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Found 67 with Last Name = 'audouze' and Initial = 'k'
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147929(4-(4-Bromo-benzyl)-2-(4-chloro-2-methoxy-phenoxyme...)
Affinity DataKi:  2nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147961((S)-4-(4-Chloro-benzyl)-2-(4-chloro-2-methoxy-phen...)
Affinity DataKi:  2.80nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147939(4-(4-Chloro-benzyl)-2-(5-chloro-2-ethoxy-phenoxyme...)
Affinity DataKi:  2.90nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147932(4-(4-Chloro-benzyl)-2-(4-chloro-2-methoxy-phenoxym...)
Affinity DataKi:  4.40nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147959(CHEMBL325789 | [4-(4-Chloro-benzyl)-morpholin-2-yl...)
Affinity DataKi:  4.5nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147960(4-(4-Chloro-benzyl)-2-(2-ethoxy-phenoxymethyl)-[1,...)
Affinity DataKi:  4.90nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147956(5-Chloro-2-{[4-(4-chloro-benzyl)-morpholin-2-ylmet...)
Affinity DataKi:  5.40nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147954(1-{4-Chloro-2-[4-(4-chloro-benzyl)-[1,4]oxazepan-2...)
Affinity DataKi:  5.5nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147950(4-(4-Chloro-benzyl)-2-(4-chloro-2-ethoxy-phenoxyme...)
Affinity DataKi:  7nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147955(4-(4-Chloro-benzyl)-2-(5-chloro-2-ethoxy-phenoxyme...)
Affinity DataKi:  9.30nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147941(4-(4-Chloro-benzyl)-2-(2-ethoxy-phenoxymethyl)-mor...)
Affinity DataKi:  13nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147953(4-(4-Chloro-benzyl)-2-(4-chloro-2-ethoxy-phenoxyme...)
Affinity DataKi:  13nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147938(4-(4-Chloro-benzyl)-2-(2-methoxy-5-nitro-phenoxyme...)
Affinity DataKi:  23nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147963(4-(4-Chloro-benzyl)-2-(2-ethoxy-4-iodo-phenoxymeth...)
Affinity DataKi:  24nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147931(4-(4-Chloro-benzyl)-2-[2-(2-methoxy-phenyl)-ethyl]...)
Affinity DataKi:  29nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147951(4-(4-Chloro-benzyl)-2-(5-fluoro-2-methoxy-phenoxym...)
Affinity DataKi:  30nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147930(2-(2-Butyl-phenoxymethyl)-4-(4-chloro-benzyl)-morp...)
Affinity DataKi:  32nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147957(4-(3,4-Dichloro-benzyl)-2-(2-methoxy-phenoxymethyl...)
Affinity DataKi:  32nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147944(4-(4-Chloro-benzyl)-2-(2-methoxy-phenoxymethyl)-mo...)
Affinity DataKi:  32nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147952(2-(2-Ethoxy-phenoxymethyl)-4-(4-nitro-benzyl)-morp...)
Affinity DataKi:  35nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147934(4-[4-(4-Chloro-benzyl)-morpholin-2-ylmethoxy]-3-et...)
Affinity DataKi:  40nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147958(5-Chloro-8-[4-(4-chloro-benzyl)-morpholin-2-ylmeth...)
Affinity DataKi:  40nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147936(4-(4-Chloro-benzyl)-2-(2-isopropoxy-phenoxymethyl)...)
Affinity DataKi:  46nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147949(4-(4-Chloro-benzyl)-2-[2-(2-methoxy-ethoxy)-phenox...)
Affinity DataKi:  52nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147948(4-(4-Chloro-benzyl)-2-(2-methoxy-phenylsulfanylmet...)
Affinity DataKi:  61nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147969(2-(2-Methoxy-phenoxymethyl)-4-(4-trifluoromethyl-b...)
Affinity DataKi:  61nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147943(4-Benzyl-2-(5-chloro-2-methoxy-phenoxymethyl)-morp...)
Affinity DataKi:  70nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147940(4-(4-Chloro-benzyl)-2-(2-methyl-pyridin-3-yloxymet...)
Affinity DataKi:  83nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147964(3-[4-(4-Chloro-benzyl)-morpholin-2-ylmethoxy]-4-me...)
Affinity DataKi:  100nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147933(2-(2-Ethoxy-phenoxymethyl)-4-(4-fluoro-benzyl)-mor...)
Affinity DataKi:  180nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147967(4-(4-Chloro-benzyl)-2-[(E)-2-(2-methoxy-phenyl)-vi...)
Affinity DataKi:  200nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147962(4-(4-Chloro-benzyl)-2-(2-methoxy-5-trifluoromethyl...)
Affinity DataKi:  250nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147946(4-(2,4-Dichloro-benzyl)-2-(2-ethoxy-phenoxymethyl)...)
Affinity DataKi:  290nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147942(4-(4-Chloro-benzyl)-2-(2-methoxy-5-nitro-phenoxyme...)
Affinity DataKi:  400nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147968(4-Benzyl-2-(4-iodo-2-methoxy-phenoxymethyl)-morpho...)
Affinity DataKi:  430nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147937(4-Benzyl-2-(4-chloro-2-methoxy-phenoxymethyl)-morp...)
Affinity DataKi:  650nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147945(4-Benzyl-2-(2-methoxy-phenoxymethyl)-morpholine | ...)
Affinity DataKi:  850nMAssay Description:In vitro ability to inhibit binding of [3H]-spiperone to human recombinant Dopamine receptor D4.2 expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147965(4-Benzyl-2-(3-chloro-5-methoxy-phenoxymethyl)-morp...)
Affinity DataKi:  920nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147935(4-(4-Chloro-benzyl)-2-(2,3-dimethoxy-phenoxymethyl...)
Affinity DataKi:  1.00E+3nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50147947((R)-4-(4-Chloro-benzyl)-2-(4-chloro-2-methoxy-phen...)
Affinity DataKi:  1.60E+3nMAssay Description:In vitro ability of compound to inhibit binding of [3H]-spiperone to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50187442(1-(6-bromo-5-(vinyloxy)pyridin-3-yl)-1,5-diazocane...)
Affinity DataIC50:  0.380nMAssay Description:Inhibition of [3H]cytisine binding to alpha4beta2 nACHR in Wistar rat cerebral cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50187445(1-(6-bromopyridin-3-yl)-1,5-diazocane | 1-(6-bromo...)
Affinity DataIC50:  0.450nMAssay Description:Inhibition of [3H]cytisine binding to alpha4beta2 nACHR in Wistar rat cerebral cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50187455(1-(6-Bromo-5-vinylpyridin-3-yl)-[1,4]diazepane | 1...)
Affinity DataIC50:  0.640nMAssay Description:Inhibition of [3H]cytisine binding to alpha4beta2 nACHR in Wistar rat cerebral cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50187447(1-(pyridin-3-yl)-1,5-diazocane | 1-pyridin-3-yl-[1...)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of [3H]cytisine binding to alpha4beta2 nACHR in Wistar rat cerebral cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50187439(1-(5-Methoxypyridin-3-yl)-[1,5]diazocane | 1-(5-me...)
Affinity DataIC50:  1nMAssay Description:Inhibition of [3H]cytisine binding to alpha4beta2 nACHR in Wistar rat cerebral cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50187438((Z)-1-(5-(prop-1-enyloxy)pyridin-3-yl)-1,4-diazepa...)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of [3H]cytisine binding to alpha4beta2 nACHR in Wistar rat cerebral cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50187453(1-(6-bromo-5-chloropyridin-3-yl)-1,4-diazepane | 1...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of [3H]cytisine binding to alpha4beta2 nACHR in Wistar rat cerebral cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50187441(1-(5-bromo-6-chloropyridin-3-yl)-1,4-diazepane | 4...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of [3H]cytisine binding to alpha4beta2 nACHR in Wistar rat cerebral cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50475830(CHEMBL210643)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of [3H]cytisine binding to alpha4beta2 nACHR in Wistar rat cerebral cortical membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Neurosearch

Curated by ChEMBL
LigandPNGBDBM50475827(CHEMBL206988)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of [3H]cytisine binding to alpha4beta2 nACHR in Wistar rat cerebral cortical membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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