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Found 178 with Last Name = 'chirkova' and Initial = 'z'
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50063522(CHEMBL3398531)
Affinity DataKi:  16nMAssay Description:Inhibition of human recombinant MAO-B assessed as kynuramine substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50063522(CHEMBL3398531)
Affinity DataKi:  18nMAssay Description:Inhibition of human recombinant MAO-A assessed as kynuramine substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50503654(CHEMBL4447183)
Affinity DataKi:  38nMAssay Description:Competitive inhibition of human MAOB expressed in insect cell microsomes using varying levels of kynuramine as substrate measured after 20 mins by Li...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50086502(2-BFi | 2-Benzofuran-2-yl-4,5-dihydro-1H-imidazole...)
Affinity DataKi:  8.30E+3nMAssay Description:Competitive inhibition of human MAOB using farnesylamine as substrate preincubated with substrate for 5 mins followed by enzyme addition by fluorimet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50086502(2-BFi | 2-Benzofuran-2-yl-4,5-dihydro-1H-imidazole...)
Affinity DataKi:  1.70E+4nMAssay Description:Competitive inhibition of human MAOA using p-trifluoromethyl benzylamine as substrate preincubated with substrate for 5 mins followed by enzyme addit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50063523(CHEMBL3398530)
Affinity DataIC50:  4nMAssay Description:Inhibition of human recombinant MAO-A assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM86779(Phthalonitrile analogue, 4h)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of human recombinant MAO-B assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM86779(Phthalonitrile analogue, 4h)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of human recombinant MAO-A assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50503651(CHEMBL4582038)
Affinity DataIC50:  12nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50063522(CHEMBL3398531)
Affinity DataIC50:  14nMAssay Description:Inhibition of human recombinant MAO-A assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50063522(CHEMBL3398531)
Affinity DataIC50:  17nMAssay Description:Inhibition of human recombinant MAO-B assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50063523(CHEMBL3398530)
Affinity DataIC50:  20nMAssay Description:Inhibition of human recombinant MAO-B assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50503663(CHEMBL4527539)
Affinity DataIC50:  30nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50503668(CHEMBL4538263)
Affinity DataIC50:  30nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50063517(CHEMBL3398524)
Affinity DataIC50:  35nMAssay Description:Inhibition of human recombinant MAO-A assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM19187((2S)-2-[({4-[(3-fluorophenyl)methoxy]phenyl}methyl...)
Affinity DataIC50:  48nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate measured after 20 mins by fluorescence spectro...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM19187((2S)-2-[({4-[(3-fluorophenyl)methoxy]phenyl}methyl...)
Affinity DataIC50:  48nMAssay Description:Inhibition of human recombinant MAO-B using kynuramine as substrate incubated for 20 mins by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50503664(CHEMBL4459969)
Affinity DataIC50:  64nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50503654(CHEMBL4447183)
Affinity DataIC50:  71nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50029816(5-Chloro-pyridine-2-carboxylic acid (2-amino-ethyl...)
Affinity DataIC50:  91nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate measured after 20 mins by fluorescence spectro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50029816(5-Chloro-pyridine-2-carboxylic acid (2-amino-ethyl...)
Affinity DataIC50:  91nMAssay Description:Inhibition of human recombinant MAO-B using kynuramine as substrate incubated for 20 mins by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50029816(5-Chloro-pyridine-2-carboxylic acid (2-amino-ethyl...)
Affinity DataIC50:  91nMAssay Description:Inhibition of human recombinant MAO-B assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50063521(CHEMBL3398532)
Affinity DataIC50:  118nMAssay Description:Inhibition of human recombinant MAO-A assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50063524(CHEMBL3398529)
Affinity DataIC50:  121nMAssay Description:Inhibition of human recombinant MAO-A assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50063519(CHEMBL3398522)
Affinity DataIC50:  129nMAssay Description:Inhibition of human recombinant MAO-A assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50063520(CHEMBL3398533)
Affinity DataIC50:  142nMAssay Description:Inhibition of human recombinant MAO-A assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50063524(CHEMBL3398529)
Affinity DataIC50:  144nMAssay Description:Inhibition of human recombinant MAO-B assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50501004(CHEMBL3799747)
Affinity DataIC50:  147nMAssay Description:Inhibition of human recombinant MAO-A using kynuramine as substrate incubated for 20 mins by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50503678(CHEMBL4444732)
Affinity DataIC50:  160nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50503661(CHEMBL4463081)
Affinity DataIC50:  216nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50503666(CHEMBL4446092)
Affinity DataIC50:  230nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50501010(CHEMBL3799006)
Affinity DataIC50:  250nMAssay Description:Inhibition of human recombinant MAO-A using kynuramine as substrate incubated for 20 mins by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50503671(CHEMBL4443215)
Affinity DataIC50:  300nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM86776(Phthalonitrile analogue, 4e)
Affinity DataIC50:  399nMAssay Description:Inhibition of human recombinant MAO-A assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50501001(CHEMBL3799754)
Affinity DataIC50:  405nMAssay Description:Inhibition of human recombinant MAO-A using kynuramine as substrate incubated for 20 mins by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50503682(CHEMBL4448928)
Affinity DataIC50:  411nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50501025(CHEMBL3797374)
Affinity DataIC50:  522nMAssay Description:Inhibition of human recombinant MAO-A using kynuramine as substrate incubated for 20 mins by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50501018(CHEMBL3799699)
Affinity DataIC50:  581nMAssay Description:Inhibition of human recombinant MAO-B using kynuramine as substrate incubated for 20 mins by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50503675(CHEMBL4444156)
Affinity DataIC50:  608nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM86776(Phthalonitrile analogue, 4e)
Affinity DataIC50:  642nMAssay Description:Inhibition of human recombinant MAO-B assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50501020(CHEMBL3799798)
Affinity DataIC50:  661nMAssay Description:Inhibition of human recombinant MAO-A using kynuramine as substrate incubated for 20 mins by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50063515(CHEMBL3398526)
Affinity DataIC50:  726nMAssay Description:Inhibition of human recombinant MAO-A assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50503682(CHEMBL4448928)
Affinity DataIC50:  751nMAssay Description:Inhibition of recombinant human MAOA expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50503681(CHEMBL4549955)
Affinity DataIC50:  756nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50501022(CHEMBL3800008)
Affinity DataIC50:  821nMAssay Description:Inhibition of human recombinant MAO-B using kynuramine as substrate incubated for 20 mins by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50503652(CHEMBL4530181)
Affinity DataIC50:  890nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50501028(CHEMBL3798677)
Affinity DataIC50:  923nMAssay Description:Inhibition of human recombinant MAO-B using kynuramine as substrate incubated for 20 mins by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50503667(CHEMBL4476431)
Affinity DataIC50:  1.06E+3nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50503651(CHEMBL4582038)
Affinity DataIC50:  1.11E+3nMAssay Description:Inhibition of recombinant human MAOA expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50501016(CHEMBL3797506)
Affinity DataIC50:  1.13E+3nMAssay Description:Inhibition of human recombinant MAO-A using kynuramine as substrate incubated for 20 mins by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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