Compile Data Set for Download or QSAR
maximum 50k data
Found 173 with Last Name = 'ayscough' and Initial = 'a'
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347034(CHEMBL1796096)
Affinity DataIC50:  5nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50131342((R)-2-[(Formyl-hydroxy-amino)-methyl]-hexanoic aci...)
Affinity DataIC50:  6nMAssay Description:Inhibition concentration against Escherichia coli peptide deformylase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347036(CHEMBL1796098)
Affinity DataIC50:  6nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase, mitochondrial(Homo sapiens (Human))
British Biotech Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50131303((S)-2-[(R)-2-Cyclohexylmethyl-3-(formyl-hydroxy-am...)
Affinity DataIC50:  6nMAssay Description:Inhibition against Escherichia coli peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50104501((R)-2-[(Formyl-hydroxy-amino)-methyl]-hexanoic aci...)
Affinity DataIC50:  7nMAssay Description:Inhibition concentration against Escherichia coli peptide deformylase.More data for this Ligand-Target Pair
TargetPeptide deformylase, mitochondrial(Homo sapiens (Human))
British Biotech Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50104501((R)-2-[(Formyl-hydroxy-amino)-methyl]-hexanoic aci...)
Affinity DataIC50:  7nMAssay Description:Inhibition against Escherichia coli peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347040(CHEMBL1796103)
Affinity DataIC50:  7nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50104501((R)-2-[(Formyl-hydroxy-amino)-methyl]-hexanoic aci...)
Affinity DataIC50:  7nMAssay Description:Inhibition concentration against Escherichia coli peptide deformylase.More data for this Ligand-Target Pair
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347047(CHEMBL1796230)
Affinity DataIC50:  8nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase, mitochondrial(Homo sapiens (Human))
British Biotech Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50131290((S)-2-[(R)-2-Cyclopentylmethyl-3-(formyl-hydroxy-a...)
Affinity DataIC50:  8nMAssay Description:Inhibition against Escherichia coli peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl hydroxylase EGLN2(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50239931(CHEMBL4067995 | US10287286, Example 142)
Affinity DataIC50:  8nMAssay Description:Inhibition of full length HIF-PHD1 (unknown origin) expressed in baculovirus infected sf9 cells using DLDLEMLAPYIPMDDDFQL/2-Oxoglutarate as substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50221045(CHEMBL3706628)
Affinity DataIC50:  9nMAssay Description:Inhibition concentration against Escherichia coli peptide deformylase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347021(CHEMBL1796080)
Affinity DataIC50:  9nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347046(CHEMBL1796228)
Affinity DataIC50:  9nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase, mitochondrial(Homo sapiens (Human))
British Biotech Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50131304((R)-2-[(Formyl-hydroxy-amino)-methyl]-heptanoic ac...)
Affinity DataIC50:  10nMAssay Description:Inhibition against Escherichia coli peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347035(CHEMBL1796097)
Affinity DataIC50:  10nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase, mitochondrial(Homo sapiens (Human))
British Biotech Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50131292((R)-2-[(Formyl-hydroxy-amino)-methyl]-4-methyl-pen...)
Affinity DataIC50:  10nMAssay Description:Inhibition against Escherichia coli peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50131314((R)-2-[(Formyl-hydroxy-amino)-methyl]-hexanoic aci...)
Affinity DataIC50:  10nMAssay Description:Inhibition concentration against Escherichia coli peptide deformylase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50131343((R)-2-[(Formyl-hydroxy-amino)-methyl]-hexanoic aci...)
Affinity DataIC50:  10nMAssay Description:Inhibition concentration against Escherichia coli peptide deformylase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347041(CHEMBL1796105)
Affinity DataIC50:  10nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347038(CHEMBL1796101)
Affinity DataIC50:  10nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50131311(1-((S)-2-{(R)-2-[(Formyl-hydroxy-amino)-methyl]-he...)
Affinity DataIC50:  10nMAssay Description:Inhibition concentration against Escherichia coli peptide deformylase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50131324((R)-2-[(Formyl-hydroxy-amino)-methyl]-hexanoic aci...)
Affinity DataIC50:  10nMAssay Description:Inhibition concentration against Escherichia coli peptide deformylase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl hydroxylase EGLN2(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50239883(CHEMBL4090769 | US10287286, Example 5)
Affinity DataIC50:  10nMAssay Description:Inhibition of full length HIF-PHD1 (unknown origin) expressed in baculovirus infected sf9 cells using DLDLEMLAPYIPMDDDFQL/2-Oxoglutarate as substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347050(CHEMBL1796104)
Affinity DataIC50:  10nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50131315((R)-2-[(Formyl-hydroxy-amino)-methyl]-hexanoic aci...)
Affinity DataIC50:  10nMAssay Description:Inhibition concentration against Escherichia coli peptide deformylase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347044(CHEMBL1796226)
Affinity DataIC50:  10nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347043(CHEMBL1796225)
Affinity DataIC50:  10nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl hydroxylase EGLN2(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50239889(CHEMBL4072842 | US10287286, Example 100)
Affinity DataIC50:  13nMAssay Description:Inhibition of full length HIF-PHD1 (unknown origin) expressed in baculovirus infected sf9 cells using DLDLEMLAPYIPMDDDFQL/2-Oxoglutarate as substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347042(CHEMBL1796106)
Affinity DataIC50:  20nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347048(CHEMBL1796229)
Affinity DataIC50:  20nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50131340((R)-2-[(Formyl-hydroxy-amino)-methyl]-hexanoic aci...)
Affinity DataIC50:  20nMAssay Description:Inhibition concentration against Escherichia coli peptide deformylase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50131345((R)-2-[(Formyl-hydroxy-amino)-methyl]-hexanoic aci...)
Affinity DataIC50:  20nMAssay Description:Inhibition concentration against Escherichia coli peptide deformylase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50131319((R)-2-[(Formyl-hydroxy-amino)-methyl]-hexanoic aci...)
Affinity DataIC50:  20nMAssay Description:Inhibition concentration against Escherichia coli peptide deformylase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50131341((R)-2-[(Formyl-hydroxy-amino)-methyl]-hexanoic aci...)
Affinity DataIC50:  20nMAssay Description:Inhibition concentration against Escherichia coli peptide deformylase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50131326((R)-2-[(Formyl-hydroxy-amino)-methyl]-hexanoic aci...)
Affinity DataIC50:  20nMAssay Description:Inhibition concentration against Escherichia coli peptide deformylase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50131312(4-((S)-Dimethyl-carbamoyl)-4-{(R)-2-[(formyl-hydro...)
Affinity DataIC50:  20nMAssay Description:Inhibition concentration against Escherichia coli peptide deformylase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50131325((R)-2-[(Formyl-hydroxy-amino)-methyl]-hexanoic aci...)
Affinity DataIC50:  20nMAssay Description:Inhibition concentration against Escherichia coli peptide deformylase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50131344((R)-2-[(Formyl-hydroxy-amino)-methyl]-hexanoic aci...)
Affinity DataIC50:  20nMAssay Description:Inhibition concentration against Escherichia coli peptide deformylase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50131310((R)-2-[(Formyl-hydroxy-amino)-methyl]-hexanoic aci...)
Affinity DataIC50:  20nMAssay Description:Inhibition concentration against Escherichia coli peptide deformylase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50131316((R)-2-[(Formyl-hydroxy-amino)-methyl]-hexanoic aci...)
Affinity DataIC50:  20nMAssay Description:Inhibition concentration against Escherichia coli peptide deformylase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase, mitochondrial(Homo sapiens (Human))
British Biotech Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50131288((R)-2-[(Formyl-hydroxy-amino)-methyl]-hex-5-enoic ...)
Affinity DataIC50:  20nMAssay Description:Inhibition against Escherichia coli peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase, mitochondrial(Homo sapiens (Human))
British Biotech Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50131295((S)-2-[(R)-2-Ethylsulfanylmethyl-3-(formyl-hydroxy...)
Affinity DataIC50:  20nMAssay Description:Inhibition against Escherichia coli peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase, mitochondrial(Homo sapiens (Human))
British Biotech Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50131301((S)-2-[(R)-2-Benzyl-3-(formyl-hydroxy-amino)-propi...)
Affinity DataIC50:  20nMAssay Description:Inhibition against Escherichia coli peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase, mitochondrial(Homo sapiens (Human))
British Biotech Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50131302((R)-2-[(Formyl-hydroxy-amino)-methyl]-5-methyl-hex...)
Affinity DataIC50:  20nMAssay Description:Inhibition against Escherichia coli peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase, mitochondrial(Homo sapiens (Human))
British Biotech Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50131307((S)-2-[(R)-2-Cyclopentyl-3-(formyl-hydroxy-amino)-...)
Affinity DataIC50:  20nMAssay Description:Inhibition against Escherichia coli peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347028(CHEMBL1796089)
Affinity DataIC50:  20nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347039(CHEMBL1796102)
Affinity DataIC50:  20nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl hydroxylase EGLN2(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50239888(CHEMBL4094292 | US10287286, Example 103)
Affinity DataIC50:  25nMAssay Description:Inhibition of full length HIF-PHD1 (unknown origin) expressed in baculovirus infected sf9 cells using DLDLEMLAPYIPMDDDFQL/2-Oxoglutarate as substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347045(CHEMBL1796227)
Affinity DataIC50:  30nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 173 total ) | Next | Last >>
Jump to: