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Found 23 with Last Name = 'aquino' and Initial = 'tm'
TargetGenome polyprotein(Dengue virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50323197(7''-O-methylamentoflavone | CHEMBL450522 | sotetsu...)
Affinity DataIC50:  160nMAssay Description:Inhibition of DENV NS5/RNA-dependent RNA polymeraseMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCruzipain(Trypanosoma cruzi)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50157741(CHEMBL374508 | E-64 | E64)
Affinity DataIC50:  400nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-Phe-Arg-aminomethylcoumarin as substrate measured after 5 mins by spectrofluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Zika virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50350203(CHEMBL1814771)
Affinity DataIC50:  500nMAssay Description:Inhibition of Zika virus RNA-dependent RNA polymeraseMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50323198(4'''-methylamentoflavone | CHEMBL220745 | podocarp...)
Affinity DataIC50:  750nMAssay Description:Inhibition of DENV NS5/RNA-dependent RNA polymeraseMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Zika virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50601689(CHEMBL5180295)
Affinity DataIC50:  1.13E+3nMAssay Description:Inhibition of Zika virus wild type RNA-dependent RNA polymerase using ATP as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Zika virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM429505(Remdesivir | US20240034730, Compound Remdesivir | ...)
Affinity DataIC50:  1.36E+3nMAssay Description:Inhibition of Zika virus RNA-dependent RNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50601687(CHEMBL5192551)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of full length His-tagged DENV-2 NS5 incubated for 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50601688(CHEMBL5199491)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of full length His-tagged DENV-2 NS5 incubated for 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCruzipain(Trypanosoma cruzi)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50187500(CHEMBL3828526)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-Phe-Arg-aminomethylcoumarin as substrate measured after 5 mins by spectrofluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50300193(2-[3-(1-Benzyl-1H-pyrazol-3-yl)-benzenesulfonylami...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of DENV-2 NS5More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50300193(2-[3-(1-Benzyl-1H-pyrazol-3-yl)-benzenesulfonylami...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of DENV-4 NS5More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGenome polyprotein(Zika virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50478971(2''C-Me-ATP | CHEMBL374931)
Affinity DataIC50:  5.26E+3nMAssay Description:Inhibition of Zika virus RNA-dependent RNA polymerase activityMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Zika virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50601690(CHEMBL2057532)
Affinity DataIC50:  8.92E+3nMAssay Description:Inhibition of Zika virus RNA-dependent RNA polymerase activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus 2)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50525250(CHEMBL4526128)
Affinity DataIC50:  9.61E+3nMAssay Description:Inhibition of DENV-2 DENV2 NS2B-NS3More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCruzipain(Trypanosoma cruzi)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50187498(CHEMBL3828195)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-Phe-Arg-aminomethylcoumarin as substrate measured after 5 mins by spectrofluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50187496(CHEMBL3827174)
Affinity DataIC50:  8.50E+4nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-Phe-Arg-aminomethylcoumarin as substrate measured after 5 mins by spectrofluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50187499(CHEMBL3827125)
Affinity DataIC50:  1.11E+5nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-Phe-Arg-aminomethylcoumarin as substrate measured after 5 mins by spectrofluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50187497(CHEMBL3827864)
Affinity DataIC50:  1.21E+5nMAssay Description:Inhibition of Trypanosoma cruzi cruzain using Z-Phe-Arg-aminomethylcoumarin as substrate measured after 5 mins by spectrofluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50601686(CHEMBL5182967)
Affinity DataIC50:  1.40E+5nMAssay Description:Inhibition of DENV-4 NS5More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetGenome polyprotein(Dengue virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50601685(CHEMBL5205786)
Affinity DataIC50:  2.10E+5nMAssay Description:Inhibition of DENV-4 NS5More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetPolyprotein P1234(Chikungunya virus (strain S27-African prototype) (...)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50450958(CHEMBL4209509)
Affinity DataEC50:  3.20E+3nMAssay Description:Inhibition of Chikungunya virus nsP2 protease infected in African green monkey Vero cells assessed as inhibition of viral-induced cytopathic effect b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolyprotein P1234(Chikungunya virus (strain S27-African prototype) (...)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50450957(CHEMBL3125915)
Affinity DataEC50:  5.00E+3nMAssay Description:Inhibition of Chikungunya virus nsP2 protease infected in African green monkey Vero cells assessed as inhibition of viral-induced cytopathic effect b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus)
Federal University Of Alagoas

Curated by ChEMBL
LigandPNGBDBM50601687(CHEMBL5192551)
Affinity DataKd:  9.10E+3nMAssay Description:Binding affinity to full length His-tagged DENV-2 NS5 assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed