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Found 32 with Last Name = 'bühlmayer' and Initial = 'p'
TargetRenin(Homo sapiens (Human))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50022582(CHEMBL53139 | Diastereomer-5-[2-[2-Benzyl-3-(2-met...)
Affinity DataIC50:  0.400nMAssay Description:In vitro inhibition of Human kideny reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50022582(CHEMBL53139 | Diastereomer-5-[2-[2-Benzyl-3-(2-met...)
Affinity DataIC50:  1nMAssay Description:In vitro inhibition of marmoset plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50022582(CHEMBL53139 | Diastereomer-5-[2-[2-Benzyl-3-(2-met...)
Affinity DataIC50:  2nMpH: 7.2Assay Description:In vitro inhibition of marmoset plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50022582(CHEMBL53139 | Diastereomer-5-[2-[2-Benzyl-3-(2-met...)
Affinity DataIC50:  2nMpH: 7.2Assay Description:In vitro inhibition of porcine plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50022582(CHEMBL53139 | Diastereomer-5-[2-[2-Benzyl-3-(2-met...)
Affinity DataIC50:  2nMAssay Description:In vitro inhibition of Human plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50022586(5-[2-[2-Benzyl-3-(2-methyl-propane-2-sulfinyl)-pro...)
Affinity DataIC50:  2nMAssay Description:In vitro inhibition of purified Human kidney renin (250 pg/mL) incubated with angiotensinogen at pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50022582(CHEMBL53139 | Diastereomer-5-[2-[2-Benzyl-3-(2-met...)
Affinity DataIC50:  3nMAssay Description:In vitro inhibition of purified Human kidney renin (250 pg/mL) incubated with angiotensinogen at pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50022587(5-[2-(2-tert-Butylsulfanylmethyl-3-phenyl-propiony...)
Affinity DataIC50:  4nMAssay Description:In vitro inhibition of purified Human kidney renin (250 pg/mL) incubated with angiotensinogen at pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50022588(CHEMBL291787 | {2-[1-(4-Butylcarbamoyl-1-cyclohexy...)
Affinity DataIC50:  4nMAssay Description:In vitro inhibition of purified Human kidney renin (250 pg/mL) incubated with angiotensinogen at pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50022584(2-Benzyl-5,5-dimethyl-4-oxo-hexanoic acid [1-(4-bu...)
Affinity DataIC50:  6nMAssay Description:In vitro inhibition of purified Human kidney renin (250 pg/mL) incubated with angiotensinogen at pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50022590(2,2-Dimethyl-propionic acid 1-[1-(4-butylcarbamoyl...)
Affinity DataIC50:  7nMAssay Description:In vitro inhibition of purified Human kidney renin (250 pg/mL) incubated with angiotensinogen at pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50022859(CHEMBL407670 | Pro-His-Pro-Phe-His-Leu[CH2NH]Val-I...)
Affinity DataIC50:  10nMAssay Description:In vitro inhibition of purified Human kidney renin (250 pg/mL) incubated with angiotensinogen at pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50022589(CHEMBL435178 | {1-[1-(4-{1-[1-Carbamoyl-2-(3H-imid...)
Affinity DataIC50:  15nMAssay Description:In vitro inhibition of purified Human kidney renin (250 pg/mL) incubated with angiotensinogen at pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50022585(5-[2-[2-(2,2-Dimethyl-propionylamino)-3-phenyl-pro...)
Affinity DataIC50:  20nMAssay Description:In vitro inhibition of purified Human kidney renin (250 pg/mL) incubated with angiotensinogen at pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50022581(2,2-Dimethyl-propionic acid 1-[1-(4-butylcarbamoyl...)
Affinity DataIC50:  20nMAssay Description:In vitro inhibition of purified Human kidney renin (250 pg/mL) incubated with angiotensinogen at pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50022591(2,2-Dimethyl-propionic acid 1-[1-(4-{1-[1-carbamoy...)
