Affinity DataIC50: 0.200nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.25nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.75nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibitory activity against FKBP12More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMpH: 7.5 T: 2°CAssay Description:Assays were performed in 96-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified kinase in the presence of ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: 3.30nMAssay Description:Inhibitory activity against FKBP12More data for this Ligand-Target Pair
Affinity DataIC50: 4nMpH: 6.0Assay Description:Inhibition of human renal renin at pH 6More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: 4.30nMAssay Description:Inhibition of ErbB2 by time resolved fluorescence assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: 4.80nMAssay Description:Inhibitory activity against FKBP12More data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: 4.80nMAssay Description:Inhibition of ErbB2 by time resolved fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.80nMAssay Description:Inhibitory activity against FKBP12More data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: 6.30nMAssay Description:Inhibition of ErbB2 by time resolved fluorescence assayMore data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: 7.20nMAssay Description:Inhibition of ErbB2 by time resolved fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMpH: 6.0Assay Description:Inhibition of human renal renin at pH 6More data for this Ligand-Target Pair
Affinity DataIC50: 9nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
Affinity DataIC50: 9nMT: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
Affinity DataIC50: 9nMT: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:In vitro inhibitory activity was tested against purified human renal reninMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMT: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMT: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair