Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 3.80nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Binding affinity to human progesterone receptor by competitive assayMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 4.60nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Binding affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Displacement of [3H]-dexamethasone from cytosolic fraction of human recombinant glucocorticoid receptor by scintillation counting analysisMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 6.40nMAssay Description:In vitro inhibition of human Coagulation factor X.More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 7.90nMAssay Description:Inhibition of class C beta-lactamase derived from Enterobacter cloacae P99More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]-dexamethasone from cytosolic fraction of human recombinant glucocorticoid receptor by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of [3H]-dexamethasone from cytosolic fraction of human recombinant glucocorticoid receptor by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of [3H]-progesterone from cytosolic fraction of human recombinant progesterone-B receptor by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]-dexamethasone from cytosolic fraction of human recombinant glucocorticoid receptor by scintillation counting analysisMore data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Nippon Roche Research Center
Nippon Roche Research Center
Affinity DataKi: 20nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of [3H]-progesterone from cytosolic fraction of human recombinant progesterone-B receptor by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Displacement of [3H]-dexamethasone from cytosolic fraction of human recombinant glucocorticoid receptor by scintillation counting analysisMore data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Nippon Roche Research Center
Nippon Roche Research Center
Affinity DataKi: 30nM IC50: 30nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Nippon Roche Research Center
Nippon Roche Research Center
Affinity DataKi: 30nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Nippon Roche Research Center
Nippon Roche Research Center
Affinity DataKi: 30nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Nippon Roche Research Center
Nippon Roche Research Center
Affinity DataKi: 30nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Nippon Roche Research Center
Nippon Roche Research Center
Affinity DataKi: 30nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Displacement of [3H]-dexamethasone from cytosolic fraction of human recombinant glucocorticoid receptor by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Displacement of [3H]-dexamethasone from cytosolic fraction of human recombinant glucocorticoid receptor by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Inhibition of GC1 extended spectrum class C beta-lactamaseMore data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Nippon Roche Research Center
Nippon Roche Research Center
Affinity DataKi: 40nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Nippon Roche Research Center
Nippon Roche Research Center
Affinity DataKi: 40nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Displacement of [3H]-dexamethasone from cytosolic fraction of human recombinant glucocorticoid receptor by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 48nMAssay Description:Inhibition of GC1 extended spectrum class C beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:Binding affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Nippon Roche Research Center
Nippon Roche Research Center
Affinity DataKi: 50nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Nippon Roche Research Center
Nippon Roche Research Center
Affinity DataKi: 50nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Nippon Roche Research Center
Nippon Roche Research Center
Affinity DataKi: 50nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Displacement of [3H]-dexamethasone from cytosolic fraction of human recombinant glucocorticoid receptor by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 55nMAssay Description:Displacement of [3H]-dexamethasone from cytosolic fraction of human recombinant glucocorticoid receptor by scintillation counting analysisMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 69nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 69nMAssay Description:Displacement of [3H]-dexamethasone from cytosolic fraction of human recombinant glucocorticoid receptor by scintillation counting analysisMore data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Nippon Roche Research Center
Nippon Roche Research Center
Affinity DataKi: 70nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Nippon Roche Research Center
Nippon Roche Research Center
Affinity DataKi: 70nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Nippon Roche Research Center
Nippon Roche Research Center
Affinity DataKi: 70nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Nippon Roche Research Center
Nippon Roche Research Center
Affinity DataKi: 80nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Nippon Roche Research Center
Nippon Roche Research Center
Affinity DataKi: 90nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Nippon Roche Research Center
Nippon Roche Research Center
Affinity DataKi: 90nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Nippon Roche Research Center
Nippon Roche Research Center
Affinity DataKi: 100nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
Affinity DataKi: 106nMAssay Description:Displacement of [3H]-dexamethasone from cytosolic fraction of human recombinant glucocorticoid receptor by scintillation counting analysisMore data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Nippon Roche Research Center
Nippon Roche Research Center
Affinity DataKi: 110nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 140nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Nippon Roche Research Center
Nippon Roche Research Center
Affinity DataKi: 140nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
Affinity DataKi: 146nMAssay Description:Displacement of [3H]-dexamethasone from cytosolic fraction of human recombinant glucocorticoid receptor by scintillation counting analysisMore data for this Ligand-Target Pair