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Found 7 with Last Name = 'avonto' and Initial = 'c'
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
National Research Council (Icb-Cnr)

Curated by ChEMBL
LigandPNGBDBM20461((6E)-N-[(4-hydroxy-3-methoxyphenyl)methyl]-8-methy...)
Affinity DataIC50:  8nMAssay Description:Antagonist activity at human TRPV1 stably transfected in HEK293 cells assessed as decrease in calcium influx preincubated for 5 mins followed by caps...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
National Research Council (Icb-Cnr)

Curated by ChEMBL
LigandPNGBDBM50554642(CHEMBL4800169)
Affinity DataIC50:  50nMAssay Description:Antagonist activity at human TRPV1 stably transfected in HEK293 cells assessed as decrease in calcium influx preincubated for 5 mins followed by caps...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50433441(PARTHENOLIDE)
Affinity DataIC50:  1.05E+3nMAssay Description:Inhibition of iNOS in mouse RAW264.7 cells assessed as LPS-induced nitric oxide production treated for 30 mins followed by LPS challenge measured aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
National Research Council (Icb-Cnr)

Curated by ChEMBL
LigandPNGBDBM50554641(CHEMBL554265)
Affinity DataIC50:  7.50E+3nMAssay Description:Antagonist activity at human TRPV1 stably transfected in HEK293 cells assessed as decrease in calcium influx preincubated for 5 mins followed by caps...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
National Research Council (Icb-Cnr)

Curated by ChEMBL
LigandPNGBDBM50554641(CHEMBL554265)
Affinity DataEC50:  5.40E+3nMAssay Description:Agonist activity at human TRPV1 stably transfected in HEK293 cells assessed as increase in calcium influx in presence of ionomycin by Fluo-4-AM dye b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
National Research Council (Icb-Cnr)

Curated by ChEMBL
LigandPNGBDBM20461((6E)-N-[(4-hydroxy-3-methoxyphenyl)methyl]-8-methy...)
Affinity DataEC50:  5.30nMAssay Description:Agonist activity at human TRPV1 stably transfected in HEK293 cells assessed as increase in calcium influx in presence of ionomycin by Fluo-4-AM dye b...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
National Research Council (Icb-Cnr)

Curated by ChEMBL
LigandPNGBDBM50554642(CHEMBL4800169)
Affinity DataEC50:  35nMAssay Description:Agonist activity at human TRPV1 stably transfected in HEK293 cells assessed as increase in calcium influx in presence of ionomycin by Fluo-4-AM dye b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed