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Found 50 with Last Name = 'bangalore' and Initial = 'pk'
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123830(4,5-dibromo-N'-(4-chlorobenzylidene)-1-methyl-...)
Affinity DataKi:  2.10E+3nM ΔG°:  -33.7kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123825(4,5-dibromo-N'-[(4-fluorophenyl)methylidene]-1...)
Affinity DataKi:  2.40E+3nM ΔG°:  -33.4kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123833(4,5-dibromo-N'-(2,4-dichlorobenzylidene)-1-met...)
Affinity DataKi:  2.60E+3nM ΔG°:  -33.2kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123832(4,5-dibromo-N'-(4-methoxybenzylidene)-1-methyl...)
Affinity DataKi:  2.90E+3nM ΔG°:  -32.9kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123823(4,5-dibromo-N'-[(2,4-dichlorophenyl)methyliden...)
Affinity DataKi:  3.10E+3nM ΔG°:  -32.7kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123831(4,5-dibromo-N'-(3,4-dimethoxybenzylidene)-1-me...)
Affinity DataKi:  3.40E+3nM ΔG°:  -32.5kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123820(4,5-dibromo-N'-[(4-chlorophenyl)methylidene]-1...)
Affinity DataKi:  3.90E+3nM ΔG°:  -32.1kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123828(4,5-dibromo-N'-(2,6-dichlorobenzylidene)-1-met...)
Affinity DataKi:  3.90E+3nM ΔG°:  -32.1kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123824(4,5-dibromo-N'-(2-hydroxybenzylidene)-1-methyl...)
Affinity DataKi:  4.70E+3nM ΔG°:  -31.6kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123815(4,5-dibromo-N'-(4-fluorobenzylidene)-1H-pyrrol...)
Affinity DataKi:  5.10E+3nM ΔG°:  -31.4kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123818(4,5-dibromo-N'-(2,6-dichlorobenzylidene)-1Hpyr...)
Affinity DataKi:  5.20E+3nM ΔG°:  -31.4kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123829(4,5-dibromo-N'-(3,4-dihydroxybenzylidene)-1-me...)
Affinity DataKi:  6.10E+3nM ΔG°:  -31.0kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123822(4,5-dibromo-N'-(4-methoxybenzylidene)-1Hpyrrol...)
Affinity DataKi:  6.55E+3nM ΔG°:  -30.8kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123826(4,5-dibromo-1-methyl-N'-(4-nitrobenzylidene)-1...)
Affinity DataKi:  6.90E+3nM ΔG°:  -30.6kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123827(4,5-dibromo-N'-(4-hydroxybenzylidene)-1-methyl...)
Affinity DataKi:  7.10E+3nM ΔG°:  -30.6kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123814(4,5-dibromo-N'-(2-hydroxybenzylidene)-1H-pyrro...)
Affinity DataKi:  8.90E+3nM ΔG°:  -30.0kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123823(4,5-dibromo-N'-[(2,4-dichlorophenyl)methyliden...)
Affinity DataKi:  9.40E+3nM ΔG°:  -29.8kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123821(4,5-dibromo-N'-(3,4-dimethoxybenzylidene)-1Hpy...)
Affinity DataKi:  1.13E+4nM ΔG°:  -29.4kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123828(4,5-dibromo-N'-(2,6-dichlorobenzylidene)-1-met...)
Affinity DataKi:  1.23E+4nM ΔG°:  -29.2kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123820(4,5-dibromo-N'-[(4-chlorophenyl)methylidene]-1...)
Affinity DataKi:  1.25E+4nM ΔG°:  -29.1kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123833(4,5-dibromo-N'-(2,4-dichlorobenzylidene)-1-met...)
Affinity DataKi:  1.29E+4nM ΔG°:  -29.0kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123827(4,5-dibromo-N'-(4-hydroxybenzylidene)-1-methyl...)
Affinity DataKi:  1.33E+4nM ΔG°:  -29.0kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123832(4,5-dibromo-N'-(4-methoxybenzylidene)-1-methyl...)
Affinity DataKi:  1.38E+4nM ΔG°:  -28.9kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123816(4,5-dibromo-N'-(4-nitrobenzylidene)-1H-pyrrole...)
Affinity DataKi:  1.44E+4nM ΔG°:  -28.7kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123817(4,5-dibromo-N'-(4-hydroxybenzylidene)-1H-pyrro...)
Affinity DataKi:  1.59E+4nM ΔG°:  -28.5kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123819(4,5-dibromo-N'-(3,4-dihydroxybenzylidene)-1Hpy...)
Affinity DataKi:  1.73E+4nM ΔG°:  -28.3kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123829(4,5-dibromo-N'-(3,4-dihydroxybenzylidene)-1-me...)
Affinity DataKi:  2.04E+4nM ΔG°:  -27.8kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123818(4,5-dibromo-N'-(2,6-dichlorobenzylidene)-1Hpyr...)
Affinity DataKi:  2.05E+4nM ΔG°:  -27.8kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123822(4,5-dibromo-N'-(4-methoxybenzylidene)-1Hpyrrol...)
Affinity DataKi:  2.12E+4nM ΔG°:  -27.7kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123831(4,5-dibromo-N'-(3,4-dimethoxybenzylidene)-1-me...)
Affinity DataKi:  2.17E+4nM ΔG°:  -27.7kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123824(4,5-dibromo-N'-(2-hydroxybenzylidene)-1-methyl...)
Affinity DataKi:  2.28E+4nM ΔG°:  -27.6kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123815(4,5-dibromo-N'-(4-fluorobenzylidene)-1H-pyrrol...)
Affinity DataKi:  2.45E+4nM ΔG°:  -27.4kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123821(4,5-dibromo-N'-(3,4-dimethoxybenzylidene)-1Hpy...)
Affinity DataKi:  2.61E+4nM ΔG°:  -27.2kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123830(4,5-dibromo-N'-(4-chlorobenzylidene)-1-methyl-...)
Affinity DataKi:  2.69E+4nM ΔG°:  -27.1kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123814(4,5-dibromo-N'-(2-hydroxybenzylidene)-1H-pyrro...)
Affinity DataKi:  3.78E+4nM ΔG°:  -26.3kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123825(4,5-dibromo-N'-[(4-fluorophenyl)methylidene]-1...)
Affinity DataKi:  3.81E+4nM ΔG°:  -26.2kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123826(4,5-dibromo-1-methyl-N'-(4-nitrobenzylidene)-1...)
Affinity DataKi:  4.05E+4nM ΔG°:  -26.1kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123817(4,5-dibromo-N'-(4-hydroxybenzylidene)-1H-pyrro...)
Affinity DataKi:  4.26E+4nM ΔG°:  -26.0kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123819(4,5-dibromo-N'-(3,4-dihydroxybenzylidene)-1Hpy...)
Affinity DataKi:  4.48E+4nM ΔG°:  -25.8kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of Kwazulu-Natal

