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Found 2128 with Last Name = 'ewing' and Initial = 't'
TargetCathepsin D(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50076285(1-Acetyl-piperidine-4-carboxylic acid (2-benzo[1,3...)
Affinity DataKi:  1.30nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50076294(1-Acetyl-piperidine-4-carboxylic acid (2-benzo[1,3...)
Affinity DataKi:  1.90nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University of California

Curated by ChEMBL
LigandPNGBDBM50076292(1-Methyl-piperidine-4-carboxylic acid {(2S,3S)-3-[...)
Affinity DataKi:  2nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University of California

Curated by ChEMBL
LigandPNGBDBM50076291(1-Methyl-piperidine-4-carboxylic acid (2-benzo[1,3...)
Affinity DataKi:  2nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University of California

Curated by ChEMBL
LigandPNGBDBM50076285(1-Acetyl-piperidine-4-carboxylic acid (2-benzo[1,3...)
Affinity DataKi:  3nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University of California

Curated by ChEMBL
LigandPNGBDBM50076294(1-Acetyl-piperidine-4-carboxylic acid (2-benzo[1,3...)
Affinity DataKi:  4nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University of California

Curated by ChEMBL
LigandPNGBDBM50076287(1-Methyl-piperidine-4-carboxylic acid [(2S,3S)-3-(...)
Affinity DataKi:  4.10nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50076293(1-Acetyl-piperidine-4-carboxylic acid (2-benzo[1,3...)
Affinity DataKi:  4.30nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University of California

Curated by ChEMBL
LigandPNGBDBM8019(2-(3-chlorophenoxy)-N-[(2S,3S)-3-hydroxy-4-{N-[2-(...)
Affinity DataKi:  4.30nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University of California

Curated by ChEMBL
LigandPNGBDBM50076293(1-Acetyl-piperidine-4-carboxylic acid (2-benzo[1,3...)
Affinity DataKi:  4.80nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50076291(1-Methyl-piperidine-4-carboxylic acid (2-benzo[1,3...)
Affinity DataKi:  5.80nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM36570(EHM)
Affinity DataKi:  9nM IC50:  14nMpH: 3.7Assay Description:A fluorometric high through-put assay for inhibitor towards human liver cathepsin D from Calbiochem.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University of California

Curated by ChEMBL
LigandPNGBDBM50076288(CHEMBL284955 | Piperidine-4-carboxylic acid [(2S,3...)
Affinity DataKi:  9nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50076292(1-Methyl-piperidine-4-carboxylic acid {(2S,3S)-3-[...)
Affinity DataKi:  9.80nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM36569(FHO)
Affinity DataKi:  14nM IC50:  18nMpH: 3.7Assay Description:A fluorometric high through-put assay for inhibitor towards human liver cathepsin D from Calbiochem.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM36567(EHO)
Affinity DataKi:  15nM IC50:  19nMpH: 3.7Assay Description:A fluorometric high through-put assay for inhibitor towards human liver cathepsin D from Calbiochem.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM36571(EHR)
Affinity DataKi:  15nM IC50:  20nMpH: 3.7Assay Description:A fluorometric high through-put assay for inhibitor towards human liver cathepsin D from Calbiochem.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50076286(CHEMBL34051 | N-(2-Benzo[1,3]dioxol-5-yl-ethyl)-N-...)
Affinity DataKi:  15nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50076287(1-Methyl-piperidine-4-carboxylic acid [(2S,3S)-3-(...)
Affinity DataKi:  58nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM36572(EHS)
Affinity DataKi:  59nM IC50:  64nMpH: 3.7Assay Description:A fluorometric high through-put assay for inhibitor towards human liver cathepsin D from Calbiochem.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM8019(2-(3-chlorophenoxy)-N-[(2S,3S)-3-hydroxy-4-{N-[2-(...)
Affinity DataKi:  63nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50076288(CHEMBL284955 | Piperidine-4-carboxylic acid [(2S,3...)
Affinity DataKi:  71nMAssay Description:Compound was tested for the inhibitory activity against human liver cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM36559(EHD)
Affinity DataKi:  73nMpH: 3.7Assay Description:A fluorometric high through-put assay for inhibitor towards human liver cathepsin D from Calbiochem.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University of California

Curated by ChEMBL
LigandPNGBDBM50076289(CHEMBL32997 | N-((1S,2S)-3-{(2-Benzo[1,3]dioxol-5-...)
Affinity DataKi:  100nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetCathepsin D(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM36561(EHJ)
Affinity DataKi:  111nMpH: 3.7Assay Description:A fluorometric high through-put assay for inhibitor towards human liver cathepsin D from Calbiochem.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM36562(EHA)
Affinity DataKi:  131nMpH: 3.7Assay Description:A fluorometric high through-put assay for inhibitor towards human liver cathepsin D from Calbiochem.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM36563(EFA)
Affinity DataKi:  171nMpH: 3.7Assay Description:A fluorometric high through-put assay for inhibitor towards human liver cathepsin D from Calbiochem.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University of California

Curated by ChEMBL
LigandPNGBDBM50076286(CHEMBL34051 | N-(2-Benzo[1,3]dioxol-5-yl-ethyl)-N-...)
Affinity DataKi:  220nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM36573(UHD)
Affinity DataKi:  224nM IC50:  229nMpH: 3.7Assay Description:A fluorometric high through-put assay for inhibitor towards human liver cathepsin D from Calbiochem.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM36564(FHA)
Affinity DataKi:  231nMpH: 3.7Assay Description:A fluorometric high through-put assay for inhibitor towards human liver cathepsin D from Calbiochem.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
University of California

