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Found 163 with Last Name = 'akimoto' and Initial = 't'
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40787(Des-N-methylcalyculin A (20))
Affinity DataIC50:  1nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40777(Hemicalyculin A (5))
Affinity DataIC50:  1nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)
Affinity DataIC50:  1nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40782(C1/C34-Calyculin A (15))
Affinity DataIC50:  1.10nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40785(Calyculinamide A (18))
Affinity DataIC50:  1.5nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40780(Calyculin A 21-acetate (13))
Affinity DataIC50:  2.10nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40790(Calyculin C (24))
Affinity DataIC50:  2.60nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40785(Calyculinamide A (18))
Affinity DataIC50:  5nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)
Affinity DataIC50:  7.5nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)
Affinity DataIC50:  8.20nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40782(C1/C34-Calyculin A (15))
Affinity DataIC50:  9nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)
Affinity DataIC50:  9nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40787(Des-N-methylcalyculin A (20))
Affinity DataIC50:  11nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40780(Calyculin A 21-acetate (13))
Affinity DataIC50:  13nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40777(Hemicalyculin A (5))
Affinity DataIC50:  14nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)
Affinity DataIC50:  14nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40781(Calyculin J (14))
Affinity DataIC50:  20nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40790(Calyculin C (24))
Affinity DataIC50:  29nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325416((S)-4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyr...)
Affinity DataIC50:  47nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)
Affinity DataIC50:  55nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325375((S)-4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyr...)
Affinity DataIC50:  55nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325371(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridaz...)
Affinity DataIC50:  73nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325370(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridaz...)
Affinity DataIC50:  79nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325415((R)-4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyr...)
Affinity DataIC50:  100nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40781(Calyculin J (14))
Affinity DataIC50:  105nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325418((S)-4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyr...)
Affinity DataIC50:  110nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)
Affinity DataIC50:  112nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325417((S)-4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyr...)
Affinity DataIC50:  140nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325414((R)-(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]py...)
Affinity DataIC50:  160nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)
Affinity DataIC50:  185nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325368((S)-4-(6-(3-chlorobenzylamino)imidazo[1,2-b]pyrida...)
Affinity DataIC50:  190nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325369(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridaz...)
Affinity DataIC50:  200nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325403((S)-4-(6-(cyclopropylamino)imidazo[1,2-b]pyridazin...)
Affinity DataIC50:  200nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325402((S)-4-(6-(isopropylamino)imidazo[1,2-b]pyridazin-3...)
Affinity DataIC50:  270nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325412(CHEMBL1223206 | N-(2-aminopropyl)-4-(6-(cyclopropy...)
Affinity DataIC50:  310nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325374((S)-4-(6-(3,4-dichlorobenzylamino)imidazo[1,2-b]py...)
Affinity DataIC50:  320nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325404((S)-4-(6-(benzylamino)imidazo[1,2-b]pyridazin-3-yl...)
Affinity DataIC50:  330nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325411(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridaz...)
Affinity DataIC50:  330nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325366((S)-4-(6-(3-(1H-imidazol-1-yl)propylamino)imidazo[...)
Affinity DataIC50:  380nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325367(CHEMBL1223136 | trans-4-(6-(4-hydroxycyclohexylami...)
Affinity DataIC50:  530nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325406((S)-4-(6-(3-hydroxypropylamino)imidazo[1,2-b]pyrid...)
Affinity DataIC50:  550nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325373(4-(6-(3,4-dichlorobenzylamino)imidazo[1,2-b]pyrida...)
Affinity DataIC50:  590nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325372(4-(6-(3,4-dichlorobenzylamino)imidazo[1,2-b]pyrida...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325401((S)-4-(6-(methylamino)imidazo[1,2-b]pyridazin-3-yl...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325393((4-(6-(3,4-dichlorobenzylamino)imidazo[1,2-b]pyrid...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296234((-)-epigallocatechin-3-(3''-O-methyl)gallate | (2R...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human recombinant MT1-MMP expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325391(4-(6-(3,4-dichlorobenzylamino)imidazo[1,2-b]pyrida...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325374((S)-4-(6-(3,4-dichlorobenzylamino)imidazo[1,2-b]py...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of recombinant IKKalpha after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325380(4-(6-(3,4-dichlorobenzylamino)imidazo[1,2-b]pyrida...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325377(4-(6-(3,4-dichlorobenzylamino)imidazo[1,2-b]pyrida...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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