TargetToll-like receptor 7(Mus musculus)
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity at gardiquimod stimulated TRL7 in mouse whole blood assessed as inhibition of IL-6 production by ELISA analysisMore data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Antagonist activity at gardiquimod stimulated TRL7 in human PBMC cells assessed as inhibition of IL-6 production by ELISA analysisMore data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Antagonist activity at gardiquimod stimulated TRL7 in human whole blood assessed as inhibition of IL-6 production by ELISA analysisMore data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 2.60nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 2.70nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 2.80nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 3.80nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 3.90nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 4.20nMAssay Description:Antagonist activity at R848 stimulated TRL8 in human whole blood assessed as inhibition of IL-6 production by ELISA analysisMore data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 6.10nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 6.10nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 7.20nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 7.60nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 8.20nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 9.40nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 72nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 74nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 75nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 81nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 92nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 93nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 97nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 99nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair