Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor expressed in CHO -K1 cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.560nMAssay Description:Displacement of [3H]Spiperone from dopamine D2 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 0.580nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor expressed in CHO -K1 cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.950nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor expressed in CHO -K1 cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.39nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor expressed in CHO -K1 cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Inhibitory activity against calf spleen purine nucleoside phosphorylase (PNP) using 2-amino-6-mercapto-7-methyl purine ribonucleoside (MESG) as subst...More data for this Ligand-Target Pair
Affinity DataKi: 1.91nMAssay Description:Antagonist activity at 5HT1AMore data for this Ligand-Target Pair
Affinity DataKi: 2.26nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor expressed in CHO -K1 cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.51nMAssay Description:Antagonist activity at 5HT1AMore data for this Ligand-Target Pair
Affinity DataKi: 2.69nMAssay Description:Antagonist activity at 5HT1AMore data for this Ligand-Target Pair
Affinity DataKi: 3.02nMAssay Description:Antagonist activity at 5HT1AMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Inhibitory activity against calf spleen purine nucleoside phosphorylase (PNP) using 2-amino-6-mercapto-7-methyl purine ribonucleoside (MESG) as subst...More data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Inhibitory activity against calf spleen purine nucleoside phosphorylase (PNP) using 2-amino-6-mercapto-7-methyl purine ribonucleoside (MESG) as subst...More data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Inhibitory activity against calf spleen purine nucleoside phosphorylase (PNP) using 2-amino-6-mercapto-7-methyl purine ribonucleoside (MESG) as subst...More data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Inhibitory activity against calf spleen purine nucleoside phosphorylase (PNP) using 2-amino-6-mercapto-7-methyl purine ribonucleoside (MESG) as subst...More data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Displacement of [3H]spiperone from human D2 DA receptor expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Inhibitory activity of the compound against calf spleen Purine nucleoside phosphorylase (PNP) using 2-amino-6-mercapto-7-methyl purine ribonucleoside...More data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Inhibitory activity against calf spleen purine nucleoside phosphorylase (PNP) using 2-amino-6-mercapto-7-methyl purine ribonucleoside (MESG) as subst...More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibitory activity against calf spleen purine nucleoside phosphorylase (PNP) using inosine as substrate at a concentration of 10 uM.More data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Inhibitory activity against calf spleen purine nucleoside phosphorylase (PNP) using 2-amino-6-mercapto-7-methyl purine ribonucleoside (MESG) as subst...More data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Inhibitory activity against calf spleen purine nucleoside phosphorylase (PNP) using 2-amino-6-mercapto-7-methyl purine ribonucleoside (MESG) as subst...More data for this Ligand-Target Pair
Affinity DataKi: 4.73nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor expressed in CHO -K1 cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Inhibitory activity against calf spleen purine nucleoside phosphorylase (PNP) using 2-amino-6-mercapto-7-methyl purine ribonucleoside (MESG) as subst...More data for this Ligand-Target Pair
Affinity DataKi: 5.49nMAssay Description:Displacement of [3H]Spiperone from dopamine D2 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 5.77nMAssay Description:Displacement of [3H]Spiperone from dopamine D2 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 5.78nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor expressed in CHO -K1 cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Inhibitory activity against calf spleen purine nucleoside phosphorylase (PNP) using 2-amino-6-mercapto-7-methyl purine ribonucleoside (MESG) as subst...More data for this Ligand-Target Pair
Affinity DataKi: 6.03nMAssay Description:Antagonist activity at 5HT1AMore data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Inhibitory activity against calf spleen purine nucleoside phosphorylase (PNP) using 2-amino-6-mercapto-7-methyl purine ribonucleoside (MESG) as subst...More data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Inhibitory activity against calf spleen purine nucleoside phosphorylase (PNP) using 2-amino-6-mercapto-7-methyl purine ribonucleoside (MESG) as subst...More data for this Ligand-Target Pair
Affinity DataKi: 6.46nMAssay Description:Antagonist activity at 5HT1AMore data for this Ligand-Target Pair
Affinity DataKi: 7.53nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor expressed in CHO -K1 cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 7.59nMAssay Description:Antagonist activity at 5HT1AMore data for this Ligand-Target Pair
Affinity DataKi: 8.20nMAssay Description:Displacement of [3H]spiperone from human D2 DA receptor expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 8.5nMAssay Description:Inhibitory activity against calf spleen purine nucleoside phosphorylase (PNP) using inosine as substrate at a concentration of 10 uM.More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Inhibitory activity against calf spleen purine nucleoside phosphorylase (PNP) using inosine as substrate at a concentration of 10 uM.More data for this Ligand-Target Pair
Affinity DataKi: 9.10nMAssay Description:Inhibitory activity against calf spleen purine nucleoside phosphorylase (PNP) using inosine as substrate at a concentration of 10 uM.More data for this Ligand-Target Pair
Affinity DataKi: 9.33nMAssay Description:Antagonist activity at 5HT1AMore data for this Ligand-Target Pair
Affinity DataKi: 9.40nMAssay Description:Inhibitory activity against calf spleen purine nucleoside phosphorylase (PNP) using inosine as substrate at a concentration of 10 uM.More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Antagonist activity at 5HT1AMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Antagonist activity at 5HT1AMore data for this Ligand-Target Pair
Affinity DataKi: 10.2nMAssay Description:Antagonist activity at 5HT1AMore data for this Ligand-Target Pair
Affinity DataKi: 10.6nMAssay Description:Inhibitory activity against calf spleen purine nucleoside phosphorylase (PNP) using inosine as substrate at a concentration of 10 uM.More data for this Ligand-Target Pair
Affinity DataKi: 10.9nMAssay Description:Inhibitory activity against calf spleen purine nucleoside phosphorylase (PNP) using inosine as substrate at a concentration of 10 uM.More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibitory activity against calf spleen purine nucleoside phosphorylase (PNP) using inosine as substrate at a concentration of 10 uM.More data for this Ligand-Target Pair
Affinity DataKi: 11.4nMAssay Description:Inhibitory activity against calf spleen purine nucleoside phosphorylase (PNP) using inosine as substrate at a concentration of 10 uM.More data for this Ligand-Target Pair
Affinity DataKi: 12.0nMAssay Description:Antagonist activity at 5HT1AMore data for this Ligand-Target Pair
Affinity DataKi: 12.9nMAssay Description:Antagonist activity at 5HT1AMore data for this Ligand-Target Pair
Affinity DataKi: 13.1nMAssay Description:Displacement of [3H]Spiperone from dopamine D2 receptor in bovine caudate nuclei synaptosomal membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 13.2nMAssay Description:Inhibitory activity against calf spleen purine nucleoside phosphorylase (PNP) using inosine as substrate at a concentration of 10 uM.More data for this Ligand-Target Pair