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Found 31 with Last Name = 'rungrotmongkol' and Initial = 't'
TargetNeuraminidase(Influenza A virus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50484774(CHEMBL1956716)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of Influenza A virus H7N3 N3 neuraminidase expressed in baculovirus using 2'-(4-Methylumbelliferyl)-alpha-D-acetyl neuraminic acid as subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50484773(OSELTAMIVIR POTTASIUM CARBOXYLATE | Oseltamivir Po...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of Influenza A virus H7N3 N3 neuraminidase expressed in baculovirus using 2'-(4-Methylumbelliferyl)-alpha-D-acetyl neuraminic acid as subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM5025(Oseltamivir | US10919856, POSITIVE CONTROL | ethyl...)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of Influenza A virus H7N3 N3 neuraminidase expressed in baculovirus using 2'-(4-Methylumbelliferyl)-alpha-D-acetyl neuraminic acid as subs...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50484775(CHEMBL1956713)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of Influenza A virus H7N3 N3 neuraminidase expressed in baculovirus using 2'-(4-Methylumbelliferyl)-alpha-D-acetyl neuraminic acid as subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Bangkok

Curated by ChEMBL
LigandPNGBDBM5446(CHEMBL553 | ERLOTINIB HYDROCHLORIDE | Erlotinib | ...)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of recombinant human DYKDDDD-tagged EGFR (669 to 1210 residues) expressed in baculovirus expression system using poly-Glu-Tyr (4:1) as sub...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM4994((3R,4R,5S)-5-amino-4-acetamido-3-(pentan-3-yloxy)c...)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of Influenza A virus (A/duck/Singapore/3/1997(H5N3)) neuraminidase N3More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM4994((3R,4R,5S)-5-amino-4-acetamido-3-(pentan-3-yloxy)c...)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of Influenza A virus (A/duck/Germany/1215/1973(H2N3)) neuraminidase N3More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50484776(CHEMBL1956717)
Affinity DataIC50:  15nMAssay Description:Inhibition of Influenza A virus H7N1 N1 neuraminidase expressed in baculovirus using 2'-(4-Methylumbelliferyl)-alpha-D-acetyl neuraminic acid as subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
University Bangkok

Curated by ChEMBL
LigandPNGBDBM50562022(CHEMBL4797515)
Affinity DataIC50:  18nMAssay Description:Inhibition of recombinant human JAK2 JH1 domain expressed in baculovirus infected insect cells using poly-Glu-Tyr (51 to 68 residues) as substrate in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
University Bangkok

Curated by ChEMBL
LigandPNGBDBM50355501(INCB-018424 | RUXOLITINIB | RUXOLITINIB PHOSPHATE ...)
Affinity DataIC50:  18nMAssay Description:Inhibition of recombinant human JAK2 JH1 domain expressed in baculovirus infected insect cells using poly-Glu-Tyr (51 to 68 residues) as substrate in...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
University Bangkok

Curated by ChEMBL
LigandPNGBDBM50562021(CHEMBL4798434)
Affinity DataIC50:  20nMAssay Description:Inhibition of recombinant human JAK2 JH1 domain expressed in baculovirus infected insect cells using poly-Glu-Tyr (51 to 68 residues) as substrate in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM5025(Oseltamivir | US10919856, POSITIVE CONTROL | ethyl...)
Affinity DataIC50:  25nMAssay Description:Inhibition of Influenza A virus H7N1 N1 neuraminidase expressed in baculovirus using 2'-(4-Methylumbelliferyl)-alpha-D-acetyl neuraminic acid as subs...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50484776(CHEMBL1956717)
Affinity DataIC50:  28nMAssay Description:Inhibition of Influenza A virus H7N3 N3 neuraminidase expressed in baculovirus using 2'-(4-Methylumbelliferyl)-alpha-D-acetyl neuraminic acid as subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Bangkok

Curated by ChEMBL
LigandPNGBDBM5446(CHEMBL553 | ERLOTINIB HYDROCHLORIDE | Erlotinib | ...)
Affinity DataIC50:  28nMAssay Description:Inhibition of human EGFR TK domain expressed in Escherichia coli BL21 (DE3) pLysS using poly-Glu-Tyr (51 to 68 residues) as substrate incubated for 1...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50484774(CHEMBL1956716)
Affinity DataIC50:  32nMAssay Description:Inhibition of Influenza A virus H7N1 N1 neuraminidase expressed in baculovirus using 2'-(4-Methylumbelliferyl)-alpha-D-acetyl neuraminic acid as subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Bangkok

Curated by ChEMBL
LigandPNGBDBM50562023(CHEMBL4750368)
Affinity DataIC50:  34nMAssay Description:Inhibition of human EGFR TK domain expressed in Escherichia coli BL21 (DE3) pLysS using poly-Glu-Tyr (51 to 68 residues) as substrate incubated for 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
University Bangkok

Curated by ChEMBL
LigandPNGBDBM50562023(CHEMBL4750368)
Affinity DataIC50:  34nMAssay Description:Inhibition of recombinant human JAK2 JH1 domain expressed in baculovirus infected insect cells using poly-Glu-Tyr (51 to 68 residues) as substrate in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM4994((3R,4R,5S)-5-amino-4-acetamido-3-(pentan-3-yloxy)c...)
Affinity DataIC50:  36nMAssay Description:Inhibition of Influenza A virus (A/Teal/Hong Kong/W312/97(H6N1)) neuraminidase N1More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50484773(OSELTAMIVIR POTTASIUM CARBOXYLATE | Oseltamivir Po...)
Affinity DataIC50:  39nMAssay Description:Inhibition of Influenza A virus H7N1 N1 neuraminidase expressed in baculovirus using 2'-(4-Methylumbelliferyl)-alpha-D-acetyl neuraminic acid as subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM4994((3R,4R,5S)-5-amino-4-acetamido-3-(pentan-3-yloxy)c...)
Affinity DataIC50:  53nMAssay Description:Inhibition of Influenza A virus (A/duck/Alberta/35/1976(H1N1)) neuraminidase N1More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50484775(CHEMBL1956713)
Affinity DataIC50:  84nMAssay Description:Inhibition of Influenza A virus H7N1 N1 neuraminidase expressed in baculovirus using 2'-(4-Methylumbelliferyl)-alpha-D-acetyl neuraminic acid as subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50377954(CHEMBL557422)
Affinity DataIC50:  91nMAssay Description:Inhibition of Torpedo californica AchE activity by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Bangkok

Curated by ChEMBL
LigandPNGBDBM50562022(CHEMBL4797515)
Affinity DataIC50:  144nMAssay Description:Inhibition of human EGFR TK domain expressed in Escherichia coli BL21 (DE3) pLysS using poly-Glu-Tyr (51 to 68 residues) as substrate incubated for 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Bangkok

Curated by ChEMBL
LigandPNGBDBM50562021(CHEMBL4798434)
Affinity DataIC50:  256nMAssay Description:Inhibition of human EGFR TK domain expressed in Escherichia coli BL21 (DE3) pLysS using poly-Glu-Tyr (51 to 68 residues) as substrate incubated for 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Mahidol University

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  590nMAssay Description:Inhibition of Torpedo californica AchE activity by Ellman's assayMore data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50484772(CHEMBL1956714)
Affinity DataIC50:  4.51E+3nMAssay Description:Inhibition of Influenza A virus H7N3 N3 neuraminidase expressed in baculovirus using 2'-(4-Methylumbelliferyl)-alpha-D-acetyl neuraminic acid as subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50484771(CHEMBL1956712)
Affinity DataIC50:  5.16E+4nMAssay Description:Inhibition of Influenza A virus H7N1 N1 neuraminidase expressed in baculovirus using 2'-(4-Methylumbelliferyl)-alpha-D-acetyl neuraminic acid as subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50484771(CHEMBL1956712)
Affinity DataIC50:  9.93E+4nMAssay Description:Inhibition of Influenza A virus H7N3 N3 neuraminidase expressed in baculovirus using 2'-(4-Methylumbelliferyl)-alpha-D-acetyl neuraminic acid as subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50484772(CHEMBL1956714)
Affinity DataIC50:  1.39E+5nMAssay Description:Inhibition of Influenza A virus H7N1 N1 neuraminidase expressed in baculovirus using 2'-(4-Methylumbelliferyl)-alpha-D-acetyl neuraminic acid as subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50243985(2-Bromoamphimedine | CHEMBL453326)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of Torpedo californica AchE activity by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Bangkok

Curated by ChEMBL
LigandPNGBDBM50562020(CHEMBL4798627)
Affinity DataIC50:  5.50E+7nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed