Affinity DataKi: 1nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Inhibition of carbonic anhydrase 9 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 4.70nMAssay Description:Inhibition of carbonic anhydrase 9 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 7.70nMAssay Description:Inhibition of carbonic anhydrase 9 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 9.20nMAssay Description:Inhibition of carbonic anhydrase 9 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Inhibition of cytosolic carbonic anhydrase 2 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Inhibition of carbonic anhydrase 9 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Inhibition of carbonic anhydrase 9 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Inhibition of carbonic anhydrase 9 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Inhibition of carbonic anhydrase 9 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 28nMAssay Description:Inhibition of cytosolic carbonic anhydrase 2 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Inhibition of cytosolic carbonic anhydrase 2 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Inhibition of cytosolic carbonic anhydrase 2 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 35nMAssay Description:Inhibition of cytosolic carbonic anhydrase 2 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Inhibition of carbonic anhydrase 9 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 39nMAssay Description:Inhibition of cytosolic carbonic anhydrase 2 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 43nMAssay Description:Inhibition of cytosolic carbonic anhydrase 2 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 44nMAssay Description:Inhibition of carbonic anhydrase 9 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 45nMAssay Description:Inhibition of cytosolic carbonic anhydrase 2 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 53nMAssay Description:Inhibition of carbonic anhydrase 9 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 57nMAssay Description:Inhibition of cytosolic carbonic anhydrase 2 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 112nMAssay Description:Inhibition of cytosolic carbonic anhydrase 1 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 122nMAssay Description:Inhibition of cytosolic carbonic anhydrase 2 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 136nMAssay Description:Inhibition of cytosolic carbonic anhydrase 2 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 252nMAssay Description:Inhibition of cytosolic carbonic anhydrase 1 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 737nMAssay Description:Inhibition of cytosolic carbonic anhydrase 1 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 742nMAssay Description:Inhibition of cytosolic carbonic anhydrase 1 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 838nMAssay Description:Inhibition of cytosolic carbonic anhydrase 1 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 936nMAssay Description:Inhibition of cytosolic carbonic anhydrase 1 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 1.04E+3nMAssay Description:Inhibition of cytosolic carbonic anhydrase 1 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 1.11E+3nMAssay Description:Inhibition of cytosolic carbonic anhydrase 1 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 1.24E+3nMAssay Description:Inhibition of cytosolic carbonic anhydrase 1 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 1.25E+3nMAssay Description:Inhibition of cytosolic carbonic anhydrase 1 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 1.65E+3nMAssay Description:Inhibition of cytosolic carbonic anhydrase 1 (unknown origin) preincubated for 15 mins by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity to human integrin alphavbeta3 receptor by TRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Antagonist activity at human CCR1 in THP1 cells assessed as inhibition of MIP-1alpha-induced chemotaxis after 3 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Binding affinity to human integrin alphavbeta3 receptor by TRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Inhibitory activity against human renin inhibition (at pH 7.4)More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Manipal College Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 3.70nMAssay Description:Inhibition of MAO-A in bovine brain mitochondria using serotonin as substrate preincubated for 30 mins measured after 30 mins by spectrofluorimetric ...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Binding affinity to human integrin alphavbeta5 receptor by TRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.5nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Antagonist activity at human CCR1 in THP1 cells assessed as inhibition of MIP-1alpha-induced chemotaxis after 3 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Binding affinity to human integrin alphavbeta3 receptor by TRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.60nMAssay Description:Inhibition of human plasma ACEMore data for this Ligand-Target Pair
Affinity DataIC50: 9.60nMAssay Description:Inhibition of Wistar rat plasma ACEMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair