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Found 141 with Last Name = 'baekelandt' and Initial = 'v'
TargetCannabinoid receptor 2(Homo sapiens (Human))
Imir K.U. Leuven

Curated by ChEMBL
LigandPNGBDBM50349311(CHEMBL1807841)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells after 1 hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Imir K.U. Leuven

Curated by ChEMBL
LigandPNGBDBM50349311(CHEMBL1807841)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]-SR141716A from human CB1 receptor expressed in CHO cells after 1 hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399718(CHEMBL2178958)
Affinity DataIC50:  3nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM482157(BDBM50379529 | LRRK2-IN-1 | US11370796, Compound L...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of recombinant LRRK2 (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50155838((S)-1-((S)-1-(4-phenylbutanoyl)pyrrolidine-2-carbo...)
Affinity DataIC50:  6nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399717(CHEMBL2178959)
Affinity DataIC50:  9nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50026589(CHEMBL2206014)
Affinity DataIC50:  10nMAssay Description:Inhibition of recombinant LRRK2 G2019S mutant (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiog...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399730(CHEMBL2178967)
Affinity DataIC50:  14nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50026589(CHEMBL2206014)
Affinity DataIC50:  15nMAssay Description:Inhibition of recombinant LRRK2 (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399732(CHEMBL2178965)
Affinity DataIC50:  17.2nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399731(CHEMBL2178966)
Affinity DataIC50:  23nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399733(CHEMBL2178964)
Affinity DataIC50:  24nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399725(CHEMBL2178972)
Affinity DataIC50:  24nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  28nMAssay Description:Inhibition of human recombinant GSK3alpha using CFFKNIVTPRTPPPSQGK-amide substrate after 60 mins incubation by LANCE methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50026597(CHEMBL3335345)
Affinity DataIC50:  31nMAssay Description:Inhibition of recombinant LRRK2 (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399737(CHEMBL2178960)
Affinity DataIC50:  32nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399734(CHEMBL2178963)
Affinity DataIC50:  33nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399740(CHEMBL2179406)
Affinity DataIC50:  39nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50026584(CHEMBL3335349)
Affinity DataIC50:  46nMAssay Description:Inhibition of recombinant LRRK2 (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  50nMAssay Description:Inhibition of human recombinant GSK3beta using CFFKNIVTPRTPPPSQGK-amide substrate after 90 mins incubation by LANCE methodMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50026584(CHEMBL3335349)
Affinity DataIC50:  64nMAssay Description:Inhibition of recombinant LRRK2 G2019S mutant (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiog...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399728(CHEMBL2178969)
Affinity DataIC50:  69nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399745(CHEMBL2178976)
Affinity DataIC50:  90nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399722(CHEMBL2178975)
Affinity DataIC50:  100nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399723(CHEMBL2178974)
Affinity DataIC50:  110nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50051539((S)-4-phenyl-1-(2-(pyrrolidine-1-carbonyl)pyrrolid...)
Affinity DataIC50:  130nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399727(CHEMBL2178970)
Affinity DataIC50:  131nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399738(CHEMBL2179408)
Affinity DataIC50:  141nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399743(CHEMBL2178978)
Affinity DataIC50:  142nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399739(CHEMBL2179407)
Affinity DataIC50:  147nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50026591(CHEMBL3335330)
Affinity DataIC50:  163nMAssay Description:Inhibition of recombinant LRRK2 (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399735(CHEMBL2178962)
Affinity DataIC50:  170nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399726(CHEMBL2178971)
Affinity DataIC50:  170nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50026586(CHEMBL3335346)
Affinity DataIC50:  194nMAssay Description:Inhibition of recombinant LRRK2 (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50026596(CHEMBL3335344)
Affinity DataIC50:  204nMAssay Description:Inhibition of recombinant LRRK2 (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50026594(CHEMBL3335333)
Affinity DataIC50:  205nMAssay Description:Inhibition of recombinant LRRK2 (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399724(CHEMBL2178973)
Affinity DataIC50:  240nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50026588(CHEMBL3335328)
Affinity DataIC50:  261nMAssay Description:Inhibition of recombinant LRRK2 (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399719(CHEMBL2178957)
Affinity DataIC50:  280nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399721(CHEMBL2178955)
Affinity DataIC50:  304nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50316820((S)-benzyl 2-(pyrrolidine-1-carbonyl)pyrrolidine-1...)
Affinity DataIC50:  350nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399729(CHEMBL2178968)
Affinity DataIC50:  357nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399744(CHEMBL2178977)
Affinity DataIC50:  364nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50026592(CHEMBL3335331)
Affinity DataIC50:  466nMAssay Description:Inhibition of recombinant LRRK2 (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399736(CHEMBL2178961)
Affinity DataIC50:  478nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399720(CHEMBL2178956)
Affinity DataIC50:  542nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399741(CHEMBL2179405)
Affinity DataIC50:  956nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399742(CHEMBL2178979)
Affinity DataIC50:  1.16E+3nMAssay Description:Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50026585(CHEMBL3335348)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of recombinant LRRK2 (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50399731(CHEMBL2178966)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells assessed as pNA release from Ala-Pro-p-nitroanilide pre-incubated with enzyme for 15 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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