Compile Data Set for Download or QSAR
maximum 50k data
Found 66 with Last Name = 'arlot' and Initial = 'y'
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50069792((2S)-2-[(2S)-2-acetamido-4-methylpentanamido]-N-[(...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against Calpain I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233094(N-{4-[7-(2-Diethylaminoethoxy)-6-methoxy-quinazoli...)
Affinity DataIC50:  1.30E+3nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233096(Methyl {4-[7-(2-diethylaminoethoxy)-6-methoxy-quin...)
Affinity DataIC50:  1.70E+3nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233106(N-{4-[6-(2-Diethylaminoethoxy)-7-methoxy-quinazoli...)
Affinity DataIC50:  1.70E+3nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233112(N-Cyclohexyl-N'-{4-[7-(2-diethylaminoethoxy)-6...)
Affinity DataIC50:  1.90E+3nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233105(N-{4-[6,7-Dimethoxy-quinazolin-4-ylamino]phenyl}-N...)
Affinity DataIC50:  2.10E+3nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233095(N-{4-[6-(2-Diethylaminoethoxy)-7-methoxy-quinazoli...)
Affinity DataIC50:  2.30E+3nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233110(N-{4-[6-(2-Diethylaminoethoxy)-7-methoxy-quinazoli...)
Affinity DataIC50:  3.40E+3nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233101(N-{4-[6-(2-Diethylaminoethoxy)-7-methoxy-quinazoli...)
Affinity DataIC50:  4.30E+3nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233109(N-{4-[7-(2-Diethylaminoethoxy)-6-methoxy-quinazoli...)
Affinity DataIC50:  5.20E+3nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233114(N-Cyclohexyl-N'-{4-[6-(2-diethylaminoethoxy)-7...)
Affinity DataIC50:  8.20E+3nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233104(N-{4-[7-(2-Diethylaminoethoxy)-6-methoxy-quinazoli...)
Affinity DataIC50:  8.30E+3nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233100(N-{4-[7-(2-Diethylaminoethoxy)-6-methoxy-quinazoli...)
Affinity DataIC50:  9.10E+3nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233098(Ethyl {4-[7-(2-diethylaminoethoxy)-6-methoxy-quina...)
Affinity DataIC50:  9.40E+3nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM5447(CHEMBL939 | GEFITINIB | Iressa | N-(3-Chloro-4-flu...)
Affinity DataIC50:  1.08E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233097(Methyl {4-[6-(2-diethylaminoethoxy)-7-methoxyquina...)
Affinity DataIC50:  1.11E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM50340921(CHEMBL1761927 | N-(4-(6,7-dimethoxyquinazolin-4-yl...)
Affinity DataIC50:  1.47E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM50340944(1-(3-chloro-4-fluorophenyl)-3-(4-(6,7-dimethoxyqui...)
Affinity DataIC50:  1.52E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM4810((3Z)-3-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-...)
Affinity DataIC50:  1.66E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233102(N-{4-[7-(2-Diethylaminoethoxy)-6-methoxy-quinazoli...)
Affinity DataIC50:  1.71E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233099(Ethyl {4-[7-(2-diethylaminoethoxy)-6-methoxyquinaz...)
Affinity DataIC50:  1.86E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233111(N-{4-[6-(2-Diethylaminoethoxy)-7-methoxy-quinazoli...)
Affinity DataIC50:  1.92E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233106(N-{4-[6-(2-Diethylaminoethoxy)-7-methoxy-quinazoli...)
Affinity DataIC50:  2.09E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233103(N-{4-[6-(2-Diethylaminoethoxy)-7-methoxy-quinazoli...)
Affinity DataIC50:  2.15E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233105(N-{4-[6,7-Dimethoxy-quinazolin-4-ylamino]phenyl}-N...)
Affinity DataIC50:  2.22E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233110(N-{4-[6-(2-Diethylaminoethoxy)-7-methoxy-quinazoli...)
Affinity DataIC50:  2.45E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233101(N-{4-[6-(2-Diethylaminoethoxy)-7-methoxy-quinazoli...)
Affinity DataIC50:  2.64E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233097(Methyl {4-[6-(2-diethylaminoethoxy)-7-methoxyquina...)
Affinity DataIC50:  2.67E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233112(N-Cyclohexyl-N'-{4-[7-(2-diethylaminoethoxy)-6...)
Affinity DataIC50:  2.82E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233103(N-{4-[6-(2-Diethylaminoethoxy)-7-methoxy-quinazoli...)
Affinity DataIC50:  2.83E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM50340927(1-(4-(6,7-dimethoxyquinazolin-4-ylamino)phenyl)-3-...)
Affinity DataIC50:  2.87E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM50380447(CHEMBL2018772 | N-{4-[7-(2-Diethylaminoethoxy)-6-m...)
Affinity DataIC50:  2.91E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233099(Ethyl {4-[7-(2-diethylaminoethoxy)-6-methoxyquinaz...)
Affinity DataIC50:  2.92E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233108(N-{4-[6-(2-Diethylaminoethoxy)-7-methoxy-quinazoli...)
Affinity DataIC50:  2.92E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233108(N-{4-[6-(2-Diethylaminoethoxy)-7-methoxy-quinazoli...)
Affinity DataIC50:  2.97E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233113(N-Cyclohexyl-N'-{4-[6,7-dimethoxy-quinazolin-4...)
Affinity DataIC50:  3.04E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM50380468(CHEMBL2018763 | N-{4-[6,7-Dimethoxy-quinazolin-4-y...)
Affinity DataIC50:  3.06E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233104(N-{4-[7-(2-Diethylaminoethoxy)-6-methoxy-quinazoli...)
Affinity DataIC50:  3.07E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM50340921(CHEMBL1761927 | N-(4-(6,7-dimethoxyquinazolin-4-yl...)
Affinity DataIC50:  3.13E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233114(N-Cyclohexyl-N'-{4-[6-(2-diethylaminoethoxy)-7...)
Affinity DataIC50:  3.23E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233102(N-{4-[7-(2-Diethylaminoethoxy)-6-methoxy-quinazoli...)
Affinity DataIC50:  3.32E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233098(Ethyl {4-[7-(2-diethylaminoethoxy)-6-methoxy-quina...)
Affinity DataIC50:  3.42E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM50340930(1-(4-(6,7-dimethoxyquinazolin-4-ylamino)phenyl)-3-...)
Affinity DataIC50:  3.45E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233107(N-{4-[7-(2-Diethylaminoethoxy)-6-methoxy-quinazoli...)
Affinity DataIC50:  3.54E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM50380467(CHEMBL2016600 | N-{4-[6,7-Dimethoxy-quinazolin-4-y...)
Affinity DataIC50:  3.63E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM50380447(CHEMBL2018772 | N-{4-[7-(2-Diethylaminoethoxy)-6-m...)
Affinity DataIC50:  4.03E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233107(N-{4-[7-(2-Diethylaminoethoxy)-6-methoxy-quinazoli...)
Affinity DataIC50:  4.32E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233100(N-{4-[7-(2-Diethylaminoethoxy)-6-methoxy-quinazoli...)
Affinity DataIC50:  4.41E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM233096(Methyl {4-[7-(2-diethylaminoethoxy)-6-methoxy-quin...)
Affinity DataIC50:  4.52E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit?? Lille Nord De France

LigandPNGBDBM50340925(CHEMBL1761931 | Ethyl {4-[6,7-dimethoxy-quinazolin...)
Affinity DataIC50:  4.79E+4nMpH: 7.5Assay Description:Kinase assays were performed in 96-well plates (Multiscreen Durapore, Millipore) using [γ-32P]ATP (Amersham Biosciences) and the synthetic polym...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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