TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Inhibition of human recombinant MAO-B assessed as kynuramine substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Inhibition of human recombinant MAO-A assessed as kynuramine substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataKi: 38nMAssay Description:Competitive inhibition of human MAOB expressed in insect cell microsomes using varying levels of kynuramine as substrate measured after 20 mins by Li...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataKi: 8.30E+3nMAssay Description:Competitive inhibition of human MAOB using farnesylamine as substrate preincubated with substrate for 5 mins followed by enzyme addition by fluorimet...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataKi: 1.70E+4nMAssay Description:Competitive inhibition of human MAOA using p-trifluoromethyl benzylamine as substrate preincubated with substrate for 5 mins followed by enzyme addit...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant MAO-A assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 4.80nMAssay Description:Inhibition of human recombinant MAO-B assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 6.60nMAssay Description:Inhibition of human recombinant MAO-A assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of human recombinant MAO-A assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of human recombinant MAO-B assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of human recombinant MAO-B assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of human recombinant MAO-A assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate measured after 20 mins by fluorescence spectro...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:Inhibition of human recombinant MAO-B using kynuramine as substrate incubated for 20 mins by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 64nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 71nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate measured after 20 mins by fluorescence spectro...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Inhibition of human recombinant MAO-B using kynuramine as substrate incubated for 20 mins by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Inhibition of human recombinant MAO-B assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 118nMAssay Description:Inhibition of human recombinant MAO-A assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 121nMAssay Description:Inhibition of human recombinant MAO-A assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 129nMAssay Description:Inhibition of human recombinant MAO-A assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 142nMAssay Description:Inhibition of human recombinant MAO-A assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 144nMAssay Description:Inhibition of human recombinant MAO-B assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 147nMAssay Description:Inhibition of human recombinant MAO-A using kynuramine as substrate incubated for 20 mins by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 216nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of human recombinant MAO-A using kynuramine as substrate incubated for 20 mins by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 399nMAssay Description:Inhibition of human recombinant MAO-A assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 405nMAssay Description:Inhibition of human recombinant MAO-A using kynuramine as substrate incubated for 20 mins by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 411nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 522nMAssay Description:Inhibition of human recombinant MAO-A using kynuramine as substrate incubated for 20 mins by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 581nMAssay Description:Inhibition of human recombinant MAO-B using kynuramine as substrate incubated for 20 mins by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 608nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 642nMAssay Description:Inhibition of human recombinant MAO-B assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 661nMAssay Description:Inhibition of human recombinant MAO-A using kynuramine as substrate incubated for 20 mins by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 726nMAssay Description:Inhibition of human recombinant MAO-A assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 751nMAssay Description:Inhibition of recombinant human MAOA expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 756nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 821nMAssay Description:Inhibition of human recombinant MAO-B using kynuramine as substrate incubated for 20 mins by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 890nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 923nMAssay Description:Inhibition of human recombinant MAO-B using kynuramine as substrate incubated for 20 mins by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 1.06E+3nMAssay Description:Inhibition of recombinant human MAOB expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 1.11E+3nMAssay Description:Inhibition of recombinant human MAOA expressed in insect cell microsomes using kynuramine as substrate preincubated with substrate for 30 mins follow...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University
Curated by ChEMBL
Yaroslavl State Technical University
Curated by ChEMBL
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of human recombinant MAO-A using kynuramine as substrate incubated for 20 mins by fluorescence spectrophotometric analysisMore data for this Ligand-Target Pair