Curated by ChEMBL
LigandPNGBDBM50076290(CHEMBL284151 | N-(2-Benzo[1,3]dioxol-5-yl-ethyl)-N...)
Affinity DataKi:  300nMAssay Description:Inhibitory activity against Plasmepsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM36565(FBB)
Affinity DataKi:  356nMpH: 3.7Assay Description:A fluorometric high through-put assay for inhibitor towards human liver cathepsin D from Calbiochem.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit [D816V](Homo sapiens (Human))
Plexxikon

US Patent
LigandPNGBDBM369320(N-[4-[6-(4-fluorophenyl)thieno[3,2- d]pyrimidin-4-...)
Affinity DataKi:  500nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMast/stem cell growth factor receptor Kit [D816V](Homo sapiens (Human))
Plexxikon

US Patent
LigandPNGBDBM369324(N-(4-fluorophenyl)-4-thieno[3,2- d]pyrimidin-4-yl-...)
Affinity DataKi:  500nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMast/stem cell growth factor receptor Kit [D816V](Homo sapiens (Human))
Plexxikon

US Patent
LigandPNGBDBM369325(N-[(1S)-1-(3-chlorophenyl)ethyl]-2,2- dimethyl-4-(...)
Affinity DataKi:  500nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMast/stem cell growth factor receptor Kit [D816V](Homo sapiens (Human))
Plexxikon

US Patent
LigandPNGBDBM369326(N-[(1S)-1-(4-fluorophenyl)ethyl]-4-[6-(4- fluoroph...)
Affinity DataKi:  500nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMast/stem cell growth factor receptor Kit [D816V](Homo sapiens (Human))
Plexxikon

US Patent
LigandPNGBDBM369327(N-[(1S)-1-(4-fluorophenypethyl]-4-[6-(2- methoxy-4...)
Affinity DataKi:  500nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMast/stem cell growth factor receptor Kit [D816V](Homo sapiens (Human))
Plexxikon

US Patent
LigandPNGBDBM369331((2R)-N-[(1S)-1-(3-chlorophenyl)ethyl]-2- methyl-4-...)
Affinity DataKi:  500nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMast/stem cell growth factor receptor Kit [D816V](Homo sapiens (Human))
Plexxikon

US Patent
LigandPNGBDBM369332((2R)-N-[(1S)-1-[3- (difluoromethoxy)phenyl]ethyl]-...)
Affinity DataKi:  500nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMast/stem cell growth factor receptor Kit [D816V](Homo sapiens (Human))
Plexxikon

US Patent
LigandPNGBDBM369333((2R)-N-[(1S)-1-(4-chloro-3-methoxy- phenyl)ethyl]-...)
Affinity DataKi:  500nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMast/stem cell growth factor receptor Kit [D816V](Homo sapiens (Human))
Plexxikon

US Patent
LigandPNGBDBM369334(N-[(1S)-1-(3-chlorophenyl)ethyl]-4-[6-(2- methoxy-...)
Affinity DataKi:  500nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMast/stem cell growth factor receptor Kit [D816V](Homo sapiens (Human))
Plexxikon

US Patent
LigandPNGBDBM369335(N-[4-(6-methyl-7H-pyrrolo[2,3- d]pyrimidin-4-yl)cy...)
Affinity DataKi:  500nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMast/stem cell growth factor receptor Kit [D816V](Homo sapiens (Human))
Plexxikon

US Patent
LigandPNGBDBM369338(N-[4-[6-(2-methoxy-4-pyridyl)-7H- pyrrolo[2,3-d]py...)
Affinity DataKi:  500nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMast/stem cell growth factor receptor Kit [D816V](Homo sapiens (Human))
Plexxikon

US Patent
LigandPNGBDBM369343(N-[1-[6-(1,3-dimethylpyrazol-4-yl)-7H- pyrrolo[2,3...)
Affinity DataKi:  500nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMast/stem cell growth factor receptor Kit [D816V](Homo sapiens (Human))
Plexxikon

US Patent
LigandPNGBDBM369344(N-[1-[6-(2-methoxy-4-pyridyl)-7H- pyrrolo[2,3-d]py...)
Affinity DataKi:  500nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMast/stem cell growth factor receptor Kit [D816V](Homo sapiens (Human))
Plexxikon

US Patent
LigandPNGBDBM369348(N-[1-[6-(2,4-dimethylthiazol-5-yl)-7H- pyrrolo[2,3...)
Affinity DataKi:  500nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Plexxikon

US Patent
LigandPNGBDBM369349(5-ethyl-N-[1-[6-(1-methylpyrazol-4-yl)- 7H-pyrrolo...)
Affinity DataKi:  500nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMast/stem cell growth factor receptor Kit [D816V](Homo sapiens (Human))
Plexxikon

US Patent
LigandPNGBDBM369349(5-ethyl-N-[1-[6-(1-methylpyrazol-4-yl)- 7H-pyrrolo...)
Affinity DataKi:  500nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMast/stem cell growth factor receptor Kit [D816V](Homo sapiens (Human))
Plexxikon

US Patent
LigandPNGBDBM369350(4-chloro-N-[1-[6-(2-methoxy-4- pyridyl)-7H-pyrrolo...)
Affinity DataKi:  500nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Plexxikon

US Patent
LigandPNGBDBM369351(4-chloro-N-[1-[6-(1,3-dimethylpyrazol- 4-yl)-7H-py...)
Affinity DataKi:  500nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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