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Found 546 with Last Name = 'baker' and Initial = 'e'
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379086(CHEMBL2012521 | CHEMBL2012522 | LY-377604)
Affinity DataKi:  0.0120nMAssay Description:Displacement of [125I]Iodocyanopindolol from human adrenergic beta2 receptor expressed in insect sf9 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379086(CHEMBL2012521 | CHEMBL2012522 | LY-377604)
Affinity DataKi:  0.0230nMAssay Description:Displacement of [125I]Iodocyanopindolol from human adrenergic beta1 receptor expressed in insect sf9 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50544441(CHEMBL4637373 | US11192850, Entry 4u)
Affinity DataKi:  1.20nMAssay Description:Competitive inhibition of Mycobacterium tuberculosis PTPB expressed in Escherichia coli BL21 (DE3) using varying levels of p-nitrophenyl phosphate as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50544440(CHEMBL4647367 | US11192850, Entry 4t)
Affinity DataKi:  2.70nMAssay Description:Competitive inhibition of Mycobacterium tuberculosis PTPB expressed in Escherichia coli BL21 (DE3) using varying levels of p-nitrophenyl phosphate as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50544442(CHEMBL4638011 | US11192850, Entry 4v)
Affinity DataKi:  4.90nMAssay Description:Competitive inhibition of Mycobacterium tuberculosis PTPB expressed in Escherichia coli BL21 (DE3) using varying levels of p-nitrophenyl phosphate as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073296(4-((S)-1-Hydroxymethyl-2-phenyl-ethylamino)-pyridi...)
Affinity DataKi:  12nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073308(4-[(R)-2-(4-Methoxy-phenyl)-1-methyl-ethylamino]-p...)
Affinity DataKi:  15nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073307(4-((R)-1-Methyl-2-phenyl-ethylamino)-pyridine-3-su...)
Affinity DataKi:  18nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073302(4-((S)-2-Cyclohexyl-1-hydroxymethyl-ethylamino)-py...)
Affinity DataKi:  18nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073297(4-[(S)-1-(4-Hydroxy-piperidin-1-ylmethyl)-2-phenyl...)
Affinity DataKi:  19nMAssay Description:In vitro inhibtion of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073283(4-[(S)-1-Hydroxymethyl-2-(4-methoxy-phenyl)-ethyla...)
Affinity DataKi:  19nMAssay Description:In vitro inhibtion of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073283(4-[(S)-1-Hydroxymethyl-2-(4-methoxy-phenyl)-ethyla...)
Affinity DataKi:  19nMAssay Description:In vitro inhibtion of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073290(4-{(S)-1-Benzyl-2-[bis-(2-methoxy-ethyl)-amino]-et...)
Affinity DataKi:  19nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073283(4-[(S)-1-Hydroxymethyl-2-(4-methoxy-phenyl)-ethyla...)
Affinity DataKi:  19nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073297(4-[(S)-1-(4-Hydroxy-piperidin-1-ylmethyl)-2-phenyl...)
Affinity DataKi:  19nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073298(4-((S)-1-Benzyl-2-morpholin-4-yl-ethylamino)-pyrid...)
Affinity DataKi:  22nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073298(4-((S)-1-Benzyl-2-morpholin-4-yl-ethylamino)-pyrid...)
Affinity DataKi:  22nMAssay Description:In vitro inhibtion of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073298(4-((S)-1-Benzyl-2-morpholin-4-yl-ethylamino)-pyrid...)
Affinity DataKi:  22nMAssay Description:In vitro inhibtion of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073287(4-[(S)-2-(4-Acetyl-piperazin-1-yl)-1-benzyl-ethyla...)
Affinity DataKi:  24nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073294(4-((S)-1-Benzyl-2-dimethylamino-ethylamino)-pyridi...)
Affinity DataKi:  24nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073294(4-((S)-1-Benzyl-2-dimethylamino-ethylamino)-pyridi...)
Affinity DataKi:  24nMAssay Description:In vitro inhibtion of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073305(4-((S)-1-Benzyl-2-piperidin-1-yl-ethylamino)-pyrid...)
Affinity DataKi:  25nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073306(4-((S)-1-Hydroxymethyl-2-phenyl-ethylamino)-pyridi...)
Affinity DataKi:  27nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50075870(4-[(S)-1-(2-Hydroxy-ethoxymethyl)-2-phenyl-ethylam...)
Affinity DataKi:  28nMAssay Description:In vitro inhibtion of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073299(4-((S)-2-Cyclohexyl-1-methylaminomethyl-ethylamino...)
Affinity DataKi:  33nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073288(4-((S)-1-Methylaminomethyl-2-phenyl-ethylamino)-py...)
Affinity DataKi:  35nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073304(4-((S)-1-Hydroxymethyl-2-phenyl-ethylamino)-pyridi...)
Affinity DataKi:  36nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073295(4-((S)-1-Hydroxymethyl-2-phenyl-ethylamino)-pyridi...)
Affinity DataKi:  39nMAssay Description:In vitro inhibtion of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073295(4-((S)-1-Hydroxymethyl-2-phenyl-ethylamino)-pyridi...)
Affinity DataKi:  39nMAssay Description:In vitro inhibtion of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073295(4-((S)-1-Hydroxymethyl-2-phenyl-ethylamino)-pyridi...)
Affinity DataKi:  39nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50075873(4-[(S)-1-Hydroxymethyl-2-(4-methoxy-phenyl)-ethyla...)
Affinity DataKi:  40nMAssay Description:In vitro inhibtion of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073293(4-((S)-1-Hydroxymethyl-2-phenyl-ethylamino)-pyridi...)
Affinity DataKi:  41nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073286(4-((S)-1-Butylaminomethyl-2-phenyl-ethylamino)-pyr...)
Affinity DataKi:  43nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073309(4-((S)-1-Benzyl-2-diethylamino-ethylamino)-pyridin...)
Affinity DataKi:  45nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073303(4-((S)-2-Phenyl-1-propylaminomethyl-ethylamino)-py...)
Affinity DataKi:  47nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073300(4-((S)-1-Benzyl-2-pyrrolidin-1-yl-ethylamino)-pyri...)
Affinity DataKi:  48nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073292(4-[(S)-1-(2-Hydroxy-ethoxymethyl)-2-phenyl-ethylam...)
Affinity DataKi:  49nMAssay Description:In vitro inhibtion of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073292(4-[(S)-1-(2-Hydroxy-ethoxymethyl)-2-phenyl-ethylam...)
Affinity DataKi:  49nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073285(4-[(S)-2-(3,4-Dimethoxy-phenyl)-1-hydroxymethyl-et...)
Affinity DataKi:  49nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073292(4-[(S)-1-(2-Hydroxy-ethoxymethyl)-2-phenyl-ethylam...)
Affinity DataKi:  49nMAssay Description:In vitro inhibtion of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50075871(4-[(S)-1-(4-Hydroxy-piperidin-1-ylmethyl)-2-phenyl...)
Affinity DataKi:  61nMAssay Description:In vitro inhibtion of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50075868(4-((S)-1-Morpholin-4-ylmethyl-2-phenyl-ethylamino)...)
Affinity DataKi:  62nMAssay Description:In vitro inhibtion of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073282(4-((S)-1-Hydroxymethyl-2-phenyl-ethylamino)-pyridi...)
Affinity DataKi:  65nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073291(4-{(S)-1-[(2-Hydroxy-ethylamino)-methyl]-2-phenyl-...)
Affinity DataKi:  72nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50075874(4-[(S)-1-Hydroxymethyl-2-(4-methoxy-phenyl)-ethyla...)
Affinity DataKi:  85nMAssay Description:In vitro inhibtion of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073284(4-[(S)-1-Benzyl-2-(3-oxo-piperazin-1-yl)-ethylamin...)
Affinity DataKi:  90nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073289(4-((S)-1-Ethylaminomethyl-2-phenyl-ethylamino)-pyr...)
Affinity DataKi:  99nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073301(4-((S)-1-Hydroxymethyl-2-phenyl-ethylamino)-pyridi...)
Affinity DataKi:  100nMAssay Description:In vitro inhibtion of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073301(4-((S)-1-Hydroxymethyl-2-phenyl-ethylamino)-pyridi...)
Affinity DataKi:  100nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Novartis Horsham Research Center

Curated by ChEMBL
LigandPNGBDBM50073281(4-((S)-1-Hydroxymethyl-2-phenyl-ethylamino)-pyridi...)
Affinity DataKi:  110nMAssay Description:In vitro binding affinity for human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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