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Found 66 with Last Name = 'Łazewska' and Initial = 'd'
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM22541(Clobenpropit | N''-[(4-chlorophenyl)methyl]{[3-(1H...)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50247055(1-(3-(3-phenylpropoxy)propyl)piperidine | CHEMBL46...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from human histamine H3 receptor expressed in rat C6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM22541(Clobenpropit | N''-[(4-chlorophenyl)methyl]{[3-(1H...)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50311769((S)-3-(1H-imidazol-4-yl)propyl 2-methylbutylcarbam...)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50074076((3-Methyl-pentyl)-carbamic acid 3-(1H-imidazol-4-y...)
Affinity DataKi:  5.10nMAssay Description:Displacement of [3H]histamine from histamine H3 receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50074088((2-Methyl-pentyl)-carbamic acid 3-(1H-imidazol-4-y...)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50074072((1-Methyl-pentyl)-carbamic acid 3-(1H-imidazol-4-y...)
Affinity DataKi:  8.70nMAssay Description:Displacement of [3H]histamine from histamine H3 receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50311768((R)-3-(1H-imidazol-4-yl)propyl pentan-2-ylcarbamat...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]histamine from histamine H3 receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50311765((R)-3-(1H-imidazol-4-yl)propyl sec-butylcarbamate ...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50311772((S)-3-(1H-imidazol-4-yl)propyl hexan-2-ylcarbamate...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]histamine from histamine H3 receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50074076((3-Methyl-pentyl)-carbamic acid 3-(1H-imidazol-4-y...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50311780(3-(1H-imidazol-4-yl)propyl 4-methylpentylcarbamate...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50074088((2-Methyl-pentyl)-carbamic acid 3-(1H-imidazol-4-y...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]histamine from histamine H3 receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50311768((R)-3-(1H-imidazol-4-yl)propyl pentan-2-ylcarbamat...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50311777((S)-3-(1H-imidazol-4-yl)propyl heptan-2-ylcarbamat...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]histamine from histamine H3 receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50074069((1-Methyl-heptyl)-carbamic acid 3-(1H-imidazol-4-y...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]histamine from histamine H3 receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50311769((S)-3-(1H-imidazol-4-yl)propyl 2-methylbutylcarbam...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]histamine from histamine H3 receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50074073((1-Methyl-hexyl)-carbamic acid 3-(1H-imidazol-4-yl...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]histamine from histamine H3 receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50311771((R)-3-(1H-imidazol-4-yl)propyl hexan-2-ylcarbamate...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]histamine from histamine H3 receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50311771((R)-3-(1H-imidazol-4-yl)propyl hexan-2-ylcarbamate...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50311765((R)-3-(1H-imidazol-4-yl)propyl sec-butylcarbamate ...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]histamine from histamine H3 receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50074087(CHEMBL1076266 | CHEMBL157493 | sec-Butyl-carbamic ...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]histamine from histamine H3 receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50074062((1-Methyl-butyl)-carbamic acid 3-(1H-imidazol-4-yl...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50311778((R,S)-3-(1H-imidazol-4-yl)propyl 6-methylheptan-2-...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]histamine from histamine H3 receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50311766((S)-3-(1H-imidazol-4-yl)propyl sec-butylcarbamate ...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]histamine from histamine H3 receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50311776((R)-3-(1H-imidazol-4-yl)propyl heptan-2-ylcarbamat...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]histamine from histamine H3 receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50074062((1-Methyl-butyl)-carbamic acid 3-(1H-imidazol-4-yl...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]histamine from histamine H3 receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50311783((R)-3-(1H-imidazol-4-yl)propyl octan-2-ylcarbamate...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]iodoproxyfan from human histamine H3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50074072((1-Methyl-pentyl)-carbamic acid 3-(1H-imidazol-4-y...)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50311781((R,S)-3-(1H-imidazol-4-yl)propyl 5-methylhexan-2-y...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50311766((S)-3-(1H-imidazol-4-yl)propyl sec-butylcarbamate ...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50311782((R,S)-3-(1H-imidazol-4-yl)propyl 2-ethylhexylcarba...)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50311776((R)-3-(1H-imidazol-4-yl)propyl heptan-2-ylcarbamat...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50311772((S)-3-(1H-imidazol-4-yl)propyl hexan-2-ylcarbamate...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50311784((S)-3-(1H-imidazol-4-yl)propyl octan-2-ylcarbamate...)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]iodoproxyfan from human histamine H3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM22914(CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)pi...)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM27213(4-[3-(4-cyclopropanecarbonylphenoxy)propyl]-1H-imi...)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50074087(CHEMBL1076266 | CHEMBL157493 | sec-Butyl-carbamic ...)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50074073((1-Methyl-hexyl)-carbamic acid 3-(1H-imidazol-4-yl...)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM22914(CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)pi...)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50311777((S)-3-(1H-imidazol-4-yl)propyl heptan-2-ylcarbamat...)
Affinity DataKi:  74nMAssay Description:Displacement of [3H]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50311778((R,S)-3-(1H-imidazol-4-yl)propyl 6-methylheptan-2-...)
Affinity DataKi:  75nMAssay Description:Displacement of [3H]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50074069((1-Methyl-heptyl)-carbamic acid 3-(1H-imidazol-4-y...)
Affinity DataKi:  91nMAssay Description:Displacement of [3H]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50247148(1-[3-(4-tert-Butylphenoxy)propyl]-4-piperidino-pip...)
Affinity DataKi:  100nMAssay Description:Displacement of [125I]iodoproxyfan from human recombinant histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50311769((S)-3-(1H-imidazol-4-yl)propyl 2-methylbutylcarbam...)
Affinity DataKi:  118nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in SF9 cells coexpressing Galphai2, Gbeta1gamma2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50074076((3-Methyl-pentyl)-carbamic acid 3-(1H-imidazol-4-y...)
Affinity DataKi:  123nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in SF9 cells coexpressing Galphai2, Gbeta1gamma2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50247120(1-[2-(3-Methoxyphenoxy)ethyl]-4-piperidino-piperid...)
Affinity DataKi:  132nMAssay Description:Displacement of [125I]iodoproxyfan from human recombinant histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50074088((2-Methyl-pentyl)-carbamic acid 3-(1H-imidazol-4-y...)
Affinity DataKi:  162nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in SF9 cells coexpressing Galphai2, Gbeta1gamma2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50247122(1-[2-(3-Trifluoromethylphenoxy)ethyl]-4-piperidino...)
Affinity DataKi:  164nMAssay Description:Displacement of [125I]iodoproxyfan from human recombinant histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50247125(1-[3-(4-Chlorophenoxy)propyl]-4-piperidino-piperid...)
Affinity DataKi:  165nMAssay Description:Displacement of [125I]iodoproxyfan from human recombinant histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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