LigandPNGBDBM123816(4,5-dibromo-N'-(4-nitrobenzylidene)-1H-pyrrole...)
Affinity DataKi:  6.63E+4nM ΔG°:  -24.8kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University of Kwazulu-Nata

LigandPNGBDBM153386(2-(4,5-Dibromo-1H-pyrrole-2-carbonyl)-N-(4-chlorop...)
Affinity DataIC50:  1.80E+3nMpH: 8.5 T: 2°CAssay Description:The synthesized compounds were assayed for the inhibitory activities against MMP-2 in 96-well microtiter plates using succinylated gelatin as the sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University of Kwazulu-Nata

LigandPNGBDBM153388(2-(1-Methyl-4,5-dibromo-1H-pyrrole-2-carbonyl)-N-(...)
Affinity DataIC50:  8.00E+3nMpH: 8.5 T: 2°CAssay Description:The synthesized compounds were assayed for the inhibitory activities against MMP-2 in 96-well microtiter plates using succinylated gelatin as the sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University of Kwazulu-Nata

LigandPNGBDBM153385(2-(4,5-Dibromo-1H-pyrrole-2-carbonyl)-N-(4-nitroph...)
Affinity DataIC50:  1.37E+4nMpH: 8.5 T: 2°CAssay Description:The synthesized compounds were assayed for the inhibitory activities against MMP-2 in 96-well microtiter plates using succinylated gelatin as the sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University of Kwazulu-Nata

LigandPNGBDBM153387(2-(1-Methyl-4,5-dibromo-1H-pyrrole-2-carbonyl)-N-(...)
Affinity DataIC50:  1.92E+4nMpH: 8.5 T: 2°CAssay Description:The synthesized compounds were assayed for the inhibitory activities against MMP-2 in 96-well microtiter plates using succinylated gelatin as the sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Kwazulu-Nata

LigandPNGBDBM153387(2-(1-Methyl-4,5-dibromo-1H-pyrrole-2-carbonyl)-N-(...)
Affinity DataIC50:  2.38E+4nMpH: 8.0 T: 2°CAssay Description:The synthesized compounds were assayed for the inhibitory activities against MMP-12 in 96-well microtiter plates using thiopeptolide as the substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Kwazulu-Nata

LigandPNGBDBM153386(2-(4,5-Dibromo-1H-pyrrole-2-carbonyl)-N-(4-chlorop...)
Affinity DataIC50:  2.90E+4nMpH: 8.0 T: 2°CAssay Description:The synthesized compounds were assayed for the inhibitory activities against MMP-12 in 96-well microtiter plates using thiopeptolide as the substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Kwazulu-Nata

LigandPNGBDBM153385(2-(4,5-Dibromo-1H-pyrrole-2-carbonyl)-N-(4-nitroph...)
Affinity DataIC50:  4.21E+4nMpH: 8.0 T: 2°CAssay Description:The synthesized compounds were assayed for the inhibitory activities against MMP-12 in 96-well microtiter plates using thiopeptolide as the substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Kwazulu-Nata

LigandPNGBDBM153388(2-(1-Methyl-4,5-dibromo-1H-pyrrole-2-carbonyl)-N-(...)
Affinity DataIC50:  4.31E+4nMpH: 8.0 T: 2°CAssay Description:The synthesized compounds were assayed for the inhibitory activities against MMP-12 in 96-well microtiter plates using thiopeptolide as the substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University of Kwazulu-Nata

LigandPNGBDBM153389(2-(1-Methyl-4,5-dibromo-1H-pyrrole-2-carbonyl-N-(f...)
Affinity DataIC50:  6.03E+4nMpH: 8.5 T: 2°CAssay Description:The synthesized compounds were assayed for the inhibitory activities against MMP-2 in 96-well microtiter plates using succinylated gelatin as the sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Kwazulu-Nata

LigandPNGBDBM153389(2-(1-Methyl-4,5-dibromo-1H-pyrrole-2-carbonyl-N-(f...)
Affinity DataIC50:  8.42E+4nMpH: 8.0 T: 2°CAssay Description:The synthesized compounds were assayed for the inhibitory activities against MMP-12 in 96-well microtiter plates using thiopeptolide as the substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed