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Found 19 with Last Name = 'arama' and Initial = 'dp'
TargetKallikrein-7(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50073221(CHEMBL3408420)
Affinity DataKi:  2.70E+4nMAssay Description:Competitive inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50073222(CHEMBL3125572)
Affinity DataKi:  5.06E+4nMAssay Description:Competitive inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 4(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50210949(CHEMBL3946523)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of recombinant human HGK using Ulight-FLGFTYVAP as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50073221(CHEMBL3408420)
Affinity DataIC50:  3.35E+4nMAssay Description:Inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 4(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50210945(CHEMBL3955556)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of recombinant human HGK using Ulight-FLGFTYVAP as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50073228(CHEMBL3408421)
Affinity DataIC50:  5.57E+4nMAssay Description:Inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50073222(CHEMBL3125572)
Affinity DataIC50:  5.70E+4nMAssay Description:Inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50073230(CHEMBL3125570)
Affinity DataIC50:  6.80E+4nMAssay Description:Inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50073231(CHEMBL3125571)
Affinity DataIC50:  7.20E+4nMAssay Description:Inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50073229(CHEMBL3408419)
Affinity DataIC50:  8.09E+4nMAssay Description:Inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50073233(CHEMBL3408416)
Affinity DataIC50:  8.39E+4nMAssay Description:Inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50073232(CHEMBL3408410)
Affinity DataIC50:  9.59E+4nMAssay Description:Inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 4(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50210950(CHEMBL3973327)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human HGK using Ulight-FLGFTYVAP as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 4(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50210948(CHEMBL3919199)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human HGK using Ulight-FLGFTYVAP as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 4(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50210947(CHEMBL3125569)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human HGK using Ulight-FLGFTYVAP as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 4(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50210946(CHEMBL3893977)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human HGK using Ulight-FLGFTYVAP as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50073227(CHEMBL3408430)
Affinity DataIC50:  1.25E+5nMAssay Description:Inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50073226(CHEMBL3408439)
Affinity DataIC50:  1.35E+5nMAssay Description:Inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50073224(CHEMBL3408441)
Affinity DataIC50:  1.49E+5nMAssay Description:Inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed