Affinity DataKi: 0.398nMAssay Description:Antagonist activity at human recombinant EP1 receptor expressed in CHO-K1 cells assessed as inhibition of PGE2-mediated intracellular calcium mobiliz...More data for this Ligand-Target Pair
Affinity DataKi: 0.780nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of VMAT2 in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of VMAT2 in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 9.70nMAssay Description:Inhibition of VMAT2 in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Inhibition of VMAT2 in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 270nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 560nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 760nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 960nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Antagonist activity at human recombinant EP3 receptor expressed in CHO-K1 cells assessed as inhibition of PGE2-mediated intracellular calcium mobiliz...More data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+3nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.70E+3nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.90E+3nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.20E+3nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.20E+3nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair