Affinity DataKi: 1.20nMAssay Description:Noncompetitive inhibition of human recombinant microsomal MAOB expressed in baculovirus infected BTI-TN-5B1- 4 cells using p-tyramine as substrate as...More data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Inhibition of human recombinant microsomal MAOB expressed in baculovirus infected BTI-TN-5B1- 4 cells using p-tyramine as substrate assessed as decre...More data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Competitive inhibition of recombinant human MAO-B using kynuramine as substrate pre-incubated for 15 mins followed by 2 fold compound dilution for 24...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Inhibition of recombinant human carbonic anhydrase 2 preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Porto
Curated by ChEMBL
University Of Porto
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Inhibition of electric eel AChE assessed as inhibition constant using acetylthiocholine iodide as substrate pretreated for 5 mins followed by substra...More data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Reversible competitive inhibition of human recombinant microsomal MAOA expressed in baculovirus infected BTI-TN-5B1- 4 cells using p-tyramine as subs...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Inhibition of recombinant human carbonic anhydrase VA preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
Affinity DataKi: 73nMAssay Description:Inhibition of recombinant human carbonic anhydrase VA preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
Affinity DataKi: 81nMAssay Description:Inhibition of recombinant human carbonic anhydrase VA preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
Affinity DataKi: 84nMAssay Description:Inhibition of recombinant human carbonic anhydrase VA preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
Affinity DataKi: 131nMAssay Description:Inhibition of recombinant human carbonic anhydrase VA preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
Affinity DataKi: 133nMAssay Description:Inhibition of recombinant human carbonic anhydrase VA preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 182nMAssay Description:Inhibition of equine BChE assessed as inhibition constant using acetylthiocholine as substrate measured for 0.5 to 1.5 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Mixed type inhibition of human AChE using acetylthiocholine iodide as substrate pretreated for 5 mins followed by substrate addition measured after 5...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
Affinity DataKi: 250nMAssay Description:Inhibition of recombinant human carbonic anhydrase 1 preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 258nMAssay Description:Inhibition of equine BChE assessed as inhibition constant using acetylthiocholine as substrate measured for 0.5 to 1.5 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataKi: 337nMAssay Description:Reversible competitive inhibition of human recombinant microsomal MAOB expressed in baculovirus infected BTI-TN-5B1- 4 cells using p-tyramine as subs...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
Affinity DataKi: 344nMAssay Description:Inhibition of recombinant human carbonic anhydrase VA preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 450nMAssay Description:Inhibition of equine BChE assessed as inhibition constant using acetylthiocholine as substrate measured for 0.5 to 1.5 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataKi: 478nMAssay Description:Reversible competitive inhibition of human recombinant microsomal MAOB expressed in baculovirus infected BTI-TN-5B1- 4 cells using p-tyramine as subs...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
Affinity DataKi: 539nMAssay Description:Inhibition of recombinant human carbonic anhydrase VA preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Porto
Curated by ChEMBL
University Of Porto
Curated by ChEMBL
Affinity DataKi: 788nMAssay Description:Inhibition of electric eel AChE assessed as inhibition constant using acetylthiocholine as substrate measured for 0.5 to 1.5 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataKi: 910nMAssay Description:Inhibition of equine BChE assessed as inhibition constant using acetylthiocholine as substrate measured for 0.5 to 1.5 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataKi: 920nMAssay Description:Inhibition of equine BChE assessed as inhibition constant using acetylthiocholine as substrate measured for 0.5 to 1.5 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
Affinity DataKi: 997nMAssay Description:Inhibition of recombinant human carbonic anhydrase VA preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.08E+3nMAssay Description:Inhibition of equine BChE assessed as inhibition constant using acetylthiocholine as substrate measured for 0.5 to 1.5 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
Affinity DataKi: 1.15E+3nMAssay Description:Inhibition of recombinant human carbonic anhydrase VA preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Porto
Curated by ChEMBL
University Of Porto
Curated by ChEMBL
Affinity DataKi: 1.34E+3nMAssay Description:Inhibition of electric eel AChE assessed as inhibition constant using acetylthiocholine as substrate measured for 0.5 to 1.5 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Porto
Curated by ChEMBL
University Of Porto
Curated by ChEMBL
Affinity DataKi: 1.37E+3nMAssay Description:Inhibition of electric eel AChE assessed as inhibition constant using acetylthiocholine as substrate measured for 0.5 to 1.5 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Inhibition of Equine serum BuChE assessed as inhibitory constants for binding the free enzyme using S-butyrylthiocholine iodide as a substrate by Cor...More data for this Ligand-Target Pair
Affinity DataKi: 2.36E+3nMAssay Description:Inhibition of equine BChE assessed as inhibition constant using acetylthiocholine as substrate measured for 0.5 to 1.5 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Porto
Curated by ChEMBL
University Of Porto
Curated by ChEMBL
Affinity DataKi: 2.79E+3nMAssay Description:Inhibition of electric eel AChE assessed as inhibition constant using acetylthiocholine as substrate measured for 0.5 to 1.5 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Porto
Curated by ChEMBL
University Of Porto
Curated by ChEMBL
Affinity DataKi: 5.20E+3nMAssay Description:Inhibition of electric eel AChE assessed as inhibition constant using acetylthiocholine iodide as substrate pretreated for 5 mins followed by substra...More data for this Ligand-Target Pair
Affinity DataKi: 6.70E+3nMAssay Description:Inhibition of Equine serum BuChE assessed as inhibitory constants for binding the enzyme-substrate complex using S-butyrylthiocholine iodide as a sub...More data for this Ligand-Target Pair
Affinity DataKi: 7.20E+3nMAssay Description:Inhibition of Equine serum BuChE assessed as inhibitory constants for binding the free enzyme using S-butyrylthiocholine iodide as a substrate by Cor...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
Affinity DataKi: 8.71E+3nMAssay Description:Inhibition of recombinant human carbonic anhydrase VA preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 9.00E+3nMAssay Description:Inhibition of Equine serum BuChE assessed as inhibitory constants for binding the free enzyme using S-butyrylthiocholine iodide as a substrate by Cor...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
Affinity DataKi: 9.76E+3nMAssay Description:Inhibition of recombinant human carbonic anhydrase VA preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of recombinant human carbonic anhydrase 1 preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of recombinant human carbonic anhydrase 1 preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of recombinant human carbonic anhydrase 2 preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of recombinant human carbonic anhydrase 1 preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of recombinant human carbonic anhydrase 1 preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of recombinant human carbonic anhydrase 1 preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of recombinant human carbonic anhydrase 1 preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of recombinant human carbonic anhydrase 1 preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of recombinant human carbonic anhydrase 1 preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of recombinant human carbonic anhydrase 2 preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of recombinant human carbonic anhydrase 2 preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
"Magna Gr£Cia" University Of Catanzaro
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of recombinant human carbonic anhydrase 2 preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair