TargetAldehyde dehydrogenase, dimeric NADP-preferring(Homo sapiens (Human))
University Of Bradford
Curated by ChEMBL
University Of Bradford
Curated by ChEMBL
Affinity DataKi: 240nMAssay Description:Competitive inhibition of N-terminal-His6 tagged recombinant human ALDH3A1 using 4-NBA and NADP+ as substrate by Michaelis-Menten based analysisMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Homo sapiens (Human))
University Of Bradford
Curated by ChEMBL
University Of Bradford
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Competitive inhibition of N-terminal-His6 tagged recombinant human ALDH3A1 using 4-NBA and NADP+ as substrate by Michaelis-Menten based analysisMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Bradford
Curated by ChEMBL
University Of Bradford
Curated by ChEMBL
Affinity DataKi: 460nMAssay Description:Competitive inhibition of N-terminal-His6 tagged recombinant human ALDH1A3 assessed as increase in Km without change in Vmax using hexanal as substra...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Bradford
Curated by ChEMBL
University Of Bradford
Curated by ChEMBL
Affinity DataKi: <1.00E+3nMAssay Description:Competitive inhibition of N-terminal-His6 tagged recombinant human ALDH1A3 assessed as increase in Km without change in Vmax using hexanal as substra...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Bradford
Curated by ChEMBL
University Of Bradford
Curated by ChEMBL
Affinity DataKi: <1.00E+3nMAssay Description:Competitive inhibition of N-terminal-His6 tagged recombinant human ALDH1A3 assessed as increase in Km without change in Vmax using hexanal as substra...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Bradford
Curated by ChEMBL
University Of Bradford
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH1A3 assessed as reduction in NADH production using hexanal and NAD+ as substrate by fluori...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Bradford
Curated by ChEMBL
University Of Bradford
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH1A3 assessed as reduction in NADH production using hexanal and NAD+ as substrate by fluori...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Bradford
Curated by ChEMBL
University Of Bradford
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH1A3 assessed as reduction in NADH production using hexanal and NAD+ as substrate by fluori...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Bradford
Curated by ChEMBL
University Of Bradford
Curated by ChEMBL
Affinity DataIC50: 310nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH1A3 assessed as reduction in NADH production using hexanal and NAD+ as substrate by fluori...More data for this Ligand-Target Pair
Affinity DataIC50: 480nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH1A1 assessed as reduction in NADH production using hexanal and NAD+ as substrate by fluori...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Bradford
Curated by ChEMBL
University Of Bradford
Curated by ChEMBL
Affinity DataIC50: 550nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH1A3 assessed as reduction in NADH production using hexanal and NAD+ as substrate by fluori...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Bradford
Curated by ChEMBL
University Of Bradford
Curated by ChEMBL
Affinity DataIC50: 630nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH1A3 assessed as reduction in NADH production using hexanal and NAD+ as substrate by fluori...More data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH1A1 assessed as reduction in NADH production using hexanal and NAD+ as substrate by fluori...More data for this Ligand-Target Pair
Affinity DataIC50: 880nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH1A1 assessed as reduction in NADH production using hexanal and NAD+ as substrate by fluori...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Bradford
Curated by ChEMBL
University Of Bradford
Curated by ChEMBL
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH1A3 assessed as reduction in NADH production using hexanal and NAD+ as substrate by fluori...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Homo sapiens (Human))
University Of Bradford
Curated by ChEMBL
University Of Bradford
Curated by ChEMBL
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH3A1 assessed as reduction in NADPH production using 4-NBA and NADP+ as substrate by fluori...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Homo sapiens (Human))
University Of Bradford
Curated by ChEMBL
University Of Bradford
Curated by ChEMBL
Affinity DataIC50: 1.61E+3nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH3A1 assessed as reduction in NADPH production using 4-NBA and NADP+ as substrate by fluori...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Bradford
Curated by ChEMBL
University Of Bradford
Curated by ChEMBL
Affinity DataIC50: 2.37E+3nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH1A3 assessed as reduction in NADH production using hexanal and NAD+ as substrate by fluori...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Bradford
Curated by ChEMBL
University Of Bradford
Curated by ChEMBL
Affinity DataIC50: 4.86E+3nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH1A3 assessed as reduction in NADH production using hexanal and NAD+ as substrate by fluori...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Homo sapiens (Human))
University Of Bradford
Curated by ChEMBL
University Of Bradford
Curated by ChEMBL
Affinity DataIC50: 5.67E+3nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH3A1 assessed as reduction in NADPH production using 4-NBA and NADP+ as substrate by fluori...More data for this Ligand-Target Pair
Affinity DataIC50: 7.08E+3nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH1A1 assessed as reduction in NADH production using hexanal and NAD+ as substrate by fluori...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Homo sapiens (Human))
University Of Bradford
Curated by ChEMBL
University Of Bradford
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH3A1 assessed as reduction in NADPH production using 4-NBA and NADP+ as substrate by fluori...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Bradford
Curated by ChEMBL
University Of Bradford
Curated by ChEMBL
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH1A3 assessed as reduction in NADH production using hexanal and NAD+ as substrate by fluori...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Bradford
Curated by ChEMBL
University Of Bradford
Curated by ChEMBL
Affinity DataIC50: 1.07E+4nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH1A3 assessed as reduction in NADH production using hexanal and NAD+ as substrate by fluori...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Homo sapiens (Human))
University Of Bradford
Curated by ChEMBL
University Of Bradford
Curated by ChEMBL
Affinity DataIC50: 1.37E+4nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH3A1 assessed as reduction in NADPH production using 4-NBA and NADP+ as substrate by fluori...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Homo sapiens (Human))
University Of Bradford
Curated by ChEMBL
University Of Bradford
Curated by ChEMBL
Affinity DataIC50: 6.41E+4nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH3A1 assessed as reduction in NADPH production using 4-NBA and NADP+ as substrate by fluori...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Bradford
Curated by ChEMBL
University Of Bradford
Curated by ChEMBL
Affinity DataIC50: 1.06E+5nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH1A3 assessed as reduction in NADH production using hexanal and NAD+ as substrate by fluori...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csir-Central Drug Research Institute (Csir-Cdri)
Curated by ChEMBL
Csir-Central Drug Research Institute (Csir-Cdri)
Curated by ChEMBL
Affinity DataEC50: 38nMAssay Description:Positive allosteric modulation of 5HT2A receptor (unknown origin) expressed in HEK293 cells co-expressing NFAT-RE assessed as increase in serotonin-i...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csir-Central Drug Research Institute (Csir-Cdri)
Curated by ChEMBL
Csir-Central Drug Research Institute (Csir-Cdri)
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Positive allosteric modulation of 5HT2B receptor (unknown origin) expressed in HEK293 cells co-expressing NFAT-RE assessed as increase in serotonin-i...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csir-Central Drug Research Institute (Csir-Cdri)
Curated by ChEMBL
Csir-Central Drug Research Institute (Csir-Cdri)
Curated by ChEMBL
Affinity DataEC50: 1.30nMAssay Description:Positive allosteric modulation of 5HT2B receptor (unknown origin) expressed in HEK293 cells co-expressing NFAT-RE assessed as increase in serotonin-i...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csir-Central Drug Research Institute (Csir-Cdri)
Curated by ChEMBL
Csir-Central Drug Research Institute (Csir-Cdri)
Curated by ChEMBL
Affinity DataEC50: 4.20nMAssay Description:Positive allosteric modulation of 5HT2C receptor (unknown origin) expressed in HEK293 cells co-expressing NFAT-RE assessed as increase in serotonin-i...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csir-Central Drug Research Institute (Csir-Cdri)
Curated by ChEMBL
Csir-Central Drug Research Institute (Csir-Cdri)
Curated by ChEMBL
Affinity DataEC50: 4.30nMAssay Description:Positive allosteric modulation of 5HT2C receptor (unknown origin) expressed in HEK293 cells co-expressing NFAT-RE assessed as increase in serotonin-i...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csir-Central Drug Research Institute (Csir-Cdri)
Curated by ChEMBL
Csir-Central Drug Research Institute (Csir-Cdri)
Curated by ChEMBL
Affinity DataEC50: 1.30nMAssay Description:Positive allosteric modulation of 5HT2B receptor (unknown origin) expressed in HEK293 cells co-expressing NFAT-RE assessed as increase in serotonin-i...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csir-Central Drug Research Institute (Csir-Cdri)
Curated by ChEMBL
Csir-Central Drug Research Institute (Csir-Cdri)
Curated by ChEMBL
Affinity DataEC50: 46nMAssay Description:Positive allosteric modulation of 5HT2A receptor (unknown origin) expressed in HEK293 cells co-expressing NFAT-RE assessed as increase in serotonin-i...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csir-Central Drug Research Institute (Csir-Cdri)
Curated by ChEMBL
Csir-Central Drug Research Institute (Csir-Cdri)
Curated by ChEMBL
Affinity DataEC50: 5nMAssay Description:Positive allosteric modulation of 5HT2C receptor (unknown origin) expressed in HEK293 cells co-expressing NFAT-RE assessed as increase in serotonin-i...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csir-Central Drug Research Institute (Csir-Cdri)
Curated by ChEMBL
Csir-Central Drug Research Institute (Csir-Cdri)
Curated by ChEMBL
Affinity DataEC50: 50nMAssay Description:Positive allosteric modulation of 5HT2A receptor (unknown origin) expressed in HEK293 cells co-expressing NFAT-RE assessed as increase in serotonin-i...More data for this Ligand-Target Pair