Compile Data Set for Download or QSAR
maximum 50k data
Found 8 with Last Name = 'arcadi' and Initial = 'a'
TargetNeutrophil elastase(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50077014(2-Furan-2-yl-benzo[d][1,3]oxazin-4-one | CHEMBL244...)
Affinity DataKi:  1.78E+3nMAssay Description:pKi against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50077011(2-Phenyl-4H-3,1-benzoxazin-4-one (3) | 2-Phenyl-be...)
Affinity DataKi:  9.55E+3nMAssay Description:pKi against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50077013(2-(6-Methoxy-3,4-dihydro-naphthalen-1-yl)-benzo[d]...)
Affinity DataIC50:  610nMAssay Description:In vitro inhibitory activity against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Dipartimento Di Scienze Fisiche E Chimiche Universit£

Curated by ChEMBL
LigandPNGBDBM50580227(CHEMBL5083277)
Affinity DataIC50:  1.13E+3nMAssay Description:Antagonist activity at recombinant human TRPM8 transfected in HEK293 cells assessed as assessed as inhibition of icilin-induced intracellular calcium...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Dipartimento Di Scienze Fisiche E Chimiche Universit£

Curated by ChEMBL
LigandPNGBDBM50580226(CHEMBL5093646)
Affinity DataIC50:  4.06E+3nMAssay Description:Antagonist activity at recombinant human TRPM8 transfected in HEK293 cells assessed as assessed as inhibition of icilin-induced intracellular calcium...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50077014(2-Furan-2-yl-benzo[d][1,3]oxazin-4-one | CHEMBL244...)
Affinity DataIC50:  5.50E+3nMAssay Description:In vitro inhibitory activity against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50077012(((E)-2-Cyclooct-1-enyl)-benzo[d][1,3]oxazin-4-one ...)
Affinity DataIC50:  7.00E+3nMAssay Description:In vitro inhibitory activity against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50077011(2-Phenyl-4H-3,1-benzoxazin-4-one (3) | 2-Phenyl-be...)
Affinity DataIC50:  1.70E+4nMAssay Description:In vitro inhibitory activity against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed