Compile Data Set for Download or QSAR
maximum 50k data
Found 111 with Last Name = 'ashizawa' and Initial = 'n'
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50311264(4-(3-(4-methoxy-3-nitrophenyl)-1H-1,2,4-triazol-5-...)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of bovine milk XOR-mediated uric acid formation after 15 mins by spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50254496(4-(3-(4-isobutoxy-3-nitrophenyl)-1H-1,2,4-triazol-...)
Affinity DataIC50:  3.70nMAssay Description:Inhibition of bovine milk XOR-mediated uric acid formation after 15 mins by spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50311262(4-(3-(4-chloro-3-nitrophenyl)-1H-1,2,4-triazol-5-y...)
Affinity DataIC50:  4.70nMAssay Description:Inhibition of bovine milk XOR-mediated uric acid formation after 15 mins by spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50311266(2-isobutoxy-5-(5-(pyridin-4-yl)-1H-1,2,4-triazol-3...)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of bovine milk XOR-mediated uric acid formation after 15 mins by spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50311275(4-(5-(pyridin-4-yl)-1H-1,2,4-triazol-3-yl)picolino...)
Affinity DataIC50:  5.30nMAssay Description:Inhibition of bovine milk XOR-mediated uric acid formation after 15 mins by spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50289610(CHEMBL44717 | [3-(4,5,7-Trifluoro-benzothiazol-2-y...)
Affinity DataIC50:  6.60nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50311279(2-phenyl-4-(5-(pyridin-4-yl)-1H-1,2,4-triazol-3-yl...)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of bovine milk XOR-mediated uric acid formation after 15 mins by spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50289614(CHEMBL288748 | [3-Chloro-5-(4,5,7-trifluoro-benzot...)
Affinity DataIC50:  7nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50311276(2-chloro-4-(5-(pyridin-4-yl)-1H-1,2,4-triazol-3-yl...)
Affinity DataIC50:  7.90nMAssay Description:Inhibition of bovine milk XOR-mediated uric acid formation after 15 mins by spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50289613(CHEMBL44743 | {Phenyl-[3-(4,5,7-trifluoro-benzothi...)
Affinity DataIC50:  8.30nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAldo-keto reductase family 1 member B1(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50289624(CHEMBL44780 | {Phenyl-[3-(4,5,7-trifluoro-benzothi...)
Affinity DataIC50:  8.40nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAldo-keto reductase family 1 member B1(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50289628(3-Carboxymethyl-5-(4,5,7-trifluoro-benzothiazol-2-...)
Affinity DataIC50:  8.70nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAldo-keto reductase family 1 member B1(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50289617(CHEMBL47614 | [3-Fluoro-5-(4,5,7-trifluoro-benzoth...)
Affinity DataIC50:  8.80nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAldo-keto reductase family 1 member B1(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50289616(CHEMBL45751 | [2-Chloro-3-(4,5,7-trifluoro-benzoth...)
Affinity DataIC50:  9.30nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAldo-keto reductase family 1 member B1(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50289621(CHEMBL46074 | [3-Bromo-5-(4,5,7-trifluoro-benzothi...)
Affinity DataIC50:  9.40nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAldo-keto reductase family 1 member B1(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50289629(CHEMBL47646 | [3-Oxo-4-(4,5,7-trifluoro-benzothiaz...)
Affinity DataIC50:  9.5nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAldo-keto reductase family 1 member B1(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50289612(CHEMBL46170 | [3-Methyl-5-(4,5,7-trifluoro-benzoth...)
Affinity DataIC50:  9.60nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAldo-keto reductase family 1 member B1(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50289625(CHEMBL43995 | {Benzyl-[3-(4,5,7-trifluoro-benzothi...)
Affinity DataIC50:  9.70nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50311277(2-bromo-4-(5-(pyridin-4-yl)-1H-1,2,4-triazol-3-yl)...)
Affinity DataIC50:  9.90nMAssay Description:Inhibition of bovine milk XOR-mediated uric acid formation after 15 mins by spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50254554(4-(3-(4-isobutoxy-3-nitrophenyl)-1H-1,2,4-triazol-...)
Affinity DataIC50:  10nMAssay Description:Inhibition of bovine milk XOR-mediated uric acid formation after 15 mins by spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50289620(CHEMBL442690 | {Methyl-[3-(4,5,7-trifluoro-benzoth...)
Affinity DataIC50:  11nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAldo-keto reductase family 1 member B1(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50289615(CHEMBL45290 | [3-Iodo-5-(4,5,7-trifluoro-benzothia...)
Affinity DataIC50:  11nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAldo-keto reductase family 1 member B1(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50289619(CHEMBL542104 | [3-Dimethylamino-5-(4,5,7-trifluoro...)
Affinity DataIC50:  12nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAldo-keto reductase family 1 member B1(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM16496(2-{3-[(4-bromo-2-fluorophenyl)methyl]-7-chloro-2,4...)
Affinity DataIC50:  12nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member B1(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50289623(CHEMBL296769 | {Methyl-[3-(4,5,7-trifluoro-benzoth...)
Affinity DataIC50:  13nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAldo-keto reductase family 1 member B1(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM16314(2-{[6-methoxy-5-(trifluoromethyl)naphthalen-1-yl]-...)
Affinity DataIC50:  16nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50311265(4-(3-(4-methoxy-3-nitrophenyl)-1H-1,2,4-triazol-5-...)
