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Found 53 with Last Name = 'quang' and Initial = 'th'
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Wonkwang University

Curated by ChEMBL
LigandPNGBDBM50036280(CHEMBL3353035)
Affinity DataIC50:  8.20E+3nMAssay Description:Inhibition of human recombinant PTP1B assessed as reduction in pNPP substrate hydrolysis incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Wonkwang University

Curated by ChEMBL
LigandPNGBDBM50036279(CHEMBL3353037)
Affinity DataIC50:  8.20E+3nMAssay Description:Inhibition of human recombinant PTP1B assessed as reduction in pNPP substrate hydrolysis incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50379793(PLUVIATILOL)
Affinity DataEC50: >6.00E+4nMAssay Description:Transactivation of GAL4-fused PPARalpha LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50379794(PINORESINOL)
Affinity DataEC50: >6.00E+4nMAssay Description:Transactivation of GAL4-fused PPARalpha LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50379795(CHEMBL2011541)
Affinity DataEC50:  1.95E+4nMAssay Description:Transactivation of GAL4-fused PPARalpha LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50379791(METHYLEUGENOL | Methyl eugenol (1))
Affinity DataEC50:  4.65E+4nMAssay Description:Transactivation of GAL4-fused PPARalpha LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50379796(CHEMBL2011543)
Affinity DataEC50:  1.57E+4nMAssay Description:Transactivation of GAL4-fused PPARalpha LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50379797(CHEMBL2011544)
Affinity DataEC50:  4.00E+3nMAssay Description:Transactivation of GAL4-fused PPARalpha LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50371235(CIPROFIBRATE)
Affinity DataEC50:  900nMAssay Description:Transactivation of GAL4-fused PPARalpha LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50379792(CHEMBL2011538)
Affinity DataEC50:  2.26E+4nMAssay Description:Transactivation of GAL4-fused PPARgamma LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50379793(PLUVIATILOL)
Affinity DataEC50:  4.87E+4nMAssay Description:Transactivation of GAL4-fused PPARgamma LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50379794(PINORESINOL)
Affinity DataEC50:  5.86E+4nMAssay Description:Transactivation of GAL4-fused PPARgamma LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50379798(PIPERITOL)
Affinity DataEC50:  1.89E+4nMAssay Description:Transactivation of GAL4-fused PPARgamma LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50379798(PIPERITOL)
Affinity DataEC50:  5.32E+4nMAssay Description:Transactivation of GAL4-fused PPARalpha LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50379795(CHEMBL2011541)
Affinity DataEC50:  2.17E+4nMAssay Description:Transactivation of GAL4-fused PPARgamma LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50379796(CHEMBL2011543)
Affinity DataEC50:  1.93E+4nMAssay Description:Transactivation of GAL4-fused PPARgamma LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50379797(CHEMBL2011544)
Affinity DataEC50:  3.60E+3nMAssay Description:Transactivation of GAL4-fused PPARgamma LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50085045(5-((4-((6-hydroxy-2,5,7,8-tetramethyl-3,4-dihydro-...)
Affinity DataEC50:  730nMAssay Description:Transactivation of GAL4-fused PPARgamma LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50379792(CHEMBL2011538)
Affinity DataEC50:  4.76E+4nMAssay Description:Transactivation of GAL4-fused PPARbeta LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50379793(PLUVIATILOL)
Affinity DataEC50:  5.31E+4nMAssay Description:Transactivation of GAL4-fused PPARbeta LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50379794(PINORESINOL)
Affinity DataEC50:  4.95E+4nMAssay Description:Transactivation of GAL4-fused PPARbeta LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50379798(PIPERITOL)
Affinity DataEC50:  3.39E+4nMAssay Description:Transactivation of GAL4-fused PPARbeta LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50379795(CHEMBL2011541)
Affinity DataEC50:  4.85E+4nMAssay Description:Transactivation of GAL4-fused PPARbeta LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50379791(METHYLEUGENOL | Methyl eugenol (1))
Affinity DataEC50:  5.06E+4nMAssay Description:Transactivation of GAL4-fused PPARbeta LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394344(CHEMBL2159607)
Affinity DataEC50:  3.01E+4nMAssay Description:Transactivation of GAL4-fused PPARbeta (delta) ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50379799(CHEMBL2011545)
Affinity DataEC50:  4.61E+4nMAssay Description:Transactivation of GAL4-fused PPARalpha LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50379799(CHEMBL2011545)
Affinity DataEC50:  5.23E+4nMAssay Description:Transactivation of GAL4-fused PPARgamma LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50379799(CHEMBL2011545)
Affinity DataEC50:  5.11E+4nMAssay Description:Transactivation of GAL4-fused PPARbeta LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50379797(CHEMBL2011544)
Affinity DataEC50:  4.90E+3nMAssay Description:Transactivation of GAL4-fused PPARbeta LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50085041(2-(4-(3-(4-acetyl-3-hydroxy-2-propylphenoxy)propox...)
Affinity DataEC50:  640nMAssay Description:Transactivation of GAL4-fused PPARbeta LBD expressed in HepG2 cells after 20 hrs by luminescence assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50085041(2-(4-(3-(4-acetyl-3-hydroxy-2-propylphenoxy)propox...)
Affinity DataEC50:  650nMAssay Description:Transactivation of GAL4-fused PPARbeta (delta) ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394341(CHEMBL465800)
Affinity DataEC50:  2.31E+4nMAssay Description:Transactivation of GAL4-fused PPARbeta (delta) ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394342(CHEMBL458899)
Affinity DataEC50:  1.56E+4nMAssay Description:Transactivation of GAL4-fused PPARbeta (delta) ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394343(CHEMBL516827)
Affinity DataEC50:  2.93E+4nMAssay Description:Transactivation of GAL4-fused PPARbeta (delta) ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394345(CHEMBL2159606)
Affinity DataEC50:  1.31E+4nMAssay Description:Transactivation of GAL4-fused PPARbeta (delta) ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394346(CHEMBL2159605)
Affinity DataEC50:  1.10E+4nMAssay Description:Transactivation of GAL4-fused PPARbeta (delta) ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50085045(5-((4-((6-hydroxy-2,5,7,8-tetramethyl-3,4-dihydro-...)
Affinity DataEC50:  720nMAssay Description:Transactivation of GAL4-fused PPARgamma ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394341(CHEMBL465800)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARgamma ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394342(CHEMBL458899)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARgamma ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394343(CHEMBL516827)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARgamma ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394344(CHEMBL2159607)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARgamma ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394345(CHEMBL2159606)
Affinity DataEC50:  3.31E+4nMAssay Description:Transactivation of GAL4-fused PPARgamma ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394346(CHEMBL2159605)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARgamma ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50371235(CIPROFIBRATE)
Affinity DataEC50:  900nMAssay Description:Transactivation of GAL4-fused PPARalpha ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394341(CHEMBL465800)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARalpha ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394342(CHEMBL458899)
Affinity DataEC50:  4.29E+4nMAssay Description:Transactivation of GAL4-fused PPARalpha ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394343(CHEMBL516827)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARalpha ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394344(CHEMBL2159607)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARalpha ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394345(CHEMBL2159606)
Affinity DataEC50: >5.00E+4nMAssay Description:Transactivation of GAL4-fused PPARalpha ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50394346(CHEMBL2159605)
Affinity DataEC50:  4.71E+4nMAssay Description:Transactivation of GAL4-fused PPARalpha ligand binding domain transfected in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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