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Found 36 with Last Name = 'bakr' and Initial = 'rb'
TargetAurora kinase A(Homo sapiens (Human))
Jouf University

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human Aurora A using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jouf University

Curated by ChEMBL
LigandPNGBDBM50004231(CHEMBL3237167)
Affinity DataIC50:  5nMAssay Description:Inhibition of AURKA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Jouf University

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human Aurora B using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543797(CHEMBL4637300)
Affinity DataIC50:  90nMAssay Description:Inhibition of human Aurora B using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jouf University

Curated by ChEMBL
LigandPNGBDBM14210(4-(4-(N-benzoylamino)anilino)-6-methoxy-7-(3-(1-mo...)
Affinity DataIC50:  110nMAssay Description:Inhibition of AURKA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Jouf University

Curated by ChEMBL
LigandPNGBDBM14210(4-(4-(N-benzoylamino)anilino)-6-methoxy-7-(3-(1-mo...)
Affinity DataIC50:  130nMAssay Description:Inhibition of AURKB (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543797(CHEMBL4637300)
Affinity DataIC50:  930nMAssay Description:Inhibition of human Aurora A using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543800(CHEMBL4645713)
Affinity DataIC50:  980nMAssay Description:Inhibition of human Aurora A using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543799(CHEMBL4640153)
Affinity DataIC50:  1.35E+3nMAssay Description:Inhibition of human Aurora B using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543801(CHEMBL4648901)
Affinity DataIC50:  1.62E+3nMAssay Description:Inhibition of human Aurora B using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543799(CHEMBL4640153)
Affinity DataIC50:  1.77E+3nMAssay Description:Inhibition of human Aurora A using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543800(CHEMBL4645713)
Affinity DataIC50:  2.99E+3nMAssay Description:Inhibition of human Aurora B using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181101(N-(3,4,5-trimethoxybenzylidene)-2-(3,6-dimethyl-1-...)
Affinity DataIC50:  4.18E+3nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181097(N-(4-methoxybenzylidene)-2-(3,6-dimethyl-1-phenyl-...)
Affinity DataIC50:  4.72E+3nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181098(N-(4-chlorobenzylidene)-2-(3,6-dimethyl-1-phenyl-1...)
Affinity DataIC50:  5.01E+3nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543796(CHEMBL4635411)
Affinity DataIC50:  6.89E+3nMAssay Description:Inhibition of human Aurora B using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543796(CHEMBL4635411)
Affinity DataIC50:  7.64E+3nMAssay Description:Inhibition of human Aurora A using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181101(N-(3,4,5-trimethoxybenzylidene)-2-(3,6-dimethyl-1-...)
Affinity DataIC50:  8.20E+3nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543802(CHEMBL4644959)
Affinity DataIC50:  8.33E+3nMAssay Description:Inhibition of human Aurora B using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181101(N-(3,4,5-trimethoxybenzylidene)-2-(3,6-dimethyl-1-...)
Affinity DataIC50:  8.37E+3nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181098(N-(4-chlorobenzylidene)-2-(3,6-dimethyl-1-phenyl-1...)
Affinity DataIC50:  9.59E+3nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181097(N-(4-methoxybenzylidene)-2-(3,6-dimethyl-1-phenyl-...)
Affinity DataIC50:  1.01E+4nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181095(N-(4-Hydroxybenzylidene)-2-(3,6-dimethyl-1-phenyl-...)
Affinity DataIC50:  1.05E+4nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181099(N-(4-chlorobenzylidene)-2-(3,6-dimethyl-1-phenyl-1...)
Affinity DataIC50:  1.15E+4nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543803(CHEMBL4639147)
Affinity DataIC50:  1.15E+4nMAssay Description:Inhibition of human Aurora B using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181101(N-(3,4,5-trimethoxybenzylidene)-2-(3,6-dimethyl-1-...)
Affinity DataIC50:  1.20E+4nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543795(CHEMBL4645551)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibition of human Aurora B using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181097(N-(4-methoxybenzylidene)-2-(3,6-dimethyl-1-phenyl-...)
Affinity DataIC50:  1.26E+4nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181097(N-(4-methoxybenzylidene)-2-(3,6-dimethyl-1-phenyl-...)
Affinity DataIC50:  1.29E+4nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181098(N-(4-chlorobenzylidene)-2-(3,6-dimethyl-1-phenyl-1...)
Affinity DataIC50:  1.29E+4nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543798(CHEMBL4641064)
Affinity DataIC50:  1.32E+4nMAssay Description:Inhibition of human Aurora B using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543798(CHEMBL4641064)
Affinity DataIC50:  1.34E+4nMAssay Description:Inhibition of human Aurora A using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543795(CHEMBL4645551)
Affinity DataIC50:  1.66E+4nMAssay Description:Inhibition of human Aurora A using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181098(N-(4-chlorobenzylidene)-2-(3,6-dimethyl-1-phenyl-1...)
Affinity DataIC50:  1.76E+4nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181096(N-(4-fluorobenzylidene)-2-(3,6-dimethyl-1-phenyl-1...)
Affinity DataIC50:  3.00E+4nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Beni-Suef University

LigandPNGBDBM181100(N-(4-Trifluoromethylbenzylidene)-2-(3,6-dimethyl-1...)
Affinity DataIC50:  3.59E+4nMAssay Description:Kinase activity was determined using Kinase-Glo Plus luminescence kinase assay kit according to the manufacturer instructions. The assays depend on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed