Affinity DataKi: 0.690nMAssay Description:Binding affinity to human Angiotensin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition of human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Inhibition of human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Inhibition of human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Inhibition of human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 86nMAssay Description:Inhibition of human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 160nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
Affinity DataKi: 206nMAssay Description:Inhibition of human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 210nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 260nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 310nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 310nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 360nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 450nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 470nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 520nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 550nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 650nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 670nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 753nMAssay Description:Inhibition of human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 820nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.70E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.70E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.70E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 2.10E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 2.60E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 2.70E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 3.10E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 4.50E+3nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 6.30E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 6.50E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 6.60E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 6.60E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 7.20E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 8.10E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human Angiotensin receptor 2More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.20E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.20E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.50E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.54E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase Y181C mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.59E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase L100I mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.80E+4nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair