL
LigandPNGBDBM50491250(CHEMBL2381071)
Affinity DataIC50:  7.90E+3nMAssay Description:Inhibition of human recombinant CYP3A4 using BFC as substrate by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50574224(CHEMBL4876584)
Affinity DataIC50:  8.73E+3nMAssay Description:Inhibition of tracer K5 binding to NanoLuc-fused TYRO3 (unknown origin) expressed in HEK293T cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM113063(US8633208, 6)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM113064(US8633208, 7)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM113066(US8633208, 9)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM113070(US8633208, 13)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM113072(US8633208, 15)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM113073(US8633208, 16)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM113076(US8633208, 19)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM113078(US8633208, 21)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM113059(US8633208, 2)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM113062(US8633208, 5)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50574227(CHEMBL4764640)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tracer K5 binding to NanoLuc-fused ABL1 (unknown origin) expressed in HEK293T cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50574225(CHEMBL4850857)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tracer K5 binding to NanoLuc-fused ABL1 (unknown origin) expressed in HEK293T cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50574224(CHEMBL4876584)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tracer K5 binding to NanoLuc-fused ABL1 (unknown origin) expressed in HEK293T cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50574221(CHEMBL4847568)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tracer K5 binding to NanoLuc-fused ABL1 (unknown origin) expressed in HEK293T cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50425829(CHEMBL2312304)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tracer K5 binding to NanoLuc-fused ABL1 (unknown origin) expressed in HEK293T cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50574227(CHEMBL4764640)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tracer K5 binding to NanoLuc-fused AXL (unknown origin) expressed in HEK293T cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50574225(CHEMBL4850857)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tracer K5 binding to NanoLuc-fused AXL (unknown origin) expressed in HEK293T cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50574224(CHEMBL4876584)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tracer K5 binding to NanoLuc-fused AXL (unknown origin) expressed in HEK293T cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM113058(US8633208, 1)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM113059(US8633208, 2)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM113061(US8633208, 4)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Rottapharm

US Patent
LigandPNGBDBM113062(US8633208, 5)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
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