Affinity DataIC50:  20nMAssay Description:In vitro inhibition of purified Human kidney renin (250 pg/mL) incubated with angiotensinogen at pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50009714(CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...)
Affinity DataIC50:  26nMAssay Description:Binding affinity against angiotensin II receptor in rat smooth muscle cell preparationsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50010146(CHEMBL322683 | {2-Butyl-5-chloro-1-[6-(1H-tetrazol...)
Affinity DataIC50:  200nMAssay Description:Binding affinity against Angiotensin II receptor in rat smooth muscle cell preparationsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50022582(CHEMBL53139 | Diastereomer-5-[2-[2-Benzyl-3-(2-met...)
Affinity DataIC50:  400nMAssay Description:In vitro inhibition of rat plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50010144(CHEMBL322071 | {2-Butyl-5-chloro-3-[6-(1H-tetrazol...)
Affinity DataIC50:  600nMAssay Description:Binding affinity against angiotensin II receptor in rat smooth muscle cell preparationsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50010154(6-(2-Butyl-5-chloro-4-hydroxymethyl-imidazol-1-ylm...)
Affinity DataIC50:  1.10E+3nMAssay Description:Binding affinity against angiotensin II receptor in rat smooth muscle cell preparationsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50010150(CHEMBL107862 | {2-Butyl-5-chloro-3-[5-(1H-tetrazol...)
Affinity DataIC50:  1.10E+3nMAssay Description:Binding affinity against angiotensin II receptor in rat smooth muscle cell preparationsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50010145(CHEMBL105525 | {2-Butyl-5-chloro-1-[6-(1H-tetrazol...)
Affinity DataIC50:  1.40E+3nMAssay Description:Binding affinity against angiotensin II receptor in rat smooth muscle cell preparationsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50010147(6-(2-Butyl-5-chloro-4-hydroxymethyl-imidazol-1-ylm...)
Affinity DataIC50:  2.80E+3nMAssay Description:Binding affinity against angiotensin II receptor in rat smooth muscle cell preparationsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Bos taurus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50022582(CHEMBL53139 | Diastereomer-5-[2-[2-Benzyl-3-(2-met...)
Affinity DataIC50:  3.20E+3nMAssay Description:In vitro inhibition of bovine cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50010155(CHEMBL320951 | {2-Butyl-5-chloro-3-[6-(1H-tetrazol...)
Affinity DataIC50:  4.10E+3nMAssay Description:Binding affinity against angiotensin II receptor in rat smooth muscle cell preparationsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50010151(6-(2-Butyl-4-chloro-5-hydroxymethyl-imidazol-1-ylm...)
Affinity DataIC50:  4.60E+3nMAssay Description:Binding affinity against angiotensin II receptor in rat smooth muscle cell preparationsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50010148(CHEMBL106934 | {2-Butyl-5-chloro-3-[6-(1H-tetrazol...)
Affinity DataIC50:  5.40E+3nMAssay Description:Binding affinity against angiotensin II receptor in rat smooth muscle cell preparationsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50022582(CHEMBL53139 | Diastereomer-5-[2-[2-Benzyl-3-(2-met...)
Affinity DataIC50:  8.20E+3nMAssay Description:In vitro inhibition of dog plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50010152(6-(2-Butyl-4-chloro-5-hydroxymethyl-imidazol-1-ylm...)
Affinity DataIC50:  8.90E+3nMAssay Description:Binding affinity against angiotensin II receptor in rat smooth muscle cell preparationsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50010153(CHEMBL105724 | {2-Butyl-5-chloro-3-[7-(1H-tetrazol...)
Affinity DataIC50:  2.00E+4nMAssay Description:Binding affinity against Angiotensin II receptor in rat smooth muscle cell preparationsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50010149(CHEMBL323179 | {2-Butyl-5-chloro-3-[8-(1H-tetrazol...)
Affinity DataIC50:  5.50E+4nMAssay Description:Binding affinity against angiotensin II receptor in rat smooth muscle cell preparationsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed