Affinity DataKi: 0.160nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.480nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in rat brain synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.720nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in rat brain synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.840nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.930nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in rat brain synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.970nMAssay Description:Displacement of [3H]CP55940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University of Connecticut
US Patent
University of Connecticut
US Patent
Affinity DataKi: 1nM ΔG°: -53.4kJ/mole IC50: 15nMT: 2°CAssay Description:All compound solutions are made to a concentration of 10 mM in DMSO. To test the stability of the compounds in enzyme assay conditions, 25 nmoles of ...More data for this Ligand-Target Pair
Affinity DataKi: 1.03nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.13nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.23nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.32nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.37nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in rat brain synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in rat brain synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]CP55940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.62nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.63nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.67nMAssay Description:Displacement of [3H]CP55940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.76nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]CP55940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University of Connecticut
US Patent
University of Connecticut
US Patent
Affinity DataKi: 2nM ΔG°: -51.6kJ/mole IC50: 21nMT: 2°CAssay Description:All compound solutions are made to a concentration of 10 mM in DMSO. To test the stability of the compounds in enzyme assay conditions, 25 nmoles of ...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University of Connecticut
US Patent
University of Connecticut
US Patent
Affinity DataKi: 2nM ΔG°: -51.6kJ/mole IC50: 25nMT: 2°CAssay Description:All compound solutions are made to a concentration of 10 mM in DMSO. To test the stability of the compounds in enzyme assay conditions, 25 nmoles of ...More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.33nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.59nMAssay Description:Displacement of [3H]CP55940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in rat brain synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.76nMAssay Description:Displacement of [3H]CP55940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.78nMAssay Description:Displacement of [3H]CP55940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University of Connecticut
US Patent
University of Connecticut
US Patent
Affinity DataKi: 3nM ΔG°: -50.6kJ/mole IC50: 39nMT: 2°CAssay Description:All compound solutions are made to a concentration of 10 mM in DMSO. To test the stability of the compounds in enzyme assay conditions, 25 nmoles of ...More data for this Ligand-Target Pair
Affinity DataKi: 3.02nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.14nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.34nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in rat brain synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 4.21nMAssay Description:Displacement of [3H]CP55940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.51nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.90nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 4.96nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.13nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.25nMAssay Description:Displacement of [3H]CP55940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.88nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University of Connecticut
US Patent
University of Connecticut
US Patent
Affinity DataKi: 6nM ΔG°: -48.8kJ/mole IC50: 100nMT: 2°CAssay Description:All compound solutions are made to a concentration of 10 mM in DMSO. To test the stability of the compounds in enzyme assay conditions, 25 nmoles of ...More data for this Ligand-Target Pair
Affinity DataKi: 6.57nMAssay Description:Displacement of [3H]CP55940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University of Connecticut
US Patent
University of Connecticut
US Patent
Affinity DataKi: 7nM ΔG°: -48.4kJ/mole IC50: 24nMT: 2°CAssay Description:All compound solutions are made to a concentration of 10 mM in DMSO. To test the stability of the compounds in enzyme assay conditions, 25 nmoles of ...More data for this Ligand-Target Pair
Affinity DataKi: 7.02nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.56nMAssay Description:Displacement of [3H]CP55940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair