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Found 286 with Last Name = 'awad' and Initial = 'ma'
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567601(CHEMBL4857595)
Affinity DataKi:  4.30nMAssay Description:Inhibition of recombinant human CA9 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50334354(4-(3-(4-fluorophenyl)ureido)benzenesulfonamide | 4...)
Affinity DataKi:  4.5nMAssay Description:Inhibition of recombinant human CA12 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567598(CHEMBL4853209)
Affinity DataKi:  5.10nMAssay Description:Inhibition of recombinant human CA12 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  5.70nMAssay Description:Inhibition of recombinant human CA12 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567599(CHEMBL4847847)
Affinity DataKi:  5.90nMAssay Description:Inhibition of recombinant human CA2 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567598(CHEMBL4853209)
Affinity DataKi:  6.5nMAssay Description:Inhibition of recombinant human CA9 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567598(CHEMBL4853209)
Affinity DataKi:  7.40nMAssay Description:Inhibition of recombinant human CA2 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567599(CHEMBL4847847)
Affinity DataKi:  7.90nMAssay Description:Inhibition of recombinant human CA12 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567596(CHEMBL4877641)
Affinity DataKi:  11nMAssay Description:Inhibition of recombinant human CA12 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  12nMAssay Description:Inhibition of recombinant human CA2 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567597(CHEMBL4860073)
Affinity DataKi:  15nMAssay Description:Inhibition of recombinant human CA2 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567597(CHEMBL4860073)
Affinity DataKi:  16nMAssay Description:Inhibition of recombinant human CA9 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567601(CHEMBL4857595)
Affinity DataKi:  20nMAssay Description:Inhibition of recombinant human CA2 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567596(CHEMBL4877641)
Affinity DataKi:  23nMAssay Description:Inhibition of recombinant human CA9 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  25nMAssay Description:Inhibition of recombinant human CA9 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567599(CHEMBL4847847)
Affinity DataKi:  30nMAssay Description:Inhibition of recombinant human CA9 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567600(CHEMBL4860400)
Affinity DataKi:  32nMAssay Description:Inhibition of recombinant human CA2 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567600(CHEMBL4860400)
Affinity DataKi:  33nMAssay Description:Inhibition of recombinant human CA12 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567601(CHEMBL4857595)
Affinity DataKi:  36nMAssay Description:Inhibition of recombinant human CA12 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567597(CHEMBL4860073)
Affinity DataKi:  42nMAssay Description:Inhibition of recombinant human CA12 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567596(CHEMBL4877641)
Affinity DataKi:  44nMAssay Description:Inhibition of recombinant human CA2 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50334354(4-(3-(4-fluorophenyl)ureido)benzenesulfonamide | 4...)
Affinity DataKi:  45nMAssay Description:Inhibition of recombinant human CA9 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567600(CHEMBL4860400)
Affinity DataKi:  46nMAssay Description:Inhibition of recombinant human CA9 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286369(2-(N',N''-Dicyclohexyl-guanidino)-3-naphthalen-2-y...)
Affinity DataKi:  60nMAssay Description:Binding affinity against human IMR 90 fetal lung fibroblast bradykinin receptor B2More data for this Ligand-Target Pair
In DepthDetails Article
TargetB2 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286372(2-(N',N''-Dicyclohexyl-guanidino)-3-naphthalen-2-y...)
Affinity DataKi:  60nMAssay Description:Binding affinity against human IMR 90 fetal lung fibroblast bradykinin receptor B2More data for this Ligand-Target Pair
In DepthDetails Article
TargetB2 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286365(2-(N',N''-Dicyclohexyl-N-methyl-guanidino)-3-napht...)
Affinity DataKi:  70nMAssay Description:Binding affinity against human IMR 90 fetal lung fibroblast bradykinin receptor B2More data for this Ligand-Target Pair
In DepthDetails Article
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567597(CHEMBL4860073)
Affinity DataKi:  72nMAssay Description:Inhibition of recombinant human CA1 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567599(CHEMBL4847847)
Affinity DataKi:  84nMAssay Description:Inhibition of recombinant human CA1 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567598(CHEMBL4853209)
Affinity DataKi:  93nMAssay Description:Inhibition of recombinant human CA1 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286357(2-(N',N''-Dicyclohexyl-guanidino)-3-naphthalen-2-y...)
Affinity DataKi:  110nMAssay Description:Binding affinity against human IMR 90 fetal lung fibroblast bradykinin receptor B2More data for this Ligand-Target Pair
In DepthDetails Article
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567600(CHEMBL4860400)
Affinity DataKi:  114nMAssay Description:Inhibition of recombinant human CA1 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567601(CHEMBL4857595)
Affinity DataKi:  130nMAssay Description:Inhibition of recombinant human CA1 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286383((S)-2-(N',N''-Di-p-tolyl-guanidino)-3-naphthalen-2...)
Affinity DataKi:  140nMAssay Description:Binding affinity against human IMR 90 fetal lung fibroblast bradykinin receptor B2More data for this Ligand-Target Pair
In DepthDetails Article
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  250nMAssay Description:Inhibition of recombinant human CA1 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286388(N,N'-Dicyclohexyl-N''-{(E)-(S)-1-naphthalen-2-ylme...)
Affinity DataKi:  250nMAssay Description:Binding affinity against human IMR 90 fetal lung fibroblast bradykinin receptor B2More data for this Ligand-Target Pair
In DepthDetails Article
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567596(CHEMBL4877641)
Affinity DataKi:  320nMAssay Description:Inhibition of recombinant human CA1 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50286369(2-(N',N''-Dicyclohexyl-guanidino)-3-naphthalen-2-y...)
Affinity DataKi:  350nMAssay Description:Binding affinity towards rat muscarinic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetB2 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286393((NE)-N-({[(1S)-1-({1-azabicyclo[2.2.2]octan-3-yl}c...)
Affinity DataKi:  410nMAssay Description:Binding affinity against human IMR 90 fetal lung fibroblast bradykinin receptor B2More data for this Ligand-Target Pair
In DepthDetails Article
TargetB2 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286390(3-Benzo[b]thiophen-2-yl-2-(N',N''-dicyclohexyl-gua...)
Affinity DataKi:  430nMAssay Description:Binding affinity against human IMR 90 fetal lung fibroblast bradykinin receptor B2More data for this Ligand-Target Pair
In DepthDetails Article
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567605(CHEMBL4877370)
Affinity DataKi:  530nMAssay Description:Inhibition of recombinant human CA12 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286364((NE)-N-({[1-({1-azabicyclo[2.2.2]octan-3-yl}carbam...)
Affinity DataKi:  550nMAssay Description:Binding affinity against human IMR 90 fetal lung fibroblast bradykinin receptor B2More data for this Ligand-Target Pair
In DepthDetails Article
TargetB2 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286364((NE)-N-({[1-({1-azabicyclo[2.2.2]octan-3-yl}carbam...)
Affinity DataKi:  550nMAssay Description:Binding affinity against human IMR 90 fetal lung fibroblast bradykinin receptor B2More data for this Ligand-Target Pair
In DepthDetails Article
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567605(CHEMBL4877370)
Affinity DataKi:  720nMAssay Description:Inhibition of recombinant human CA9 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286367(N,N'-Dicyclohexyl-N''-{(Z)-(S)-1-naphthalen-2-ylme...)
Affinity DataKi:  760nMAssay Description:Binding affinity against human IMR 90 fetal lung fibroblast bradykinin receptor B2More data for this Ligand-Target Pair
In DepthDetails Article
TargetB2 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286392(Bis-[4-(tripentyl-lambda*5*-phosphanylmethyl)-phen...)
Affinity DataKi:  770nMAssay Description:Binding affinity against human IMR 90 fetal lung fibroblast bradykinin receptor B2More data for this Ligand-Target Pair
In DepthDetails Article
TargetB2 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286370(N-(1-Aza-bicyclo[2.2.2]oct-3-yl)-N-benzyl-2-(N',N'...)
Affinity DataKi:  820nMAssay Description:Binding affinity against human IMR 90 fetal lung fibroblast bradykinin receptor B2More data for this Ligand-Target Pair
In DepthDetails Article
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567602(CHEMBL4856530)
Affinity DataKi:  850nMAssay Description:Inhibition of recombinant human CA12 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50567602(CHEMBL4856530)
Affinity DataKi:  930nMAssay Description:Inhibition of recombinant human CA9 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kafrelsheikh University

Curated by ChEMBL
LigandPNGBDBM50334354(4-(3-(4-fluorophenyl)ureido)benzenesulfonamide | 4...)
Affinity DataKi:  960nMAssay Description:Inhibition of recombinant human CA2 pre-incubated for 15 mins measured by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286381(2-(N',N''-Dicyclohexyl-guanidino)-3-naphthalen-1-y...)
Affinity DataKi:  1.03E+3nMAssay Description:Binding affinity against human IMR 90 fetal lung fibroblast bradykinin receptor B2More data for this Ligand-Target Pair
In DepthDetails Article
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