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Found 148 with Last Name = 'aschenbrenner' and Initial = 'a'
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318983(2-((1-(3-(9H-carbazol-4-yloxy)-2-hydroxypropyl)pip...)
Affinity DataKi:  0.100nMAssay Description:Antagonist activity at human adrenergic beta-1 receptor expressed in CHOK1 cells assessed as inhibition of cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318987(1-(9H-carbazol-4-yloxy)-3-(4-(pyridin-3-ylmethyl)p...)
Affinity DataKi:  0.100nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318989((1-(3-(9H-carbazol-4-yloxy)-2-hydroxypropyl)piperi...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318986(1-(9H-carbazol-4-yloxy)-3-(4-(4-methoxybenzyl)pipe...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318988((1-(3-(9H-carbazol-4-yloxy)-2-hydroxypropyl)piperi...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318990((1-(3-(9H-carbazol-4-yloxy)-2-hydroxypropyl)piperi...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318985(1-(9H-carbazol-4-yloxy)-3-(4-benzylpiperidin-1-yl)...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM34143(CHEMBL175835 | E-6837)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318987(1-(9H-carbazol-4-yloxy)-3-(4-(pyridin-3-ylmethyl)p...)
Affinity DataKi:  1nMAssay Description:Antagonist activity at human adrenergic beta-1 receptor expressed in CHOK1 cells assessed as inhibition of cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318979(1-(2-isopropylphenoxy)-3-morpholinopropan-2-ol | C...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318980(1-(2-allylphenoxy)-3-(1-methylpiperidin-4-ylamino)...)
Affinity DataKi:  2.40nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318999(2-((1-(3-(9H-carbazol-4-yloxy)-2-hydroxypropyl)pip...)
Affinity DataKi:  3nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318986(1-(9H-carbazol-4-yloxy)-3-(4-(4-methoxybenzyl)pipe...)
Affinity DataKi:  3.40nMAssay Description:Antagonist activity at human adrenergic beta-1 receptor expressed in CHOK1 cells assessed as inhibition of cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318999(2-((1-(3-(9H-carbazol-4-yloxy)-2-hydroxypropyl)pip...)
Affinity DataKi:  7nMAssay Description:Antagonist activity at human adrenergic beta-1 receptor expressed in CHOK1 cells assessed as inhibition of cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318978(1-(2-allylphenoxy)-3-morpholinopropan-2-ol | CHEMB...)
Affinity DataKi:  7nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318983(2-((1-(3-(9H-carbazol-4-yloxy)-2-hydroxypropyl)pip...)
Affinity DataKi:  8nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50223292(CHEMBL249034 | N-(4-chlorobenzyl)-2-nitro-5-(piper...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318977(1-((1-(2-hydroxy-3-(2-isopropylphenoxy)propyl)pipe...)
Affinity DataKi:  9nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50223281(5-(4-methylpiperazin-1-yl)-2-nitro-N-(1-phenylethy...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318979(1-(2-isopropylphenoxy)-3-morpholinopropan-2-ol | C...)
Affinity DataKi:  12nMAssay Description:Antagonist activity at human adrenergic beta-1 receptor expressed in CHOK1 cells assessed as inhibition of cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318989((1-(3-(9H-carbazol-4-yloxy)-2-hydroxypropyl)piperi...)
Affinity DataKi:  13nMAssay Description:Antagonist activity at human adrenergic beta-1 receptor expressed in CHOK1 cells assessed as inhibition of cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50319004(2-(1-(2-hydroxy-3-(2-isopropylphenoxy)propyl)piper...)
Affinity DataKi:  13nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318985(1-(9H-carbazol-4-yloxy)-3-(4-benzylpiperidin-1-yl)...)
Affinity DataKi:  14nMAssay Description:Antagonist activity at human adrenergic beta-1 receptor expressed in CHOK1 cells assessed as inhibition of cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318988((1-(3-(9H-carbazol-4-yloxy)-2-hydroxypropyl)piperi...)
Affinity DataKi:  16nMAssay Description:Antagonist activity at human adrenergic beta-1 receptor expressed in CHOK1 cells assessed as inhibition of cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318975(2-((1-(2-hydroxy-3-(2-isopropylphenoxy)propyl)pipe...)
Affinity DataKi:  17nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318981(1-(2-isopropylphenoxy)-3-(1-methylpiperidin-4-ylam...)
Affinity DataKi:  17nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50223306(CHEMBL248658 | N-(2-(2-methoxyphenoxy)ethyl)-5-(4-...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50223288(CHEMBL399962 | N-(furan-2-ylmethyl)-2-nitro-5-(pip...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50223309(5-(4-methylpiperazin-1-yl)-2-nitro-N-(2-(o-tolylox...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318998(2-((1-(3-(1H-indol-4-yloxy)-2-hydroxypropyl)piperi...)
Affinity DataKi:  27nMAssay Description:Antagonist activity at human adrenergic beta-1 receptor expressed in CHOK1 cells assessed as inhibition of cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50223303(1-methyl-4-(4-nitro-3-phenoxyphenyl)piperazine | C...)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50223294(CHEMBL401294 | N-benzyl-2-nitro-5-(piperazin-1-yl)...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318990((1-(3-(9H-carbazol-4-yloxy)-2-hydroxypropyl)piperi...)
Affinity DataKi:  32nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta-1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50223304(2-nitro-N-phenethyl-5-(piperazin-1-yl)benzenamine ...)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318982(2-((1-(3-(9H-carbazol-4-yloxy)-2-hydroxypropyl)pip...)
Affinity DataKi:  37nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318973(2-((1-(2-hydroxy-3-(2-isopropylphenoxy)propyl)pipe...)
Affinity DataKi:  38nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50319003(2-(1-(3-(2-allylphenoxy)-2-hydroxypropyl)piperidin...)
Affinity DataKi:  40nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50223277(2-(benzylamino)-4-(4-methylpiperazin-1-yl)benzonit...)
Affinity DataKi:  47nMAssay Description:Binding affinity at 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318974(2-((1-(3-(2-allylphenoxy)-2-hydroxypropyl)piperidi...)
Affinity DataKi:  50nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318984(2-(1-(3-(9H-carbazol-4-yloxy)-2-hydroxypropyl)pipe...)
Affinity DataKi:  57nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50223293(CHEMBL399478 | N-(4-chlorobenzyl)-5-(4-methylpiper...)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50223305(CHEMBL251005 | N-(furan-2-ylmethyl)-5-(4-methylpip...)
Affinity DataKi:  61nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50319002(2-(2-(4-(2-hydroxy-3-(2-isopropylphenoxy)propyl)pi...)
Affinity DataKi:  70nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318987(1-(9H-carbazol-4-yloxy)-3-(4-(pyridin-3-ylmethyl)p...)
Affinity DataKi:  72nMAssay Description:Antagonist activity at human adrenergic beta3 receptor expressed in CHOK1 cells assessed as inhibition of cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318984(2-(1-(3-(9H-carbazol-4-yloxy)-2-hydroxypropyl)pipe...)
Affinity DataKi:  76nMAssay Description:Antagonist activity at human adrenergic beta-1 receptor expressed in CHOK1 cells assessed as inhibition of cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318972(2-((1-(3-(2-allylphenoxy)-2-hydroxypropyl)piperidi...)
Affinity DataKi:  78nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318992(2-((1-(3-(2-allylphenoxy)-2-hydroxypropyl)piperidi...)
Affinity DataKi:  80nMAssay Description:Antagonist activity at human adrenergic beta-1 receptor expressed in CHOK1 cells assessed as inhibition of cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318976(1-((1-(3-(2-allylphenoxy)-2-hydroxypropyl)piperidi...)
Affinity DataKi:  80nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50223290(CHEMBL398337 | N-(2-(4-tert-butylphenoxy)ethyl)-5-...)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]LSD from 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50318991(2-((1-(2-hydroxy-3-(2-isopropyl-5-methylphenoxy)pr...)
Affinity DataKi:  80nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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