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Found 82 with Last Name = 'nomura' and Initial = 'w'
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50286290(CHEMBL4174314)
Affinity DataIC50:  0.497nMAssay Description:Inhibition of vitronectin binding to integrin alphaVbeta3 in HDF pretreated for 20 mins followed by vitronectin addition measured after 40 mins by cr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Tokyo Medical And Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50517802(CHEMBL4457992)
Affinity DataIC50:  1.60nMAssay Description:Competitive inhibition of TAMRAAc-TZ14011 binding to CXCR4 (unknown origin) expressed in CHO cells in presence of ZnCl2 by NanoBRET assay relative to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50286289(CHEMBL4166054)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of vitronectin binding to human integrin alphaVbeta3 measured after 4 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Tokyo Medical And Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50517800(CHEMBL4451705)
Affinity DataIC50:  3.5nMAssay Description:Competitive inhibition of TAMRAAc-TZ14011 binding to CXCR4 (unknown origin) expressed in CHO cells in presence of ZnCl2 by NanoBRET assay relative to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50286288(CHEMBL4159636)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of vitronectin binding to human integrin alphaVbeta3 measured after 4 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482161(CHEMBL1082256)
Affinity DataIC50:  4nMAssay Description:Inhibition of HIV1 integrase strand transfer activity after 1 hr by densitometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Tokyo Medical And Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50517803(CHEMBL4529751)
Affinity DataIC50:  4.5nMAssay Description:Competitive inhibition of TAMRAAc-TZ14011 binding to CXCR4 (unknown origin) expressed in CHO cells in presence of ZnCl2 by NanoBRET assay relative to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482160(CHEMBL1082257)
Affinity DataIC50:  5nMAssay Description:Inhibition of HIV1 integrase strand transfer activity after 1 hr by densitometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Tokyo Medical And Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50517804(CHEMBL4548792)
Affinity DataIC50:  5.70nMAssay Description:Competitive inhibition of TAMRAAc-TZ14011 binding to CXCR4 (unknown origin) expressed in CHO cells in presence of ZnCl2 by NanoBRET assay relative to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482160(CHEMBL1082257)
Affinity DataIC50:  6nMAssay Description:Inhibition of HIV1 integrase 3'-end processing activity after 1 hr by densitometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50237601(CHEMBL411941 | CycloRGDfV | [(2S,5R,8S,11S)-5-Benz...)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of vitronectin binding to human integrin alphaVbeta3 measured after 4 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Tokyo Medical And Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50517798(CHEMBL4568686)
Affinity DataIC50:  7.90nMAssay Description:Competitive inhibition of TAMRAAc-TZ14011 binding to CXCR4 (unknown origin) expressed in CHO cells in presence of ZnCl2 by NanoBRET assay relative to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482161(CHEMBL1082256)
Affinity DataIC50:  8nMAssay Description:Inhibition of HIV1 integrase 3'-end processing activity after 1 hr by densitometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482699(CHEMBL1241174)
Affinity DataIC50:  10nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Tokyo Medical And Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50517799(CHEMBL4531581)
Affinity DataIC50:  10nMAssay Description:Competitive inhibition of TAMRAAc-TZ14011 binding to CXCR4 (unknown origin) expressed in CHO cells in presence of ZnCl2 by NanoBRET assay relative to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50237601(CHEMBL411941 | CycloRGDfV | [(2S,5R,8S,11S)-5-Benz...)
Affinity DataIC50:  11nMAssay Description:Inhibition of vitronectin binding to integrin alphaVbeta3 in HDF pretreated for 20 mins followed by vitronectin addition measured after 40 mins by cr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482700(CHEMBL1241178)
Affinity DataIC50:  31nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Tokyo Medical And Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50517801(CHEMBL4532299)
Affinity DataIC50:  32nMAssay Description:Competitive inhibition of TAMRAAc-TZ14011 binding to CXCR4 (unknown origin) expressed in CHO cells in presence of ZnCl2 by NanoBRET assay relative to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482700(CHEMBL1241178)
Affinity DataIC50:  40nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482160(CHEMBL1082257)
Affinity DataIC50:  40nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Tokyo Medical And Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50128522(CHEMBL3627930)
Affinity DataIC50:  44nMAssay Description:Displacement of fluorescently-labeled-TZ14011 from CXCR4 in human Jurkat cells incubated for 30 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482714(CHEMBL1241175)
Affinity DataIC50:  47nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482698(CHEMBL1241173)
Affinity DataIC50:  50nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482710(CHEMBL1241189)
Affinity DataIC50:  50nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482699(CHEMBL1241174)
Affinity DataIC50:  50nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482720(CHEMBL1241183)
Affinity DataIC50:  60nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482161(CHEMBL1082256)
Affinity DataIC50:  60nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482709(CHEMBL1241187)
Affinity DataIC50:  60nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482704(CHEMBL1241184)
Affinity DataIC50:  60nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482703(CHEMBL1241182)
Affinity DataIC50:  60nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482701(CHEMBL1241179)
Affinity DataIC50:  60nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482719(CHEMBL1241176)
Affinity DataIC50:  65nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482712(CHEMBL1241169)
Affinity DataIC50:  70nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482716(CHEMBL1240540)
Affinity DataIC50:  70nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482713(CHEMBL1241172)
Affinity DataIC50:  70nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482702(CHEMBL1241181)
Affinity DataIC50:  80nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482717(CHEMBL1241180)
Affinity DataIC50:  80nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482698(CHEMBL1241173)
Affinity DataIC50:  80nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Tokyo Medical And Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50128523(CHEMBL3628613)
Affinity DataIC50:  86nMAssay Description:Displacement of fluorescently-labeled-TZ14011 from CXCR4 in human Jurkat cells incubated for 30 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482160(CHEMBL1082257)
Affinity DataIC50:  90nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482708(CHEMBL1241191)
Affinity DataIC50:  90nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482708(CHEMBL1241191)
Affinity DataIC50:  90nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482712(CHEMBL1241169)
Affinity DataIC50:  100nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482720(CHEMBL1241183)
Affinity DataIC50:  100nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482711(CHEMBL1241170)
Affinity DataIC50:  110nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482710(CHEMBL1241189)
Affinity DataIC50:  110nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482713(CHEMBL1241172)
Affinity DataIC50:  110nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482697(CHEMBL1241171)
Affinity DataIC50:  110nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482716(CHEMBL1240540)
Affinity DataIC50:  120nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tokyo Medical And Dental University

Curated by ChEMBL
LigandPNGBDBM50482707(CHEMBL1241188)
Affinity DataIC50:  120nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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