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Found 192 with Last Name = 'antoni' and Initial = 'f'
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164588(1-[1-(2-Chloro-phenyl)-cyclopropyl]-6-fluoro-2-met...)
Affinity DataKi:  0.180nMAssay Description:Inhibitory constant for Dopamine receptor D1-likeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM82247(8-Chloro-3-methyl-5-phenyl-2,3,4,5-tetrahydro-1H-b...)
Affinity DataKi:  8.10nMAssay Description:Inhibitory constant for [3H]SCH-23390 binding to Dopamine receptor D1-like of porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Bari

Curated by ChEMBL
LigandPNGBDBM50292901(CHEMBL454373 | N-(3-((4'-(trifluoromethyl)biphenyl...)
Affinity DataKi:  57nMAssay Description:Inhibition of human factor 10a by amydolitic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Bari

Curated by ChEMBL
LigandPNGBDBM50292898(CHEMBL453387 | N-(3-((3',5'-difluorobiphenyl-4-yl)...)
Affinity DataKi:  130nMAssay Description:Inhibition of human factor 10a by amydolitic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164591(((1R,2R)-5-Fluoro-6-methoxy-1-phenyl-indan-2-yl)-d...)
Affinity DataKi:  170nMAssay Description:Inhibitory constant for [3H]YM-09151-2 binding to Dopamine receptor D2-like in porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Bari

Curated by ChEMBL
LigandPNGBDBM50292892(CHEMBL490298 | N-{3-[(3'-fluoro-1,1'-biphenyl-4-yl...)
Affinity DataKi:  177nMAssay Description:Inhibition of human factor 10a by amydolitic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164580((1R,2R)-6-Fluoro-2-(methyl-propyl-amino)-1-phenyl-...)
Affinity DataKi:  240nMAssay Description:Inhibitory constant for [3H]YM-09151-2 binding to Dopamine receptor D2-like in porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164593(((1R,2R)-6-Fluoro-5-methoxy-1-phenyl-indan-2-yl)-m...)
Affinity DataKi:  270nMAssay Description:Inhibitory constant for [3H]YM-09151-2 binding to Dopamine receptor D2-like in porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164604(Allyl-((1R,2R)-6-fluoro-5-methoxy-1-phenyl-indan-2...)
Affinity DataKi:  310nMAssay Description:Inhibitory constant for [3H]YM-09151-2 binding to Dopamine receptor D2-like in porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164605(((1R,2R)-5-Fluoro-6-methoxy-1-phenyl-indan-2-yl)-m...)
Affinity DataKi:  480nMAssay Description:Inhibitory constant for [3H]YM-09151-2 binding to Dopamine receptor D2-like in porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Bari

Curated by ChEMBL
LigandPNGBDBM50292894(CHEMBL490491 | N-(3-((2',4'-difluorobiphenyl-4-yl)...)
Affinity DataKi:  512nMAssay Description:Inhibition of human factor 10a by amydolitic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Bari

Curated by ChEMBL
LigandPNGBDBM50292895(CHEMBL489694 | N-(3-((2',3'-difluorobiphenyl-4-yl)...)
Affinity DataKi:  548nMAssay Description:Inhibition of human factor 10a by amydolitic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164595(((1R,2R)-6-Fluoro-5-methoxy-1-phenyl-indan-2-yl)-d...)
Affinity DataKi:  550nMAssay Description:Inhibitory constant for [3H]YM-09151-2 binding to Dopamine receptor D2-like in porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164598((1R,2R)-2-(Allyl-methyl-amino)-6-fluoro-1-phenyl-i...)
Affinity DataKi:  640nMAssay Description:Inhibitory constant for [3H]YM-09151-2 binding to Dopamine receptor D2-like in porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164587(Allyl-((1R,2R)-5-fluoro-6-methoxy-1-phenyl-indan-2...)
Affinity DataKi:  640nMAssay Description:Inhibitory constant for [3H]YM-09151-2 binding to Dopamine receptor D2-like in porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164590((2R,3R)-6-Fluoro-2-(methyl-propyl-amino)-3-phenyl-...)
Affinity DataKi:  650nMAssay Description:Inhibitory constant for [3H]YM-09151-2 binding to Dopamine receptor D2-like in porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Bari

Curated by ChEMBL
LigandPNGBDBM50292900(CHEMBL508488 | N-(3-((3',4',5'-trifluorobiphenyl-4...)
Affinity DataKi:  666nMAssay Description:Inhibition of human factor 10a by amydolitic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Bari

Curated by ChEMBL
LigandPNGBDBM50292893(CHEMBL524125 | N-(3-((2'-fluorobiphenyl-4-yl)metho...)
Affinity DataKi:  767nMAssay Description:Inhibition of human factor 10a by amydolitic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164586((2R,3R)-2-Dipropylamino-6-fluoro-3-phenyl-indan-5-...)
Affinity DataKi:  920nMAssay Description:Inhibitory constant for [3H]YM-09151-2 binding to Dopamine receptor D2-like in porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164596((2R,3R)-2-(Allyl-methyl-amino)-6-fluoro-3-phenyl-i...)
Affinity DataKi:  960nMAssay Description:Inhibitory constant for [3H]YM-09151-2 binding to Dopamine receptor D2-like in porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Bari

Curated by ChEMBL
LigandPNGBDBM50292887(CHEMBL491672 | N-{[3-(1,1'-biphenyl-4-yl)methoxy]p...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of human factor 10a by amydolitic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM84637(CAS_85760-74-3 | CHEMBL240773 | NSC_54562 | QUINPI...)
Affinity DataKi:  1.26E+3nMAssay Description:Inhibitory constant for [3H]YM-09151-2 binding to Dopamine receptor D2-like in porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Bari

Curated by ChEMBL
LigandPNGBDBM50292896(CHEMBL508759 | N-(3-((2',5'-difluorobiphenyl-4-yl)...)
Affinity DataKi:  1.27E+3nMAssay Description:Inhibition of human factor 10a by amydolitic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Bari

Curated by ChEMBL
LigandPNGBDBM50292897(CHEMBL455203 | N-(3-((2',6'-difluorobiphenyl-4-yl)...)
Affinity DataKi:  1.45E+3nMAssay Description:Inhibition of human factor 10a by amydolitic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164603(((1R,2R)-5-Fluoro-6-methoxy-1-phenyl-indan-2-yl)-d...)
Affinity DataKi:  1.90E+3nMAssay Description:Inhibitory constant for [3H]YM-09151-2 binding to Dopamine receptor D2-like in porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Bari

Curated by ChEMBL
LigandPNGBDBM50292886(CHEMBL491283 | N-(3-(biphenyl-4-ylmethoxy)phenyl)-...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of human factor 10a by amydolitic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM55121(3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...)
Affinity DataKi:  2.44E+3nMAssay Description:Inhibitory constant for [3H]SCH-23390 binding to Dopamine receptor D1-like of porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Bari

Curated by ChEMBL
LigandPNGBDBM50292884(CHEMBL523099 | N-(3-(biphenyl-4-ylmethoxy)phenyl)p...)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibition of human factor 10a by amydolitic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164599(((1R,2R)-5-Fluoro-6-methoxy-1-phenyl-indan-2-yl)-m...)
Affinity DataKi:  2.60E+3nMAssay Description:Inhibitory constant for [3H]YM-09151-2 binding to Dopamine receptor D2-like in porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164592(((1R,2R)-6-Fluoro-5-methoxy-1-phenyl-indan-2-yl)-m...)
Affinity DataKi:  3.10E+3nMAssay Description:Inhibitory constant for [3H]YM-09151-2 binding to Dopamine receptor D2-like in porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM55121(3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...)
Affinity DataKi:  3.31E+3nMAssay Description:Inhibitory constant for [3H]YM-09151-2 binding to Dopamine receptor D2-like in porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCoagulation factor X(Homo sapiens (Human))
University Of Bari

Curated by ChEMBL
LigandPNGBDBM50292891(CHEMBL490297 | N-(3-((4'-fluorobiphenyl-4-yl)metho...)
Affinity DataKi:  3.87E+3nMAssay Description:Inhibition of human factor 10a by amydolitic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164583((1R,2R)-6-Fluoro-2-methylamino-1-phenyl-indan-5-ol...)
Affinity DataKi:  4.30E+3nMAssay Description:Inhibitory constant for [3H]YM-09151-2 binding to Dopamine receptor D2-like in porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164589(((1R,2R)-6-Fluoro-5-methoxy-1-phenyl-indan-2-yl)-d...)
Affinity DataKi:  4.30E+3nMAssay Description:Inhibitory constant for [3H]YM-09151-2 binding to Dopamine receptor D2-like in porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164581((2R,3R)-2-Dimethylamino-6-fluoro-3-phenyl-indan-5-...)
Affinity DataKi:  4.50E+3nMAssay Description:Inhibitory constant for [3H]YM-09151-2 binding to Dopamine receptor D2-like in porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164584((2R,3R)-6-Fluoro-2-methylamino-3-phenyl-indan-5-ol...)
Affinity DataKi:  5.10E+3nMAssay Description:Inhibitory constant for [3H]YM-09151-2 binding to Dopamine receptor D2-like in porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Bari

Curated by ChEMBL
LigandPNGBDBM50292890(CHEMBL489110 | N-(3-(biphenyl-4-ylmethoxy)phenyl)-...)
Affinity DataKi:  5.20E+3nMAssay Description:Inhibition of human factor 10a by amydolitic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164600((1R,2R)-2-Dimethylamino-6-fluoro-1-phenyl-indan-5-...)
Affinity DataKi:  5.90E+3nMAssay Description:Inhibitory constant for [3H]SCH-23390 binding to Dopamine receptor D1-like of porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164583((1R,2R)-6-Fluoro-2-methylamino-1-phenyl-indan-5-ol...)
Affinity DataKi:  7.20E+3nMAssay Description:Inhibitory constant for [3H]SCH-23390 binding to Dopamine receptor D1-like of porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164589(((1R,2R)-6-Fluoro-5-methoxy-1-phenyl-indan-2-yl)-d...)
Affinity DataKi:  7.60E+3nMAssay Description:Inhibitory constant for [3H]SCH-23390 binding to Dopamine receptor D1-like of porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164581((2R,3R)-2-Dimethylamino-6-fluoro-3-phenyl-indan-5-...)
Affinity DataKi:  7.70E+3nMAssay Description:Inhibitory constant for [3H]SCH-23390 binding to Dopamine receptor D1-like of porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164602((1R,2R)-2-Amino-6-fluoro-1-phenyl-indan-5-ol; hydr...)
Affinity DataKi:  8.30E+3nMAssay Description:Inhibitory constant for [3H]SCH-23390 binding to Dopamine receptor D1-like of porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164598((1R,2R)-2-(Allyl-methyl-amino)-6-fluoro-1-phenyl-i...)
Affinity DataKi:  9.00E+3nMAssay Description:Inhibitory constant for [3H]SCH-23390 binding to Dopamine receptor D1-like of porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Bari

Curated by ChEMBL
LigandPNGBDBM50292899(CHEMBL453359 | N-(3-((2',4',6'-trifluorobiphenyl-4...)
Affinity DataKi:  9.47E+3nMAssay Description:Inhibition of human factor 10a by amydolitic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164594((2R,3R)-2-Amino-6-fluoro-3-phenyl-indan-5-ol; hydr...)
Affinity DataKi:  9.60E+3nMAssay Description:Inhibitory constant for [3H]SCH-23390 binding to Dopamine receptor D1-like of porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164584((2R,3R)-6-Fluoro-2-methylamino-3-phenyl-indan-5-ol...)
Affinity DataKi:  9.60E+3nMAssay Description:Inhibitory constant for [3H]SCH-23390 binding to Dopamine receptor D1-like of porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164580((1R,2R)-6-Fluoro-2-(methyl-propyl-amino)-1-phenyl-...)
Affinity DataKi:  1.20E+4nMAssay Description:Inhibitory constant for [3H]SCH-23390 binding to Dopamine receptor D1-like of porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164582((1R,2R)-2-Dipropylamino-6-fluoro-1-phenyl-indan-5-...)
Affinity DataKi:  1.20E+4nMAssay Description:Inhibitory constant for [3H]YM-09151-2 binding to Dopamine receptor D2-like in porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164601((1R,2R)-6-Fluoro-5-methoxy-1-phenyl-indan-2-ylamin...)
Affinity DataKi:  1.20E+4nMAssay Description:Inhibitory constant for [3H]YM-09151-2 binding to Dopamine receptor D2-like in porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50164596((2R,3R)-2-(Allyl-methyl-amino)-6-fluoro-3-phenyl-i...)
Affinity DataKi:  1.30E+4nMAssay Description:Inhibitory constant for [3H]SCH-23390 binding to Dopamine receptor D1-like of porcine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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