Affinity DataIC50:  17nMAssay Description:Inhibition of bovine milk XOR-mediated uric acid formation after 15 mins by spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50254499(2-isobutoxy-5-(5-(2-methylpyridin-4-yl)-1H-1,2,4-t...)
Affinity DataIC50:  17nMAssay Description:Inhibition of bovine milk XOR-mediated uric acid formation after 15 mins by spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50311274(4,4'-(1H-1,2,4-triazole-3,5-diyl)dipicolinonitrile...)
Affinity DataIC50:  18nMAssay Description:Inhibition of bovine milk XOR-mediated uric acid formation after 15 mins by spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50289626(CHEMBL297861 | [2-(4,5,7-Trifluoro-benzothiazol-2-...)
Affinity DataIC50:  19nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAldo-keto reductase family 1 member B1(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50289611(CHEMBL45352 | {Phenethyl-[3-(4,5,7-trifluoro-benzo...)
Affinity DataIC50:  21nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAldo-keto reductase family 1 member B1(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50289622(CHEMBL44941 | {Benzyl-[3-(4,5,7-trifluoro-benzothi...)
Affinity DataIC50:  23nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50311285(2-isobutoxy-5-(5-(pyridin-4-yl)-1H-1,2,4-triazol-3...)
Affinity DataIC50:  24nMAssay Description:Inhibition of bovine milk XOR-mediated uric acid formation after 15 mins by spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50311282(2-methyl-4-(3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl...)
Affinity DataIC50:  28nMAssay Description:Inhibition of bovine milk XOR-mediated uric acid formation after 15 mins by spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50311263(4-(3-(4-chloro-3-nitrophenyl)-1H-1,2,4-triazol-5-y...)
Affinity DataIC50:  30nMAssay Description:Inhibition of bovine milk XOR-mediated uric acid formation after 15 mins by spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50254503(2-(2-(2-methoxyethoxy)ethoxy)-5-(3-(2-methylpyridi...)
Affinity DataIC50:  31nMAssay Description:Inhibition of bovine milk XOR-mediated uric acid formation after 15 mins by spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50158460((3,5-dibromo-4-hydroxyphenyl)(2-ethyl-1-benzofuran...)
Affinity DataIC50:  35nMAssay Description:Inhibition of URAT1 (unknown origin) transfected in dog MDCK cells assessed as inhibition of [14C]uric acid uptake by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50561689(Dotinurad | Fyu-981)
Affinity DataIC50:  37nMAssay Description:Inhibition of human URAT1 expressed in Xenopus laevis oocytes assessed as inhibition of [14C]uric acid uptake measured after 60 mins by liquid scinti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50289618(CHEMBL296780 | [4-(4,5,7-Trifluoro-benzothiazol-2-...)
Affinity DataIC50:  38nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50311284(5-(5-(pyridin-4-yl)-1H-1,2,4-triazol-3-yl)picolino...)
Affinity DataIC50:  38nMAssay Description:Inhibition of bovine milk XOR-mediated uric acid formation after 15 mins by spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50311273(4-(5-(2-chloropyridin-4-yl)-1H-1,2,4-triazol-3-yl)...)
Affinity DataIC50:  39nMAssay Description:Inhibition of bovine milk XOR-mediated uric acid formation after 15 mins by spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50158460((3,5-dibromo-4-hydroxyphenyl)(2-ethyl-1-benzofuran...)
Affinity DataIC50:  41nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50158460((3,5-dibromo-4-hydroxyphenyl)(2-ethyl-1-benzofuran...)
Affinity DataIC50:  41nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50311272(4-(3-(6-(isobutylthio)pyridin-3-yl)-1H-1,2,4-triaz...)
Affinity DataIC50:  46nMAssay Description:Inhibition of bovine milk XOR-mediated uric acid formation after 15 mins by spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50311278(2-fluoro-4-(5-(pyridin-4-yl)-1H-1,2,4-triazol-3-yl...)
Affinity DataIC50:  48nMAssay Description:Inhibition of bovine milk XOR-mediated uric acid formation after 15 mins by spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50289627(6-(4,5,7-Trifluoro-benzothiazol-2-yl)-hexanoic aci...)
Affinity DataIC50:  50nMAssay Description:Inhibitory concentration against porcine lens aldose reductase (AR) with DL-glyceraldehyde as the substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50311268(4-(3-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl)...)
Affinity DataIC50:  59nMAssay Description:Inhibition of bovine milk XOR-mediated uric acid formation after 15 mins by spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50311270(2-methyl-4-(5-(2-phenylpyridin-4-yl)-1H-1,2,4-tria...)
Affinity DataIC50:  59nMAssay Description:Inhibition of bovine milk XOR-mediated uric acid formation after 15 mins by spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50311271(2-isobutoxy-4-(3-(2-methylpyridin-4-yl)-1H-1,2,4-t...)
Affinity DataIC50:  63nMAssay Description:Inhibition of bovine milk XOR-mediated uric acid formation after 15 mins by spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Fuji Yakuhin

Curated by ChEMBL
LigandPNGBDBM50311267(2-chloro-4-(3-(2-methylpyridin-4-yl)-1H-1,2,4-tria...)
Affinity DataIC50:  89nMAssay Description:Inhibition of bovine milk XOR-mediated uric acid formation after 15 mins by spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 111 total ) | Next | Last >>
Jump to: